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公开(公告)号:US06380221B1
公开(公告)日:2002-04-30
申请号:US09631450
申请日:2000-08-03
申请人: Damian O. Arnaiz , Yuo-Ling Chou , Brian D. Griedel , Rushad E. Karanjawala , Monica J. Kochanny , Wheeseong Lee , Amy Mei Liang , Michael M. Morrissey , Gary B. Phillips , Karna Lyn Sacchi , Steven T. Sakata , Kenneth J. Shaw , R. Michael Snider , Shung C. Wu , Bin Ye , Zuchun Zhao
发明人: Damian O. Arnaiz , Yuo-Ling Chou , Brian D. Griedel , Rushad E. Karanjawala , Monica J. Kochanny , Wheeseong Lee , Amy Mei Liang , Michael M. Morrissey , Gary B. Phillips , Karna Lyn Sacchi , Steven T. Sakata , Kenneth J. Shaw , R. Michael Snider , Shung C. Wu , Bin Ye , Zuchun Zhao
IPC分类号: A61K3144
CPC分类号: C07D401/04 , C07D333/38 , C07D333/70 , C07D409/06 , C07D409/12 , C07D409/14 , C07D413/14 , C07D417/14 , C07D473/06 , C07D473/34
摘要: This invention is directed to compounds of formula (III): wherein B, C, D, E, R1, R2 and R3 are disclosed herein. These components are disclosed as being useful as anti-coagulants.
摘要翻译: 本发明涉及式(III)化合物:其中B,C,D,E,R 1,R 2和R 3在本文中公开。 这些组分被公开用作抗凝剂。
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公开(公告)号:US6140351A
公开(公告)日:2000-10-31
申请号:US187459
申请日:1998-11-05
申请人: Damian O. Arnaiz , Yuo-Ling Chou , Brian D. Griedel , Rushad E. Karanjawala , Monica J. Kochanny , Wheeseong Lee , Amy Mei Liang , Michael M. Morrissey , Gary B. Phillips , Karna Lyn Sacchi , Steven T. Sakata , Kenneth J. Shaw , R. Michael Snider , Shung C. Wu , Bin Ye , Zuchun Zhao
发明人: Damian O. Arnaiz , Yuo-Ling Chou , Brian D. Griedel , Rushad E. Karanjawala , Monica J. Kochanny , Wheeseong Lee , Amy Mei Liang , Michael M. Morrissey , Gary B. Phillips , Karna Lyn Sacchi , Steven T. Sakata , Kenneth J. Shaw , R. Michael Snider , Shung C. Wu , Bin Ye , Zuchun Zhao
IPC分类号: C07D333/38 , C07D333/70 , C07D401/04 , C07D409/06 , C07D409/12 , C07D409/14 , C07D413/14 , C07D417/14 , C07D473/06 , C07D473/34 , A61K31/44 , C07D409/00 , C07D411/00
CPC分类号: C07D401/04 , C07D333/38 , C07D333/70 , C07D409/06 , C07D409/12 , C07D409/14 , C07D413/14 , C07D417/14 , C07D473/06 , C07D473/34
摘要: This invention is directed to compounds of formula (III): ##STR1## wherein B, C, D, E, R.sup.1, R.sup.2 and R.sup.3 are disclosed herein. These compounds are disclosed as being useful as anti-coagulants.
摘要翻译: 本发明涉及式(III)化合物:其中B,C,D,E,R 1,R 2和R 3在本文中公开。 这些化合物被公开用作抗凝剂。
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公开(公告)号:US06498185B1
公开(公告)日:2002-12-24
申请号:US09631452
申请日:2000-08-03
申请人: Damian O. Arnaiz , Yuo-Ling Chou , Brian D. Griedel , Rushad E. Karanjawala , Monica J. Kochanny , Wheeseong Lee , Amy Mei Liang , Michael M. Morrissey , Gary B. Phillips , Karna Lyn Sacchi , Steven T. Sakata , Kenneth J. Shaw , R. Michael Snider , Shung C. Wu , Bin Ye , Zuchun Zhao
发明人: Damian O. Arnaiz , Yuo-Ling Chou , Brian D. Griedel , Rushad E. Karanjawala , Monica J. Kochanny , Wheeseong Lee , Amy Mei Liang , Michael M. Morrissey , Gary B. Phillips , Karna Lyn Sacchi , Steven T. Sakata , Kenneth J. Shaw , R. Michael Snider , Shung C. Wu , Bin Ye , Zuchun Zhao
IPC分类号: A01N4306
CPC分类号: C07D401/04 , C07D333/38 , C07D333/70 , C07D409/06 , C07D409/12 , C07D409/14 , C07D413/14 , C07D417/14 , C07D473/06 , C07D473/34
摘要: This invention is directed to compounds of formula (III): wherein B, C, D, E, R1, R2 and R3 are disclosed herein. These compounds are disclosed as being useful as anti coagulants.
摘要翻译: 本发明涉及式(III)化合物:其中B,C,D,E,R 1,R 2和R 3在本文中公开。 公开了这些化合物作为抗凝剂。
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4.
公开(公告)号:US5849759A
公开(公告)日:1998-12-15
申请号:US570057
申请日:1995-12-08
IPC分类号: C07D235/04 , A61K31/00 , A61K31/4427 , A61K31/445 , A61K31/4465 , A61K31/4523 , A61K31/454 , A61P7/00 , A61P7/02 , C07C257/18 , C07D235/06 , C07D401/12 , C07D211/52
CPC分类号: C07D401/12
摘要: Compounds of formula (I): ##STR1## wherein: n, A, R.sup.1, R.sup.2, R.sup.3, and R.sup.4 have meanings as defined herein, or a pharmaceutically acceptable salt thereof, are useful as anti-coagulants.
摘要翻译: 式(I)的化合物:其中:n,A,R 1,R 2,R 3和R 4具有如本文所定义的含义或其药学上可接受的盐,可用作抗凝剂。
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5.Imidazolidinedione analogs useful as anticoagulants and antithrombotics 失效
标题翻译: 用作抗凝血剂和抗血栓药物的咪唑烷二酮类似物公开(公告)号:US07053112B2
公开(公告)日:2006-05-30
申请号:US10668920
申请日:2003-09-23
IPC分类号: C07D231/04 , A61K31/4166
CPC分类号: C07D235/02 , C07D233/76 , C07D233/78 , C07D401/06 , C07D491/04
摘要: A compound is disclosed, which is useful in treating a mammal having a disease-state characterized by thrombotic activity. The compound is of the following formula: wherein A, B, R1, R2, R3 and R4 are as defined herein or an isomer or isomeric mixture thereof or a pharmaceutically acceptable salt thereof.
摘要翻译: 公开了一种化合物,其可用于治疗具有以血栓形成活性为特征的疾病状态的哺乳动物。 该化合物具有下式:其中A,B,R 1,R 2,R 3和R 4, SUB>如本文所定义,或其异构体或异构体混合物或其药学上可接受的盐。
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