公开(公告)号：US4790869A

公开(公告)日：1988-12-13

申请号：US9924

申请日：1987-02-02

申请人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Hiroshi Shimoharada ,  Tsunezo Yoshida ,  Masahiko Ikeguchi

发明人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Hiroshi Shimoharada ,  Tsunezo Yoshida ,  Masahiko Ikeguchi

IPC分类号： A01N47/36 ,  C07D275/02 ,  C07D275/03 ,  C07D521/00 ,  A01N43/54 ,  C07D239/47 ,  C07D417/12

CPC分类号： C07D275/03 ,  A01N47/36 ,  C07D521/00

摘要： A sulfonamide compound and a salt thereof is represented by the following general formula: ##STR1## wherein each of X.sub.1, X.sub.2, and X.sub.3 independently represents a hydrogen atom or a halogen atom, each of Y.sub.1, Y.sub.2, and Y.sub.3 independently represents a halogen atom, and R represents a methyl group or a methoxy group, and is effective as an active ingredient of a herbicidal composition.

摘要翻译： 磺酰胺化合物及其盐由以下通式表示：其中X1，X2和X3各自独立地表示氢原子或卤素原子，Y1，Y2和Y3各自独立地表示卤素原子 R表示甲基或甲氧基，作为除草组合物的有效成分是有效的。

公开(公告)号：US4835282A

公开(公告)日：1989-05-30

申请号：US244062

申请日：1988-09-14

申请人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Hiroshi Shimoharada ,  Tsunezo Yoshida ,  Masahiko Ikeguchi

发明人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Hiroshi Shimoharada ,  Tsunezo Yoshida ,  Masahiko Ikeguchi

IPC分类号： A01N47/36 ,  C07D275/02 ,  C07D275/03 ,  C07D521/00

CPC分类号： C07D275/03 ,  A01N47/36 ,  C07D521/00

摘要： A sulfonamide compound and a salt thereof is represented by the following general formula: ##STR1## wherein each of X.sub.1, X.sub.2, and X.sub.3 independently represents a hydrogen atom or a halogen atom, each of Y.sub.1, Y.sub.2, and Y.sub.3 independently represents a halogen atom, and R represents a methyl group or a methoxy group, and is effective as an active ingredient of a herbicidal composition.

公开(公告)号：US4935528A

公开(公告)日：1990-06-19

申请号：US301984

申请日：1989-01-26

申请人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Koji Hayashi ,  Masahiko Ikeguchi ,  Tsunezo Yoshida

发明人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Koji Hayashi ,  Masahiko Ikeguchi ,  Tsunezo Yoshida

IPC分类号： A01N47/36 ,  C07D409/12

CPC分类号： C07D409/12 ,  A01N47/36

摘要： A thiophenesulfonamide compound having the formula: ##STR1## wherein X is a halogenoalkoxyalkyl group, and Y is ##STR2## wherein A is .dbd.N-- or .dbd.CH--, and each of Z.sub.1 and Z.sub.2 is a methyl group or a methoxy group, and its salt.

摘要翻译： 具有下式的噻吩磺酰胺化合物：其中X是卤代烷氧基烷基，Y是其中A是= N-或= CH-，并且Z 1和Z 2各自是甲基或甲氧基 组，及其盐。

公开(公告)号：US4822402A

公开(公告)日：1989-04-18

申请号：US865467

申请日：1986-05-21

申请人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Koji Hayashi ,  Masahiko Ikeguchi ,  Tsunezo Yoshida

发明人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Koji Hayashi ,  Masahiko Ikeguchi ,  Tsunezo Yoshida

IPC分类号： A01N47/36 ,  C07D409/12 ,  A01N43/54

CPC分类号： C07D409/12 ,  A01N47/36

摘要： A thiophenesulfonamide compound having the formula: ##STR1## wherein X is a halogenoalkoxyalkyl group, and Y is ##STR2## wherein A is .dbd.N-- or .dbd.CH--, and each of Z.sub.1 and Z.sub.2 is a methyl group or a methoxy group, and its salt.

摘要翻译： 具有下式的噻吩磺酰胺化合物：其中X是卤代烷氧基烷基，Y是其中A是= N-或= CH-，并且Z 1和Z 2各自是甲基或甲氧基 组，及其盐。

公开(公告)号：US20100317528A1

公开(公告)日：2010-12-16

申请号：US12521649

申请日：2007-12-27

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Tatsuya Okita ,  Hiroshi Hata

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Tatsuya Okita ,  Hiroshi Hata

IPC分类号： A01N43/56 ,  C07D231/20 ,  A01P13/00

CPC分类号： A01N43/56 ,  C07C317/22 ,  C07D231/20 ,  C07D405/10 ,  C07D413/10

摘要： To provide a novel herbicide which has a wide range of applications to agricultural or non-agricultural fields and various methods for application such as soil treatment and foliage treatment and which exhibits excellent herbicidal effects.A herbicide containing a benzoylpyrazole compound represented by the formula (I) or its salt, as an active ingredient: wherein R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is hydroxy, R4 is alkyl, haloalkyl or the like, R5 is halogen, cyano, cyanoalkyl or the like, and R6 is haloalkyl, halogen or the like.

摘要翻译： 提供一种广泛应用于农业或非农业领域的新型除草剂和各种施用方法如土壤处理和叶面处理，并且具有优异的除草效果。 一种除草剂，其含有式（I）表示的苯甲酰基吡唑化合物或其盐作为活性成分：其中R1是烷基或环烷基，R2是氢原子或烷基，R3是羟基，R4是烷基，卤代烷基等， R5是卤素，氰基，氰基烷基等，R6是卤代烷基，卤素等。

公开(公告)号：US20110282070A1

公开(公告)日：2011-11-17

申请号：US13188402

申请日：2011-07-21

申请人： Hiroshi SHIMOHARADA ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi SHIMOHARADA ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： C07D413/10 ,  C07C317/46 ,  C07C51/60 ,  C07D231/20 ,  C07D405/10

CPC分类号： C07D231/20 ,  C07D405/12 ,  C07D413/12

摘要： A benzoylpyrazole compound represented by the formula (I) or its salt: wherein R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is alkyl; cycloalkyl; haloalkyl; alkoxyalkyl; alkoxycarbonylalkyl; alkenyl; or arylalkyl which may be substituted by R8, R4 is alkyl; haloalkyl; alkoxy; halogen; nitro; cyano; alkylthio; alkylsulfinyl; or alkylsulfonyl, R5 is a hydrogen atom; alkyl; alkenyl; alkynyl; halogen; cyano; cyanoalkyl; cyanoalkeny; haloalkyl; alkoxyalkyl; haloalkoxyalkyl; amino(thiocarbonyl)alkyl which may be substituted by at least one substituent selected from alkyl, cyano, is cyanoalkyl, (alkylthio)carbonylalkyl, alkyl(thiocarbonyl)alkyl, —C(O)OR7 and —C(O)SR7; thiocyanatoalkyl; alkoxy; alkenyloxy; alkynyloxy; haloalkoxy; alkoxyalkoxy; haloalkoxyalkoxy; alkoxyhaloalkoxy; haloalkoxyhaloalkoxy; alkoxyalkoxyalkyl; alkylthio; alkoxyalkylthio; haloalkoxyalkylthio; alkoxyhaloalkylthio; haloalkoxyhaloalkylthio; alkylthioalkylthio; haloalkylthioalkylthio; alkylthiohaloalkylthio; haloalkylthiohaloalkylthio; alkylthioalkoxy; alkylsulfonyl; alkylsulfonylalkyl; alkoxycarbonylalkyl; alkoxycarbonylalkoxy; heterocyclylalkyl; heterocyclyloxy; heterocyclylalkoxy; heterocyclylalkoxyalkyl; heterocyclyloxyalkyl; cycloalkyloxy; —OC(O)SR7; —OC(O)OR7; —C(O)OR7; —C(O)SR7; —C(S)OR7; —C(S)SR7; aminoalkyl which may be substituted by at least one substituent selected from alkyl, cyano, cyanoalkyl, (alkylthio)carbonylalkyl, alkyl(thiocarbonyl)alkyl, —C(O)OR7 and —C(O)SR7; or 4,5-dihydroisoxazol-3-yl which may be substituted by R9, R6 is haloalkyl; halogen; nitro; cyano; alkylthio; alkylsulfinyl; or alkylsulfonyl, R7 is alkyl; haloalkyl; alkoxyalkyl; alkenyl; haloalkenyl; alkynyl; or arylalkyl which may be substituted by R10, and each of R8, R9 and R10 which are independent of one another, is halogen; alkyl; or alkoxy.

公开(公告)号：US08030498B2

公开(公告)日：2011-10-04

申请号：US12094734

申请日：2006-12-13

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： C07D231/20 ,  A61K31/415

CPC分类号： C07D231/20 ,  C07D405/12 ,  C07D413/12

摘要： A benzoylpyrazole compound represented by the formula (I) or its salt, useful as herbicides and intermediates thereof.

摘要翻译： 由式（I）表示的苯甲酰基吡唑化合物或其盐，可用作除草剂及其中间体。

公开(公告)号：US20090286683A1

公开(公告)日：2009-11-19

申请号：US12094734

申请日：2006-12-13

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： A01N43/56 ,  C07D231/18 ,  C07D405/10 ,  A01P13/00

CPC分类号： C07D231/20 ,  C07D405/12 ,  C07D413/12

摘要： A benzoylpyrazole compound represented by the formula (I) or its salt, useful as herbicides and intermediates thereof.

摘要翻译： 由式（I）表示的苯甲酰基吡唑化合物或其盐，可用作除草剂及其中间体。

公开(公告)号：US08466088B2

公开(公告)日：2013-06-18

申请号：US12525554

申请日：2008-02-01

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： A01N63/00

CPC分类号： A01N43/56 ,  A01N33/18 ,  A01N37/20 ,  A01N37/22 ,  A01N37/36 ,  A01N37/40 ,  A01N39/04 ,  A01N41/10 ,  A01N43/10 ,  A01N43/40 ,  A01N43/653 ,  A01N43/70 ,  A01N43/707 ,  A01N43/80 ,  A01N43/82 ,  A01N43/88 ,  A01N47/06 ,  A01N47/30 ,  A01N47/36 ,  A01N57/20 ,  A01N2300/00

摘要： Provided is an herbicidal composition which can be applied at a low dose as compared with individual application, and thus is effective to reduce the environmental load on a place where the composition is applied or a periphery thereof, of which the herbicidal spectrum is enlarged, and of which the herbicidal effects last over a long period of time. The herbicidal composition has as active ingredients (a) a herbicidal benzoylpyrazole compound represented by the formula (I) or its salt: wherein Q is —C(O)SR3 or a hydrogen atom, R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is alkyl, cycloalkyl or the like, R4 is alkyl, haloalkyl or the like, R5 is a hydrogen atom, alkyl or the like, R6 is haloalkyl, halogen or the like, and (b) a further herbicidal compound.

摘要翻译： 本发明提供了与单独使用相比可以以低剂量施用的除草组合物，因此有效地降低施用组合物的地方或其周边，增加除草频谱的环境负荷，以及 其除草效果持续很长时间。 除草组合物具有（a）式（I）表示的除草酰苯并吡唑化合物或其盐：其中Q为-C（O）SR 3或氢原子，R 1为烷基或环烷基，R 2为氢原子 或烷基，R 3是烷基，环烷基等，R 4是烷基，卤代烷基等，R 5是氢原子，烷基等，R 6是卤代烷基，卤素等，和（b）另外的除草化合物。

公开(公告)号：US20100099563A1

公开(公告)日：2010-04-22

申请号：US12525554

申请日：2008-02-01

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： A01N43/56 ,  A01N43/66 ,  A01N43/40

CPC分类号： A01N43/56 ,  A01N33/18 ,  A01N37/20 ,  A01N37/22 ,  A01N37/36 ,  A01N37/40 ,  A01N39/04 ,  A01N41/10 ,  A01N43/10 ,  A01N43/40 ,  A01N43/653 ,  A01N43/70 ,  A01N43/707 ,  A01N43/80 ,  A01N43/82 ,  A01N43/88 ,  A01N47/06 ,  A01N47/30 ,  A01N47/36 ,  A01N57/20 ,  A01N2300/00

摘要： To provide a herbicidal composition which can be applied at a low dose as compared with individual application, and thus is effective to reduce the environmental load on a place where the composition is applied or a periphery thereof, of which the herbicidal spectrum is enlarged, and of which the herbicidal effects last over a long period of time.A herbicidal composition which comprises as active ingredients (a) a herbicidal benzoylpyrazole compound represented by the formula (I) or its salt: wherein Q is —C(O)SR3 or a hydrogen atom, R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is alkyl, cycloalkyl or the like, R4 is alkyl, haloalkyl or the like, R5 is a hydrogen atom, alkyl or the like, R6 is haloalkyl, halogen or the like, and (b) other herbicidal compound.

摘要翻译： 提供与单独施用相比可以以低剂量施用的除草组合物，因此有效地减少施用组合物的地方或其周边，其除草频谱扩大的环境负荷，以及 其除草效果持续很长时间。 一种除草组合物，其包含作为活性成分的（a）由式（I）表示的除草酰苯并吡唑化合物或其盐：其中Q为-C（O）SR 3或氢原子，R 1为烷基或环烷基，R 2为氢 原子或烷基，R3是烷基，环烷基等，R4是烷基，卤代烷基等，R5是氢原子，烷基等，R6是卤代烷基，卤素等，和（b）其它除草化合物。