2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi
    3.
    发明授权
    2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi 失效
    2-(吡啶-2-基) - 嘧啶及其用于控制​​有害真菌的用途

    公开(公告)号:US07786043B2

    公开(公告)日:2010-08-31

    申请号:US11632342

    申请日:2005-07-22

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

    摘要翻译: 本发明涉及通式(I)的2-(吡啶-2-基) - 嘧啶化合物及其用于控制​​致病真菌的用途,作为作为活性成分的植物保护产品含有这种化合物:通式 (I)中,k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素,OH,CN,NO 2,C 1 -C 4烷基,C 1 -C 4烷基卤,C 1 -C 4烷氧基,C 1 -C 4烷氧基卤化物,C 2 -C 4烯基,C 2 -C 4炔基, C8环烷基,C1-C4烷氧基-C1-C4烷基,氨基,苯氧基,其任选被卤素或C 1 -C 4烷基取代,NHR,NR 2,C(R a)= N-OR b,S(= O)p A1或C (ΟO)A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-,其中Alk表示直链或支链C 1 -C 4亚烷基,和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤,C1-C4烷氧基,C1-C4烷氧基卤化物,羟基,卤素,CN或NO2; 其中当满足以下三个条件中的至少一个时,R2还可以表示氢或C1-C4烷基:n表示3,4或5; k表示1,2或3; 如果m不等于0,则基团R1中的至少一个表示与卤素,C 1 -C 4烷基,C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团, R3表示C1-C4烷基。

    2-(Pyridin-2-yl)-pyrimidines and Their Use for Controlling Harmful Fungi
    4.
    发明申请
    2-(Pyridin-2-yl)-pyrimidines and Their Use for Controlling Harmful Fungi 审中-公开
    2-(吡啶-2-基) - 嘧啶及其用于控制​​有害真菌的用途

    公开(公告)号:US20100286175A1

    公开(公告)日:2010-11-11

    申请号:US12840392

    申请日:2010-07-21

    IPC分类号: A01N43/54 C07D401/04 A01P3/00

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

    摘要翻译: 本发明涉及通式(I)的2-(吡啶-2-基) - 嘧啶化合物及其用于控制​​致病真菌的用途,作为作为活性成分的植物保护产品含有这种化合物:通式 (I)中,k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素,OH,CN,NO 2,C 1 -C 4烷基,C 1 -C 4烷基卤,C 1 -C 4烷氧基,C 1 -C 4烷氧基卤化物,C 2 -C 4烯基,C 2 -C 4炔基, C8环烷基,C1-C4烷氧基-C1-C4烷基,氨基,苯氧基,其任选被卤素或C 1 -C 4烷基取代,NHR,NR 2,C(R a)= N-OR b,S(= O)p A1或C (ΟO)A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-,其中Alk表示直链或支链C 1 -C 4亚烷基,和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤,C1-C4烷氧基,C1-C4烷氧基卤化物,羟基,卤素,CN或NO2; 其中当满足以下三个条件中的至少一个时,R2还可以表示氢或C1-C4烷基:n表示3,4或5; k表示1,2或3; 如果m不等于0,则基团R1中的至少一个表示与卤素,C 1 -C 4烷基,C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团, R3表示C1-C4烷基。

    2-substituted pyrimidines
    9.
    发明授权
    2-substituted pyrimidines 失效
    2-取代的嘧啶

    公开(公告)号:US07488732B2

    公开(公告)日:2009-02-10

    申请号:US10549936

    申请日:2004-03-30

    摘要: 2-Substituted pyrimidines of the formula I in which the index n and the substituents L, Ra, Rb, Rc, Rz, Ru, Rv, A′, A″ and A′″ are as defined in the description and: R1 is C3-C10-alkyl, C3-C10-alkenyl, C3-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S, R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl, and R3 is cyano, CO2Ra, C(═O)NRzRb, C(═O)—N—ORb, C(═S)—NRaRb, C(═NORa)NRzRb, C(═NRa)NRzRb, C(═O)NRa—NRzRb, C(═N—NRzRc)NRaRb, C(═O)Ra, C(═NORb)Ra, C(═N—NRzRb)Ra, CRaRb—ORz, CRaRb—NRzRc, ON(═CRaRb), O—C(═O)Ra, NRaRb′, NRa(C(═O)Rb), NRa(C(═O)ORb), NRa(C(═O)—NRzRb), NRa(C(═NRc)Rb), NRa(N═CRcRb), NRa—NRzRb, NRz—ORa, NRa(C(═NRc)—NRzRb), NRa(C(═NORc)Rb), processes for preparing these compounds, compositions comprising these compounds and their pesticidal use are described.

    摘要翻译: 其中指数n和取代基L,Ra,Rb,Rc,Rz,Ru,Rv,A',A“和A”'如说明书中所定义的式I的2-取代的嘧啶:R1 C 3 -C 10 - 烷基,C 3 -C 10 - 烯基,C 3 -C 10 - 炔基,C 3 -C 12 - 环烷基,C 3 -C 10 - 环烯基或五至十元饱和的部分不饱和或芳族杂环,其通过碳 并且含有一至四个由O,N和S组成的组的杂原子,R2是卤素,氰基,C1-C4-烷基,C2-C4-烯基,C2-C4-炔基,C1-C4-烷氧基,C3-C4 - 烯氧基或C 3 -C 4 - 炔氧基,其中R 2的烷基,烯基和炔基可以被卤素,氰基,硝基,C 1 -C 2 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代,并且R 3是氰基,CO 2 R a,C( -O)NR z R b,C(-O)-N-OR b,C(-S)-NR a R b,C(-NOR a)NR z R b,C(-NR a)NR z R b,C(O)NR a -NR b R b,C -NRaRb,C(-O)Ra,C(-NORb)Ra,C(-N-NRzRb)Ra,CRaRb-ORz,CRaRb-NRzRc,ON(-CRaRb),OC(-O)Ra,NRaRb ,NR a(C(-O)R b),NR a(C(-O)R b),NR a(C(-O)OR b) NRa-N RzRb,NRz-ORa,NRa(C(-NRc)-NRzRb),NRa(C(-NORc)Rb),制备这些化合物的方法,包含这些化合物的组合物及其杀虫剂用途。