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公开(公告)号:US20100261714A1
公开(公告)日:2010-10-14
申请号:US12756276
申请日:2010-04-08
申请人: Claudio STURINO , Patrick DEROY , Martin DUPLESSIS , Paul J. EDWARDS , Anne-Marie FAUCHER , Teddy HALMOS , Clint JAMES , Jean-Eric LACOSTE , Eric MALENFANT , Joannie MINVILLE , Louis MORENCY , Sebastien MORIN , Martin TREMBLAY , Christiane YOAKIM
发明人: Claudio STURINO , Patrick DEROY , Martin DUPLESSIS , Paul J. EDWARDS , Anne-Marie FAUCHER , Teddy HALMOS , Clint JAMES , Jean-Eric LACOSTE , Eric MALENFANT , Joannie MINVILLE , Louis MORENCY , Sebastien MORIN , Martin TREMBLAY , Christiane YOAKIM
IPC分类号: A61K31/519 , C07D491/048 , C07D413/14 , A61K31/5377 , A61K31/496 , C07D495/04 , A61K31/542 , A61P31/18 , A61K31/497
CPC分类号: C07D491/048 , C07D487/04 , C07D491/147 , C07D513/04 , C07D519/00
摘要: Compounds of formula (I): wherein R1, R2, A1, A2, A3, A4, X and Y are as defined herein, are useful as inhibitors of HIV replication.
摘要翻译: 式(I)化合物:其中R1,R2,A1,A2,A3,A4,X和Y如本文所定义,可用作HIV复制的抑制剂。
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公开(公告)号:US20110230465A1
公开(公告)日:2011-09-22
申请号:US12883677
申请日:2010-09-16
申请人: Timothy STAMMERS , Xavier BARBEAU , Pierre BEAULIEU , Megan BERTRAND-LAPERLE , Christian BROCHU , Paul J. EDWARDS , Pasquale FORGIONE , Cédrickx GODBOUT , Oliver HUCKE , Marc-André JOLY , Serge LANDRY , Olivier LEPAGE , Julie NAUD , Marc PESANT , Martin POIRIER , Maude POIRIER , Bounkham THAVONEKHAM
发明人: Timothy STAMMERS , Xavier BARBEAU , Pierre BEAULIEU , Megan BERTRAND-LAPERLE , Christian BROCHU , Paul J. EDWARDS , Pasquale FORGIONE , Cédrickx GODBOUT , Oliver HUCKE , Marc-André JOLY , Serge LANDRY , Olivier LEPAGE , Julie NAUD , Marc PESANT , Martin POIRIER , Maude POIRIER , Bounkham THAVONEKHAM
IPC分类号: A61K31/517 , C07D401/12 , C07D401/14 , C07D239/88 , C07D413/14 , C07D405/12 , C07D417/14 , C07D487/04 , C07C251/48 , C07C233/13 , C07C211/29 , C07C255/58 , C07C255/59 , C07C237/44 , C07F5/04 , C07D213/74 , C07D239/30 , A61K31/5377 , A61K31/541 , A61P31/14
CPC分类号: C07D401/12 , A61K31/14 , A61K31/517 , C07C211/29 , C07C233/11 , C07C237/44 , C07C251/48 , C07C255/58 , C07C255/59 , C07D401/14 , C07D403/12 , C07D409/14 , C07D413/12 , C07F5/025
摘要: Compounds of formula I: wherein X, R2, R3, R5 and R6 are defined herein, are useful as inhibitors of the hepatitis C virus NS5B polymerase.
摘要翻译: 式I化合物:其中X,R 2,R 3,R 5和R 6在本文中定义,可用作丙型肝炎病毒NS5B聚合酶的抑制剂。
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