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公开(公告)号:US5240928A
公开(公告)日:1993-08-31
申请号:US665518
申请日:1991-03-06
申请人: Eric E. Allen , Stephen E. de Laszlo , Prasun K. Chakravarty , William J. Greenlee , Arthur A. Patchett , Thomas F. Walsh
发明人: Eric E. Allen , Stephen E. de Laszlo , Prasun K. Chakravarty , William J. Greenlee , Arthur A. Patchett , Thomas F. Walsh
IPC分类号: C07D239/70 , C07D239/90 , C07D239/91 , C07D403/10
CPC分类号: C07D403/10 , C07D239/70 , C07D239/90 , C07D239/91
摘要: Novel substituted quinazolinones of the formula (I), which are useful as angiotensin II antagonists, are disclosed. ##STR1##
摘要翻译: 公开了可用作血管紧张素II拮抗剂的式(I)的新型取代喹唑啉酮。 (一)
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2.Substituted pyridopyrimidinones and related heterocycles as angiotensin II antagonists 失效
标题翻译: 取代的吡啶并嘧啶酮和相关杂环作为血管紧张素II拮抗剂公开(公告)号:US5330987A
公开(公告)日:1994-07-19
申请号:US894036
申请日:1992-06-04
申请人: Eric E. Allen , Prasun K. Chakravarty , Stephen E. de Laszlo , William J. Greenlee , Arthur A. Patchett , Thomas F. Walsh
发明人: Eric E. Allen , Prasun K. Chakravarty , Stephen E. de Laszlo , William J. Greenlee , Arthur A. Patchett , Thomas F. Walsh
IPC分类号: A61K31/505 , A61P9/00 , A61P9/12 , C07D471/04 , C07D403/12 , C07D487/04
CPC分类号: C07D471/04
摘要: Novel substituted pyridopyrimidinones of formula (I), which are useful as angiotensin II antagonists, are disclosed. ##STR1##
摘要翻译: 公开了可用作血管紧张素II拮抗剂的式(I)的新型取代的吡啶并嘧啶酮。 (一)
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公开(公告)号:US5250521A
公开(公告)日:1993-10-05
申请号:US794533
申请日:1991-11-25
申请人: Eric E. Allen , William J. Greenlee , Prasun K. Chakravarty , Malcolm MacCoss , Arthur A. Patchett , Thomas F. Walsh
发明人: Eric E. Allen , William J. Greenlee , Prasun K. Chakravarty , Malcolm MacCoss , Arthur A. Patchett , Thomas F. Walsh
IPC分类号: C07D487/04 , A61K31/505 , A61K31/535 , A61K31/54
CPC分类号: C07D487/04
摘要: Novel substituted pyrazolopyrimidines of formula (I) which are useful as angiotensin II antagonists, are disclosed. ##STR1##
摘要翻译: 公开了用作血管紧张素II拮抗剂的式(I)的新型取代吡唑并嘧啶。 (一)
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公开(公告)号:US5100897A
公开(公告)日:1992-03-31
申请号:US550951
申请日:1990-07-16
申请人: Eric E. Allen , William J. Greenlee , Prasun K. Chakravarty , Arthur A. Patchett , Thomas F. Walsh
发明人: Eric E. Allen , William J. Greenlee , Prasun K. Chakravarty , Arthur A. Patchett , Thomas F. Walsh
IPC分类号: A61K31/505 , A61P9/12 , A61P27/02 , C07D239/36 , C07D239/42 , C07D239/52 , C07D403/10 , C07D403/12 , C07F9/46
CPC分类号: C07D239/36 , C07D239/52 , C07D403/10
摘要: Novel substituted pyrimidinones of formula (I) which are useful as angiotensin II antagonists, are disclosed. ##STR1##
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公开(公告)号:US5260285A
公开(公告)日:1993-11-09
申请号:US794534
申请日:1991-11-25
申请人: Eric E. Allen , William J. Greenlee , Prasun K. Chakravarty , Malcolm MacCoss , Arthur A. Patchett , Thomas F. Walsh
发明人: Eric E. Allen , William J. Greenlee , Prasun K. Chakravarty , Malcolm MacCoss , Arthur A. Patchett , Thomas F. Walsh
IPC分类号: C07D487/04 , A61K31/675 , A61K31/50 , A61K31/505
CPC分类号: C07D487/04
摘要: Novel substituted imidazopyridazines of formula (I) which are useful as angiotensin II antagonists, are disclosed. ##STR1##
摘要翻译: 公开了可用作血管紧张素II拮抗剂的式(I)的新型取代咪唑并哒嗪。 (一)
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6.Substituted quinazolinones bearing acidic functional groups as angiotensin II antagonists 失效
标题翻译: 带有酸性官能团的取代喹唑啉酮作为血管紧张素II拮抗剂公开(公告)号:US5441959A
公开(公告)日:1995-08-15
申请号:US108465
申请日:1993-08-18
申请人: Prasun K. Chakravarty , Stephen E. de Laszlo , Tomasz W. Glinka , William J. Greenlee , Nathan B. Mantlo , Arthur A. Patchett
发明人: Prasun K. Chakravarty , Stephen E. de Laszlo , Tomasz W. Glinka , William J. Greenlee , Nathan B. Mantlo , Arthur A. Patchett
IPC分类号: A61K31/505 , A61K31/517 , A61P9/12 , A61P27/02 , A61P43/00 , C07D239/70 , C07D239/80 , C07D239/91 , C07D401/04 , C07D401/12 , C07D403/12 , C07D413/10 , C07D417/10 , C07D419/10 , C07D521/00 , C07D239/72 , C07D239/90
CPC分类号: C07D249/08 , C07D231/12 , C07D233/56 , C07D239/70 , C07D239/91 , C07D401/04 , C07D413/10 , C07D417/10
摘要: Novel substituted quinazolinones of the formula (I) are useful as angiotensin II antagonists. ##STR1##
摘要翻译: 式(I)的新型取代喹唑啉酮可用作血管紧张素II拮抗剂。 (一)
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公开(公告)号:US5385894A
公开(公告)日:1995-01-31
申请号:US222354
申请日:1994-04-04
申请人: Stephen E. de Laszlo , Tomasz W. Glinka , William J. Greenlee , Prasun K. Chakravarty , Arthur A. Patchett
发明人: Stephen E. de Laszlo , Tomasz W. Glinka , William J. Greenlee , Prasun K. Chakravarty , Arthur A. Patchett
IPC分类号: C07D239/90 , C07D401/14 , C07D403/10 , C07D405/14 , C07D409/14 , A61K31/505 , C07D239/91
CPC分类号: C07D401/14 , C07D239/90 , C07D403/10 , C07D405/14 , C07D409/14
摘要: Novel disubstituted 6-aminoquinazolinones of the Formula (I), are useful as angiotensin II antagonists: ##STR1##
摘要翻译: 式(I)的新型二取代的6-氨基喹唑啉酮可用作血管紧张素II拮抗剂:图1(I)
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8.Substituted quinazolinones bearing acidic functional groups as angiotensin II antagonists 失效
标题翻译: 作为ANGIOTENSIN II拮抗剂的作为酸性功能组的替代喹唑啉酮公开(公告)号:US5238942A
公开(公告)日:1993-08-24
申请号:US867794
申请日:1992-04-16
申请人: Prasun K. Chakravarty , William J. Greenlee , Nathan B. Mantlo , Arthur A. Patchett , Dooseop Kim , Stephen E. de Laszlo , Tomasz W. Glinka
发明人: Prasun K. Chakravarty , William J. Greenlee , Nathan B. Mantlo , Arthur A. Patchett , Dooseop Kim , Stephen E. de Laszlo , Tomasz W. Glinka
IPC分类号: A61K31/505 , A61K31/517 , A61P9/12 , A61P27/02 , A61P43/00 , C07D239/70 , C07D239/80 , C07D239/91 , C07D401/04 , C07D401/12 , C07D403/12 , C07D413/10 , C07D417/10 , C07D419/10 , C07D521/00
CPC分类号: C07D249/08 , C07D231/12 , C07D233/56 , C07D239/70 , C07D239/91 , C07D401/04 , C07D413/10 , C07D417/10
摘要: Novel substituted quinazolinones of the formula (I) are useful as angiotensin II antagonists. ##STR1##
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公开(公告)号:US5157026A
公开(公告)日:1992-10-20
申请号:US840241
申请日:1992-02-24
申请人: Prasun K. Chakravarty , William J. Greenlee , Nathan B. Mantlo , Arthur A. Patchett , Thomas F. Walsh
发明人: Prasun K. Chakravarty , William J. Greenlee , Nathan B. Mantlo , Arthur A. Patchett , Thomas F. Walsh
IPC分类号: C07D471/04 , C07D473/00 , C07D473/04 , C07D473/30 , C07D473/32 , C07D473/40 , C07F9/6561
CPC分类号: C07D471/04 , C07D473/00 , C07D473/04 , C07D473/30 , C07D473/32 , C07D473/40 , C07F9/6561
摘要: Substituted Imidazo-fused 6-membered heterocycles of structural formula: ##STR1## wherein A, B, C, and D are independently carbon atoms or nitrogen atoms are angiotensin II antagonists useful in the treatment of hypertension and congestive heart failure.
摘要翻译: 取代的具有结构式的咪唑并稠合的6元杂环:其中A,B,C和D独立地为碳原子或氮原子是可用于治疗高血压和充血性心力衰竭的血管紧张素II拮抗剂。
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10.Imidazole angiotensin II antagonists incorporating acidic functional groups 失效
标题翻译: 咪唑安定剂II加入酸性功能组的拮抗剂公开(公告)号:US5126342A
公开(公告)日:1992-06-30
申请号:US590971
申请日:1990-10-01
申请人: Prasun K. Chakravarty , William J. Greenlee , Elizabeth M. Naylor , Arthur A. Patchett , Thomas F. Walsh
发明人: Prasun K. Chakravarty , William J. Greenlee , Elizabeth M. Naylor , Arthur A. Patchett , Thomas F. Walsh
IPC分类号: A61K31/415 , A61K31/675 , A61K45/06 , A61P3/00 , A61P9/12 , A61P27/02 , A61P43/00 , C07D233/54 , C07D233/64 , C07D233/68 , C07D233/70 , C07D233/84 , C07D233/88 , C07D233/90 , C07D403/04 , C07D403/06 , C07D403/12 , C07D407/04 , C07D521/00 , C07F9/6506
CPC分类号: C07D233/64 , C07D231/12 , C07D233/56 , C07D233/68 , C07D233/88 , C07D233/90 , C07D249/08 , C07D403/04 , C07D403/06 , C07F9/65061
摘要: There are disclosed substituted imidazole derivatives of Formula I which are useful as angiotensin II antagonists. ##STR1##
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