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公开(公告)号:US20100029678A1
公开(公告)日:2010-02-04
申请号:US12509698
申请日:2009-07-27
申请人: Amjad ALI , Iyassu K. Sebhat , Cristopher L. Franklin , Kathleen M. Rupprecht , Robert K. Baker , Ravi P. Nargund , Lin Yan , Pei Huo , Dong-Ming Shen , Nicoletta Almirante , Stefano Biondi , Massimiliano Ferrario , Alessia Nicotra
发明人: Amjad ALI , Iyassu K. Sebhat , Cristopher L. Franklin , Kathleen M. Rupprecht , Robert K. Baker , Ravi P. Nargund , Lin Yan , Pei Huo , Dong-Ming Shen , Nicoletta Almirante , Stefano Biondi , Massimiliano Ferrario , Alessia Nicotra
IPC分类号: A61K31/496 , C07D491/02 , A61K31/4355 , C07D241/04 , A61P9/12
CPC分类号: C07D491/04 , C07D519/00
摘要: A compound having the structure wherein X is selected from the group consisting of: a bond, —NHCH2(CH2)nCH2OC(O)—, —CH2NHC(O)CH2NHC(O)—, —CH2OC(O)—, —OCH(CH3)OC(O)—, —OCH2OC(O)—, —O—, —NR1—, —CR1R3—, —(CH2)p—, —(CH2)qNR1C(O)—, —CHR5NR2C(O)—, —(CH2)qC(O)—, —(CH2)qC(O)—, —(CH2)qC(O)NR1—, or a pharmaceutically acceptable salt thereof, and methods of using the compounds for treating, hypertension.
摘要翻译: 具有结构的化合物,其中X选自:-NHCH 2(CH 2)n CH 2 OC(O) - , - CH 2 NHC(O)CH 2 NHC(O) - , - CH 2 OC(O) - , - OCH CH 3)OC(O) - , - OCH 2 OC(O) - , - O - , - NR 1 - ,CR 1 R 3 - , - (CH 2)p - , - (CH 2)q NR1C , - (CH2)qC(O) - , - (CH2)qC(O) - , - (CH2)qC(O)NR1-或其药学上可接受的盐,以及使用该化合物治疗高血压的方法。