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公开(公告)号:US20100261714A1
公开(公告)日:2010-10-14
申请号:US12756276
申请日:2010-04-08
申请人: Claudio STURINO , Patrick DEROY , Martin DUPLESSIS , Paul J. EDWARDS , Anne-Marie FAUCHER , Teddy HALMOS , Clint JAMES , Jean-Eric LACOSTE , Eric MALENFANT , Joannie MINVILLE , Louis MORENCY , Sebastien MORIN , Martin TREMBLAY , Christiane YOAKIM
发明人: Claudio STURINO , Patrick DEROY , Martin DUPLESSIS , Paul J. EDWARDS , Anne-Marie FAUCHER , Teddy HALMOS , Clint JAMES , Jean-Eric LACOSTE , Eric MALENFANT , Joannie MINVILLE , Louis MORENCY , Sebastien MORIN , Martin TREMBLAY , Christiane YOAKIM
IPC分类号: A61K31/519 , C07D491/048 , C07D413/14 , A61K31/5377 , A61K31/496 , C07D495/04 , A61K31/542 , A61P31/18 , A61K31/497
CPC分类号: C07D491/048 , C07D487/04 , C07D491/147 , C07D513/04 , C07D519/00
摘要: Compounds of formula (I): wherein R1, R2, A1, A2, A3, A4, X and Y are as defined herein, are useful as inhibitors of HIV replication.
摘要翻译: 式(I)化合物:其中R1,R2,A1,A2,A3,A4,X和Y如本文所定义,可用作HIV复制的抑制剂。
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公开(公告)号:US20080221159A1
公开(公告)日:2008-09-11
申请号:US11746303
申请日:2007-05-09
申请人: Youla S. TSANTRIZOS , Michael BOES , Christian BROCHU , Craig FENWICK , Stephen MASON , Marc PESANT , Eric MALENFANT
发明人: Youla S. TSANTRIZOS , Michael BOES , Christian BROCHU , Craig FENWICK , Stephen MASON , Marc PESANT , Eric MALENFANT
IPC分类号: A61K31/47 , C07D215/06 , C07D215/12 , A61K31/4709 , A61P31/18 , A61K31/352 , C07D215/227 , C07D311/02
CPC分类号: C07D215/22 , C07D215/14 , C07D215/18 , C07D215/227 , C07D311/08 , C07D311/12 , C07D311/14 , C07D401/04 , C07D401/12 , C07D405/04 , C07D409/04 , C07D413/12
摘要: Compounds of formula I: wherein a, b, c, X, R2, R3, R4, R6 and R7 are defined herein, are useful as inhibitors of HIV replication.
摘要翻译: 式I化合物:其中a,b,c,X,R 2,R 3,R 4,R 6, / SUP>和R>在本文中定义,可用作HIV复制的抑制剂。
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