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公开(公告)号:US09273028B2
公开(公告)日:2016-03-01
申请号:US13882449
申请日:2011-10-28
申请人: Brian T. Hopkins , Daniel Scott , Patrick Conlon , Tracy J. Jenkins , Noel Powell , Bing Guan , Julio H. Cuervo , Deping Wang , Art Taveras
发明人: Brian T. Hopkins , Daniel Scott , Patrick Conlon , Tracy J. Jenkins , Noel Powell , Bing Guan , Julio H. Cuervo , Deping Wang , Art Taveras
IPC分类号: A01N43/00 , A61K31/00 , C07D401/12 , C07D403/04 , C07D413/12 , C07D471/04 , C07D487/04 , C07D519/00 , C07D473/34 , C07D513/04
CPC分类号: A61K31/553 , A61K31/4545 , A61K31/496 , A61K31/506 , A61K31/519 , A61K31/52 , A61K31/5377 , A61K31/55 , C07D401/12 , C07D403/04 , C07D413/12 , C07D471/04 , C07D473/34 , C07D487/04 , C07D513/04 , C07D519/00
摘要: The present invention provides compounds useful as inhibitors of Tec family kinases, compositions thereof, and methods of using the same.
摘要翻译: 本发明提供可用作Tec家族激酶抑制剂的化合物,其组合物及其使用方法。
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公开(公告)号:US20120157443A1
公开(公告)日:2012-06-21
申请号:US13393192
申请日:2010-09-03
申请人: Minna Bui , Patrick Conlon , Julio H. Cuervo , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Tracy J. Jenkins , Gnanasambandam Kumaravel , Alexey A. Lugovskoy , Doug Marcotte , Noel Powell , Daniel Scott , Laura Silvian , Art Taveras , Deping Wang , Min Zhong
发明人: Minna Bui , Patrick Conlon , Julio H. Cuervo , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Tracy J. Jenkins , Gnanasambandam Kumaravel , Alexey A. Lugovskoy , Doug Marcotte , Noel Powell , Daniel Scott , Laura Silvian , Art Taveras , Deping Wang , Min Zhong
IPC分类号: A61K31/553 , C07D487/04 , A61K31/519 , C07D401/04 , A61K31/506 , C07D473/34 , A61K31/52 , C07D417/14 , C07D413/12 , C07D401/14 , A61K31/55 , A61P37/06 , A61P29/00 , A61P35/00 , A61P35/02 , C12N9/99
CPC分类号: C07D487/14 , A61K31/519 , C07D401/04 , C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D473/34 , C07D487/04
摘要: The present invention provides compounds useful as inhibitors of Btk, compositions thereof, and methods of using the same.
摘要翻译: 本发明提供了可用作Btk抑制剂的化合物,其组合物及其使用方法。
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公开(公告)号:US08785440B2
公开(公告)日:2014-07-22
申请号:US13393192
申请日:2010-09-03
申请人: Minna Bui , Patrick Conlon , Julio H. Cuervo , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Tracy J. Jenkins , Gnanasambandam Kumaravel , Alexey A. Lugovskoy , Doug Marcotte , Noel Powell , Daniel Scott , Laura Silvian , Art Taveras , Deping Wang , Min Zhong
发明人: Minna Bui , Patrick Conlon , Julio H. Cuervo , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Tracy J. Jenkins , Gnanasambandam Kumaravel , Alexey A. Lugovskoy , Doug Marcotte , Noel Powell , Daniel Scott , Laura Silvian , Art Taveras , Deping Wang , Min Zhong
IPC分类号: A61K31/535
CPC分类号: C07D487/14 , A61K31/519 , C07D401/04 , C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D473/34 , C07D487/04
摘要: The present invention provides compounds useful as inhibitors of Btk, compositions thereof, and methods of using the same.
摘要翻译: 本发明提供了可用作Btk抑制剂的化合物,其组合物及其使用方法。
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公开(公告)号:US20130345192A1
公开(公告)日:2013-12-26
申请号:US13882449
申请日:2011-10-28
申请人: Brian T. Hopkins , Daniel Scott , Patrick Conlon , Tracy J. Jenkins , Noel Powell , Bing Guan , Julio H. Cuervo , Deping Wang , Art Taveras
发明人: Brian T. Hopkins , Daniel Scott , Patrick Conlon , Tracy J. Jenkins , Noel Powell , Bing Guan , Julio H. Cuervo , Deping Wang , Art Taveras
IPC分类号: C07D401/12 , C07D513/04 , C07D473/34 , C07D471/04 , C07D487/04
CPC分类号: A61K31/553 , A61K31/4545 , A61K31/496 , A61K31/506 , A61K31/519 , A61K31/52 , A61K31/5377 , A61K31/55 , C07D401/12 , C07D403/04 , C07D413/12 , C07D471/04 , C07D473/34 , C07D487/04 , C07D513/04 , C07D519/00
摘要: The present invention provides compounds useful as inhibitors of Tec family kinases, compositions thereof, and methods of using the same.
摘要翻译: 本发明提供可用作Tec家族激酶抑制剂的化合物,其组合物及其使用方法。
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公开(公告)号:US20120157442A1
公开(公告)日:2012-06-21
申请号:US13393191
申请日:2010-09-03
申请人: Minna Bui , Patrick Conlon , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Alexey Ishchenko , Tracy J. Jenkins , Gnanasambandam Kumaravel , Doug Marcotte , Noel Powell , Daniel Scott , Art Taveras , Deping Wang , Min Zhong
发明人: Minna Bui , Patrick Conlon , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Alexey Ishchenko , Tracy J. Jenkins , Gnanasambandam Kumaravel , Doug Marcotte , Noel Powell , Daniel Scott , Art Taveras , Deping Wang , Min Zhong
IPC分类号: A61K31/553 , A61K31/519 , A61K31/5377 , C07D401/04 , A61K31/506 , A61P35/02 , A61K31/55 , C12N9/99 , A61P37/06 , A61P29/00 , A61P35/00 , C07D487/04 , C07D471/04
CPC分类号: C07D473/34 , C07D239/70 , C07D401/04 , C07D471/04 , C07D487/04
摘要: The present invention provides compounds useful as inhibitors of Btk, compositions thereof, and methods of using the same.
摘要翻译: 本发明提供了可用作Btk抑制剂的化合物,其组合物及其使用方法。
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公开(公告)号:US09029359B2
公开(公告)日:2015-05-12
申请号:US13393191
申请日:2010-09-03
申请人: Minna Bui , Patrick Conlon , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Alexey Ishchenko , Tracy J. Jenkins , Gnanasambandam Kumaravel , Doug Marcotte , Noel Powell , Daniel Scott , Art Taveras , Deping Wang , Min Zhong
发明人: Minna Bui , Patrick Conlon , Daniel A. Erlanson , Junfa Fan , Bing Guan , Brian T. Hopkins , Alexey Ishchenko , Tracy J. Jenkins , Gnanasambandam Kumaravel , Doug Marcotte , Noel Powell , Daniel Scott , Art Taveras , Deping Wang , Min Zhong
IPC分类号: C07D473/34 , C07D471/04 , C07D239/70 , C07D401/04 , C07D487/04
CPC分类号: C07D473/34 , C07D239/70 , C07D401/04 , C07D471/04 , C07D487/04
摘要: The present invention provides compounds useful as inhibitors of Btk, compositions thereof, and methods of using the same.
摘要翻译: 本发明提供了可用作Btk抑制剂的化合物,其组合物及其使用方法。
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公开(公告)号:US08618042B2
公开(公告)日:2013-12-31
申请号:US11698299
申请日:2007-01-25
IPC分类号: A01N61/00
CPC分类号: C07D211/74 , A61K38/00 , A61K47/6889 , C07D225/02 , C07D233/64 , C07D233/82 , C07D253/10 , C07D305/14 , C07D309/14 , C07D309/30 , C07D315/00 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/14 , C07D407/08 , C07D407/14 , C07D413/10 , C07D413/14 , C07D491/153 , C07D491/22
摘要: Binding molecules are described.
摘要翻译: 描述了结合分子。
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公开(公告)号:US09546165B2
公开(公告)日:2017-01-17
申请号:US13499835
申请日:2010-10-05
申请人: Joseph Arndt , Timothy Chan , Kevin Guckian , Gnanasambandam Kumaravel , Wen-Cherng Lee , Edward Yin-Shiang Lin , Daniel Scott , Lihong Sun , Jermaine Thomas , Kurt van Vloten , Deping Wang , Lei Zhang , Daniel Erlanson
发明人: Joseph Arndt , Timothy Chan , Kevin Guckian , Gnanasambandam Kumaravel , Wen-Cherng Lee , Edward Yin-Shiang Lin , Daniel Scott , Lihong Sun , Jermaine Thomas , Kurt van Vloten , Deping Wang , Lei Zhang , Daniel Erlanson
IPC分类号: C07D471/04 , C07D487/04 , C07D239/94 , C07D241/26 , C07D213/82 , C07D213/85 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D409/04 , C07D409/14 , C07D417/14 , C07D473/34 , C07D491/052 , C07D519/00 , C07D241/28 , C07D498/04
CPC分类号: C07D471/04 , A61K31/437 , A61K31/4439 , A61K31/444 , A61K31/452 , A61K31/4725 , A61K31/496 , A61K31/497 , A61K31/498 , A61K31/4985 , A61K31/517 , A61K31/519 , A61K31/53 , A61K31/5377 , A61K31/5383 , C07D213/82 , C07D213/85 , C07D241/26 , C07D241/28 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D409/04 , C07D409/14 , C07D417/14 , C07D473/34 , C07D487/04 , C07D491/052 , C07D498/04 , C07D519/00
摘要: The present invention provides compounds useful as inhibitors of PDK1. The present invention also provides compositions thereof, and methods of treating PDK1-mediated diseases.
摘要翻译: 本发明提供了可用作PDK1抑制剂的化合物。 本发明还提供了其组合物,以及治疗PDK1介导的疾病的方法。
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公开(公告)号:US20120208819A1
公开(公告)日:2012-08-16
申请号:US13499835
申请日:2010-10-05
申请人: Joseph Arndt , Timothy Chan , Kevin Guckian , Gnanasambandam Kumaravel , Wen-Cherng Lee , Edward Yin-Shiang Lin , Daniel Scott , Lihong Sun , Jermaine Thomas , Kurt van Vloten , Deping Wang , Lei Zhang , Daniel Erlanson
发明人: Joseph Arndt , Timothy Chan , Kevin Guckian , Gnanasambandam Kumaravel , Wen-Cherng Lee , Edward Yin-Shiang Lin , Daniel Scott , Lihong Sun , Jermaine Thomas , Kurt van Vloten , Deping Wang , Lei Zhang , Daniel Erlanson
IPC分类号: A61K31/53 , C07D401/14 , C07D409/14 , A61P35/00 , A61K31/444 , A61K31/519 , A61K31/4439 , A61K31/517 , C07D471/04 , C07D401/12
CPC分类号: C07D471/04 , A61K31/437 , A61K31/4439 , A61K31/444 , A61K31/452 , A61K31/4725 , A61K31/496 , A61K31/497 , A61K31/498 , A61K31/4985 , A61K31/517 , A61K31/519 , A61K31/53 , A61K31/5377 , A61K31/5383 , C07D213/82 , C07D213/85 , C07D241/26 , C07D241/28 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D409/04 , C07D409/14 , C07D417/14 , C07D473/34 , C07D487/04 , C07D491/052 , C07D498/04 , C07D519/00
摘要: The present invention provides compounds useful as inhibitors of PDK1. The present invention also provides compositions thereof, and methods of treating PDK1-mediated diseases.
摘要翻译: 本发明提供了可用作PDK1抑制剂的化合物。 本发明还提供了其组合物,以及治疗PDK1介导的疾病的方法。
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公开(公告)号:US20070066533A1
公开(公告)日:2007-03-22
申请号:US11600145
申请日:2006-11-16
申请人: Wen-Cherng Lee , R. Pepinsky , Mark Cornebise , Daniel Scott , Russell Petter
发明人: Wen-Cherng Lee , R. Pepinsky , Mark Cornebise , Daniel Scott , Russell Petter
IPC分类号: A61K38/17 , A61K31/4015
CPC分类号: C07K5/06165
摘要: Cell adhesion inhibitors can interact with VLA-4 molecules and inhibits VLA-4 dependent cell adhesion. An inhibitor including a polyethylene glycol moiety can have advantageous pharmaceutical properties.
摘要翻译: 细胞粘附抑制剂可与VLA-4分子相互作用并抑制VLA-4依赖性细胞粘附。 包含聚乙二醇部分的抑制剂可以具有有利的药物性质。
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