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公开(公告)号:US08232391B2
公开(公告)日:2012-07-31
申请号:US12833682
申请日:2010-07-09
申请人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, Jr. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
发明人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, Jr. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
IPC分类号: C07D279/10 , A61K31/54
CPC分类号: A61K31/4375 , A61K31/444 , A61K31/4453 , A61K31/4709 , A61K31/498 , A61K31/538 , A61K31/5383 , A61K31/5415 , A61K31/55 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Antibacterial compounds, compositions containing them, and methods of use for the inhibition of bacterial activity and the treatment, prevention or inhibition of bacterial infection.
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公开(公告)号:US20100274005A1
公开(公告)日:2010-10-28
申请号:US12833752
申请日:2010-07-09
申请人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, JR. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
发明人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, JR. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
IPC分类号: C07D487/04 , C07D471/04 , C07D417/14 , C07D403/14 , C07D498/04
CPC分类号: A61K31/4375 , A61K31/444 , A61K31/4453 , A61K31/4709 , A61K31/498 , A61K31/538 , A61K31/5383 , A61K31/5415 , A61K31/55 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Antibacterial compounds, compositions containing them, and methods of use for the inhibition of bacterial activity and the treatment, prevention or inhibition of bacterial infection.
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公开(公告)号:US08242275B2
公开(公告)日:2012-08-14
申请号:US12833621
申请日:2010-07-09
申请人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, Jr. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
发明人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, Jr. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
IPC分类号: C07D471/02
CPC分类号: A61K31/4375 , A61K31/444 , A61K31/4453 , A61K31/4709 , A61K31/498 , A61K31/538 , A61K31/5383 , A61K31/5415 , A61K31/55 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Antibacterial compounds, compositions containing them, and methods of use for the inhibition of bacterial activity and the treatment, prevention or inhibition of bacterial infection.
摘要翻译: 抗菌化合物,含有它们的组合物,以及用于抑制细菌活性和治疗,预防或抑制细菌感染的方法。
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公开(公告)号:US20100274004A1
公开(公告)日:2010-10-28
申请号:US12833682
申请日:2010-07-09
申请人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, JR. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J.M. Wiener
发明人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brian J. Morrow , S. Timothy Motley , Alejandro Santillan, JR. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J.M. Wiener
IPC分类号: C07D487/04 , C07D471/04 , C07D417/14 , C07D403/14 , C07D498/04
CPC分类号: A61K31/4375 , A61K31/444 , A61K31/4453 , A61K31/4709 , A61K31/498 , A61K31/538 , A61K31/5383 , A61K31/5415 , A61K31/55 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Antibacterial compounds, compositions containing them, and methods of use for the inhibition of bacterial activity and the treatment, prevention or inhibition of bacterial infection.
摘要翻译: 抗菌化合物,含有它们的组合物,以及用于抑制细菌活性和治疗,预防或抑制细菌感染的方法。
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公开(公告)号:US20100280240A1
公开(公告)日:2010-11-04
申请号:US12833621
申请日:2010-07-09
申请人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brain J. Morrow , S. Timothy Motley , Alejandro Santillan, JR. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J.M. Wiener
发明人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Brain J. Morrow , S. Timothy Motley , Alejandro Santillan, JR. , Karen J. Shaw , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J.M. Wiener
IPC分类号: C07D487/04 , C07D471/04 , C07D417/14 , C07D403/14 , C07D498/04
CPC分类号: A61K31/4375 , A61K31/444 , A61K31/4453 , A61K31/4709 , A61K31/498 , A61K31/538 , A61K31/5383 , A61K31/5415 , A61K31/55 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Antibacterial compounds, compositions containing them, and methods of use for the inhibition of bacterial activity and the treatment, prevention or inhibition of bacterial infection.
摘要翻译: 抗菌化合物,含有它们的组合物,以及用于抑制细菌活性和治疗,预防或抑制细菌感染的方法。
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公开(公告)号:US07842810B2
公开(公告)日:2010-11-30
申请号:US11393558
申请日:2006-03-30
申请人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Alejandro Santillan, Jr. , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
发明人: Brett D. Allison , Laurent Gomez , Cheryl A. Grice , Michael D. Hack , Alejandro Santillan, Jr. , Kimberly L. Schwarz , Liu Y. Tang , Hariharan Venkatesan , John J. M. Wiener
IPC分类号: C07D215/00
CPC分类号: A61K31/4375 , A61K31/444 , A61K31/4453 , A61K31/4709 , A61K31/498 , A61K31/538 , A61K31/5383 , A61K31/5415 , A61K31/55 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Antibacterial compounds, compositions containing them, and methods of use for the inhibition of bacterial activity and the treatment, prevention or inhibition of bacterial infection.
摘要翻译: 抗菌化合物,含有它们的组合物,以及用于抑制细菌活性和治疗,预防或抑制细菌感染的方法。
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公开(公告)号:US07202269B2
公开(公告)日:2007-04-10
申请号:US10976067
申请日:2004-10-28
申请人: Tristin K. Barclay , Alejandro Santillán, Jr. , Liu Y. Tang , Hariharan Venkatesan , Ronald L. Wolin
发明人: Tristin K. Barclay , Alejandro Santillán, Jr. , Liu Y. Tang , Hariharan Venkatesan , Ronald L. Wolin
IPC分类号: A61K31/40 , A61K31/17 , C07D207/06 , C07C335/18
CPC分类号: C07D295/13 , C07C275/28 , C07C275/36 , C07C279/28 , C07D213/56 , C07D277/30 , C07D333/20 , C07D333/24
摘要: Certain α-, β-, and γ-amino acid derivatives are disclosed as selective GlyT2 inhibitors for the treatment of central nervous system (CNS) conditions such as muscle spasticity, tinnitus, epilepsy and neuropathic pain.
摘要翻译: 公开了某些α-,β-和γ-氨基酸衍生物作为选择性GlyT2抑制剂用于治疗中枢神经系统(CNS)病症如肌肉痉挛,耳鸣,癫痫和神经性疼痛。
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公开(公告)号:US07276610B2
公开(公告)日:2007-10-02
申请号:US10919734
申请日:2004-08-17
申请人: Charles Q. Huang , Timothy W. Lovenberg , Alejandro Santillán, Jr. , Liu Y. Tang , Ronald L. Wolin
发明人: Charles Q. Huang , Timothy W. Lovenberg , Alejandro Santillán, Jr. , Liu Y. Tang , Ronald L. Wolin
IPC分类号: C07D211/60 , C07D207/04 , C07D223/02 , C07D265/30 , C07D295/02 , A61K31/445
CPC分类号: C07D295/192 , C07C237/30 , C07D211/46 , C07D333/20 , C07D333/38
摘要: The invention provides novel GlyT2 inhibiting compounds useful in modulating, treating, or preventing: anxiolytic disorders; a condition requiring treatment of injured mammalian nerve tissue; a condition amenable to treatment through administration of a neurotrophic factor; a neurological disorder; or obesity; an obesity-related disorder.
摘要翻译: 本发明提供了用于调节,治疗或预防:抗焦虑障碍的新型GlyT2抑制化合物; 需要治疗受损哺乳动物神经组织的病症; 适用于通过施用神经营养因子治疗的病症; 神经障碍 或肥胖; 肥胖相关疾病。
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公开(公告)号:US07915420B2
公开(公告)日:2011-03-29
申请号:US11780133
申请日:2007-07-19
申请人: Charles Q. Huang , Timothy W. Lovenberg , Alejandro Santillán, Jr. , Liu Y. Tang , Ronald L. Wolin
发明人: Charles Q. Huang , Timothy W. Lovenberg , Alejandro Santillán, Jr. , Liu Y. Tang , Ronald L. Wolin
IPC分类号: A61K31/4535 , C07D211/04 , C07D409/02
CPC分类号: C07D295/192 , C07C237/30 , C07D211/46 , C07D333/20 , C07D333/38
摘要: The invention provides novel GlyT2 inhibiting compounds useful in modulating, treating, or preventing: anxiolytic disorders; a condition requiring treatment of injured mammalian nerve tissue; a condition amenable to treatment through administration of a neurotrophic factor; a neurological disorder; or obesity; an obesity-related disorder.
摘要翻译: 本发明提供了用于调节,治疗或预防:抗焦虑障碍的新型GlyT2抑制化合物; 需要治疗受损哺乳动物神经组织的病症; 适用于通过施用神经营养因子治疗的病症; 神经障碍 或肥胖; 肥胖相关疾病。
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