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公开(公告)号:US08440672B2
公开(公告)日:2013-05-14
申请号:US12377136
申请日:2007-08-29
申请人: Anthony Ogawa , Feroze Ujjainwalla , Ellen K. Vande Bunte , Lin Chu , Debra Ondeyka , Ihor Kopka , Bing Li , Hyun Ok , Minal J. Patel , Jinyou Xu , Rosemary Sisco
发明人: Anthony Ogawa , Feroze Ujjainwalla , Ellen K. Vande Bunte , Lin Chu , Debra Ondeyka , Ihor Kopka , Bing Li , Hyun Ok , Minal J. Patel , Jinyou Xu , Rosemary Sisco
IPC分类号: A61K31/506 , A61K31/501 , A61K31/444 , C07D401/14 , C07D401/04
CPC分类号: C07D413/14 , C07D401/14 , C07D417/14
摘要: The instant invention provides compounds of Formula I which are 5-lipoxygenase activating protein inhibitors. Compounds of Formula (I) are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供了作为5-脂氧合酶活化蛋白抑制剂的式I化合物。 式(I)的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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公开(公告)号:US20100168076A1
公开(公告)日:2010-07-01
申请号:US12377136
申请日:2007-08-29
申请人: Anthony Ogawa , Feroze Ujjainwalla , Ellenk Vande Bunte , Lin Chu , Debra Ondeyka , Ihor Kopka , Bing Li , Hyun Ok , Minal J. Patel , Jinyou Xu , Rosemary Sisco
发明人: Anthony Ogawa , Feroze Ujjainwalla , Ellenk Vande Bunte , Lin Chu , Debra Ondeyka , Ihor Kopka , Bing Li , Hyun Ok , Minal J. Patel , Jinyou Xu , Rosemary Sisco
IPC分类号: A61K31/444 , C07D413/14 , A61K31/5377 , C07D401/14 , A61K31/501 , A61K31/506 , A61P11/02 , A61P11/00 , A61P29/00 , A61P37/08
CPC分类号: C07D413/14 , C07D401/14 , C07D417/14
摘要: The instant invention provides compounds of Formula I which are 5-lipoxygenase activating protein inhibitors. Compounds of Formula (I) are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供了作为5-脂氧合酶活化蛋白抑制剂的式I化合物。 式(I)的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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公开(公告)号:US20100190761A1
公开(公告)日:2010-07-29
申请号:US12665223
申请日:2008-06-16
申请人: Anthony Ogawa , Feroze Ujjainwalla , Ellen K. Vande Bunte , Lin Chu , Debra Ondeyka , Ihor E. Kopka , Bing Li , Hyun O. Ok , Minal Patel , Rosemary Sisco
发明人: Anthony Ogawa , Feroze Ujjainwalla , Ellen K. Vande Bunte , Lin Chu , Debra Ondeyka , Ihor E. Kopka , Bing Li , Hyun O. Ok , Minal Patel , Rosemary Sisco
IPC分类号: A61K31/4439 , C07D413/12 , C07D401/12 , C07D213/54 , C07D413/14 , A61K31/506 , A61K31/4545 , A61K31/439 , A61K31/5377 , A61K31/4245 , A61P9/10 , A61P11/06 , A61P11/00
CPC分类号: C07D401/12 , C07D209/30 , C07D213/65 , C07D237/20 , C07D401/10 , C07D403/04 , C07D403/10 , C07D413/10 , C07D413/12 , C07D417/12 , C07D471/04 , C07D487/04 , C07D513/04
摘要: The instant invention provides compounds of Formula I which are 5-lipoxygenase activating protein inhibitors: formula (I). Compounds of Formula I are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供式I化合物,它是5-脂氧合酶活化蛋白抑制剂:式(I)。 式I的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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公开(公告)号:US09029377B2
公开(公告)日:2015-05-12
申请号:US13382469
申请日:2010-06-28
申请人: Anthony Ogawa , Feroze Ujjainwalla , Lin Chu , Bing Li , Lan Wei , Jinyou Xu , Hyun Ok , Aaron Lackner , Ihor Kopka
发明人: Anthony Ogawa , Feroze Ujjainwalla , Lin Chu , Bing Li , Lan Wei , Jinyou Xu , Hyun Ok , Aaron Lackner , Ihor Kopka
IPC分类号: A61K31/50 , A61K31/4965 , A61K31/505 , A61K31/44 , A61K31/4245 , A61K31/4196 , A61K31/42 , C07D487/00 , C07D401/00 , C07D403/00 , C07D231/02 , C07D271/00 , C07D261/02 , C07D249/08 , G01C23/00 , G08G5/00
CPC分类号: G01C23/00 , G08G5/0056
摘要: Cyclohexyl sulfonamide compounds which are platelet-activating factor (PAF) receptor antagonists. Said compounds may be useful, for example, for the treatment of atherosclerosis or other PAF-mediated disorders, including inflammatory, cardiovascular, and immune disorders.
摘要翻译: 作为血小板活化因子(PAF)受体拮抗剂的环己基磺酰胺化合物。 所述化合物可用于例如治疗动脉粥样硬化或其它PAF介导的病症,包括炎性,心血管和免疫疾病。
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公开(公告)号:US20120108595A1
公开(公告)日:2012-05-03
申请号:US13382469
申请日:2010-06-28
申请人: Anthony Ogawa , Feroze Ujjainwalla , Lin Chu , Bing Li , Lan Wei , Jinyou Xu , Hyun Ok , Aaron Lackner , Ihor Kopka
发明人: Anthony Ogawa , Feroze Ujjainwalla , Lin Chu , Bing Li , Lan Wei , Jinyou Xu , Hyun Ok , Aaron Lackner , Ihor Kopka
IPC分类号: A61K31/4196 , C07D471/04 , C07D249/08 , C07D401/12 , C07D403/12 , C07D405/12 , C07D487/04 , C07F5/04 , A61K31/4245 , A61K31/437 , A61K31/4439 , A61K31/506 , A61K31/422 , A61K31/519 , A61K31/497 , A61P9/10 , A61P29/00 , A61P19/02 , A61P11/06 , A61P1/04 , A61P1/00 , A61P17/06 , C07D413/12
CPC分类号: G01C23/00 , G08G5/0056
摘要: Cyclohexyl sulfonamide compounds which are platelet-activating factor (PAF) receptor antagonists. Said compounds may be useful, for example, for the treatment of atherosclerosis or other PAF-mediated disorders, including inflammatory, cardiovascular, and immune disorders.
摘要翻译: 作为血小板活化因子(PAF)受体拮抗剂的环己基磺酰胺化合物。 所述化合物可用于例如治疗动脉粥样硬化或其它PAF介导的病症,包括炎性,心血管和免疫疾病。
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公开(公告)号:US20090258851A1
公开(公告)日:2009-10-15
申请号:US12296117
申请日:2007-04-06
申请人: LIN Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
发明人: LIN Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
IPC分类号: A61K31/397 , A61K31/5377 , A61K31/501 , A61K31/506 , A61K31/4545 , A61K31/444 , C07D413/14 , C07D403/14 , C07D401/14 , C07D417/14 , A61P9/10 , A61P11/06
CPC分类号: C07D213/65 , C07D401/14 , C07D413/14 , C07D417/14
摘要: The instant invention provides compounds of Formula II which are 5-lipoxygenase activating protein inhibitors. Compounds of Formula II are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供了作为5-脂氧合酶活化蛋白抑制剂的式II化合物。 式II的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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公开(公告)号:US08426413B2
公开(公告)日:2013-04-23
申请号:US13403643
申请日:2012-02-23
申请人: Lin Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L. Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
发明人: Lin Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L. Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
IPC分类号: A61K31/506 , A61K31/501 , A61K31/444 , C07D401/14 , C07D401/04
CPC分类号: C07D213/65 , C07D401/14 , C07D413/14 , C07D417/14
摘要: The instant invention provides compounds of Formula II which are 5-lipoxygenase activating protein inhibitors. Compounds of Formula II are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供了作为5-脂氧合酶活化蛋白抑制剂的式II化合物。 式II的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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公开(公告)号:US20120149674A1
公开(公告)日:2012-06-14
申请号:US13403643
申请日:2012-02-23
申请人: Lin Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L. Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
发明人: Lin Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L. Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
IPC分类号: A61K31/444 , C07D417/14 , C07D401/14 , A61K31/5377 , A61P11/06 , A61K31/506 , A61K31/4439 , A61K31/501 , A61P9/10 , A61P11/00 , C07D413/14 , A61K31/4545
CPC分类号: C07D213/65 , C07D401/14 , C07D413/14 , C07D417/14
摘要: The instant invention provides compounds of Formula II which are 5-lipoxygenase activating protein inhibitors. Compounds of Formula II are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供了作为5-脂氧合酶活化蛋白抑制剂的式II化合物。 式II的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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公开(公告)号:US08124628B2
公开(公告)日:2012-02-28
申请号:US12296117
申请日:2007-04-06
申请人: Lin Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L. Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
发明人: Lin Chu , Bing Li , Anthony K. Ogawa , Hyun O. Ok , Debra L. Ondeyka , Minal Patel , Rosemary Sisco , Feroze Ujjainwalla , Jinyou Xu
IPC分类号: A61K31/5377 , A61K31/506 , A61K31/501 , A61K31/4545 , A61K31/444 , A61K31/4439 , C07D417/14 , C07D413/14 , C07D407/14 , C07D401/14
CPC分类号: C07D213/65 , C07D401/14 , C07D413/14 , C07D417/14
摘要: The instant invention provides compounds of Formula II which are 5-lipoxygenase activating protein inhibitors. Compounds of Formula II are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供了作为5-脂氧合酶活化蛋白抑制剂的式II化合物。 式II的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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公开(公告)号:US20070287736A1
公开(公告)日:2007-12-13
申请号:US11665242
申请日:2005-10-14
申请人: Lin Chu , Ihor Kopka , Bing Li , Anthony Ogawa , Feroze Ujjainwalla
发明人: Lin Chu , Ihor Kopka , Bing Li , Anthony Ogawa , Feroze Ujjainwalla
IPC分类号: A61K31/443 , A61K31/4439 , A61P9/10 , C07D401/02 , C07D413/02
CPC分类号: C07D213/30 , C07D401/12 , C07D401/14 , C07D413/12
摘要: The instant invention provides compounds of formula I which are 5-lipoxygenase activating protein inhibitors. Compounds of formula I are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti-inflammatory and cytoprotective agents.
摘要翻译: 本发明提供了作为5-脂氧合酶活化蛋白抑制剂的式I化合物。 式I的化合物可用作抗动脉粥样硬化,抗哮喘,抗过敏,抗炎和细胞保护剂。
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