公开(公告)号：US06441044B1

公开(公告)日：2002-08-27

申请号：US09763685

申请日：2001-02-26

申请人： Ingo Rose ,  Frank Wetterich ,  Karl Eicken ,  Joachim Rheinheimer ,  Gisela Lorenz ,  Eberhard Ammermann ,  Thomas Grote ,  Siegfried Strathmann

发明人： Ingo Rose ,  Frank Wetterich ,  Karl Eicken ,  Joachim Rheinheimer ,  Gisela Lorenz ,  Eberhard Ammermann ,  Thomas Grote ,  Siegfried Strathmann

IPC分类号： A01N3718

CPC分类号： A01N53/00 ,  C07C233/58 ,  C07C255/48 ,  C07C271/24 ,  C07C2601/02

摘要： The present invention relates to cycloalkylcarboxamides of formula I where: A is optionally substituted C3-C6-cycloalkyl; Alk is straight-chain or branched C1-C6-alkylene; R1 is optionally substituted C1-C6-alkyl or C2-C6-alkenyl; R2, R3 is hydrogen, or is optionally halogenated C1-C6-alkyl or C2-C6-alkenyl; W is an optionally substituted fused bicyclic ring system having in each case six ring atoms, where one or two carbon ring atoms may be replaced by nitrogen atoms; and their agriculturally useful salts. Furthermore, the invention relates to fungicidal compositions comprising a compound of formula I as crop protection agent.

摘要翻译： 本发明涉及式I的环烷基甲酰胺，其中：A为任选取代的C 3 -C 6 - 环烷基; Alk为直链或支链C 1 -C 6亚烷基; R 1为任选取代的C 1 -C 6 - 烷基或C 2 -C 6 - 烯基; R 2 ，R 3是氢，或任选被卤代的C 1 -C 6 - 烷基或C 2 -C 6 - 烯基; W是任选取代的稠合双环体系，其各自为六个环原子，其中一个或两个碳环原子可被氮取代 原子及其农业上有用的盐。此外，本发明涉及杀真菌组合物，其包含式I化合物作为作物保护剂。

公开(公告)号：US20050187265A1

公开(公告)日：2005-08-25

申请号：US11061470

申请日：2005-02-22

申请人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： A61P31/10 ,  A01N37/52 ,  A61K31/165 ,  C07C259/14 ,  C07D333/22 ,  A61K31/381 ,  A61K31/415 ,  A61K31/44 ,  C07C259/10

CPC分类号： C07C259/14 ,  A01N37/52 ,  C07C2601/02

摘要： Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described. In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1-C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1-C6-alkyl, thienyl-C1-C4-alkyl, or pyrazolyl-C1-C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy, C1-C6-alkylcarbonyl; n is 0-5; p is, depending on the number of free valencies, 0-4.

摘要翻译： 描述了新的苯甲酰胺肟衍生物，其制备方法和中间体及其作为杀真菌剂的用途。 在本发明的上下文中，苯甲酰胺肟衍生物是式I的化合物，其中：A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基，其中一个碳可被氧，氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基 ，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基，噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基，R 3 - （CH 3）3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 - 烷基，C 1 - C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基 C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基，C 1 -C 4烷基硫基，C 1 -C 4 - -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量，0-4。

公开(公告)号：US06919485B2

公开(公告)日：2005-07-19

申请号：US10469688

申请日：2002-03-09

申请人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Norbert Götz ,  Karl Eicken ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Norbert Götz ,  Karl Eicken ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N35/04 ,  C07C45/46 ,  C07C49/84 ,  C07C45/00 ,  A01N35/00

CPC分类号： C07C49/84 ,  A01N35/04 ,  C07C45/46

摘要： The invention relates to benzophenones of formula (I), in which the substituents have the following meanings: X represents halogen; R1 represents hydrogen, halogen, C1-C6 alkyl, halo-C1-C2 alkyl, C1-C4 alkoxy, oxyhalomethyl or nitro, and; R2 represents hydrogen, C1-C6 alkyl, benzyl, cyclohexylmethyl or C3-C6 alkenyl. The invention also relates to the production of these benzophenones and to their use as fungicides

摘要翻译： 本发明涉及式（I）的二苯甲酮，其中取代基具有以下含义：X表示卤素; R 1表示氢，卤素，C 1 -C 6烷基，卤代C 1 -C 3 烷基，C 1 -C 4烷氧基，氧卤甲基或硝基，和; R 2表示氢，C 1 -C 6烷基，苄基，环己基甲基或C 3 -C 3 > 6个烯基。 本发明还涉及这些二苯甲酮的制备及其作为杀真菌剂的用途

公开(公告)号：US06476061B1

公开(公告)日：2002-11-05

申请号：US09831406

申请日：2001-05-09

申请人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Gerhard Hamprecht

发明人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Gerhard Hamprecht

IPC分类号： A61N4336

CPC分类号： C07D207/50 ,  A01N43/36

摘要： The invention relates to fungicides containing compounds of formula (I) as their active agents, the radicals in said formula (I) having the following meanings: R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-halogenalkylcarbonyl; R2 is hydrogen, C1-C6-alkyl or C1-C6-halogenalkyl; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, C1-C6-halogenalkyl, C1-C6-alkoxy, C1-C6-halogenalkoxy, C1-C6-alkylsulfonyl, C1-C6-halogenalkylsulfonyl, formyl, cyano, C1-C6-alkylthio or phenyl which can optionally be substituted by halogen atoms, C1-C6-alkyl or C1-C6-halogenalkyl groups, and to their agriculturally usable salts. The invention also relates to methods for combating fungi in plants using these fungicides.

摘要翻译： 本发明涉及含有式（I）化合物作为其活性剂的杀真菌剂，所述式（I）中的基团具有以下含义：R 1是氢，C 1 -C 6 - 烷基，C 1 -C 6 - 烷基羰基，甲酰基或C 1 -C 6烷基， C6-卤代烷基羰基; R2是氢，C1-C6-烷基或C1-C6-卤代烷基; R3-R12是氢，卤素，C1-C8-环烷基，C1-C6-烷基，C1-C6-卤代烷基，C1-C6-烷氧基，C1-C6-卤代烷氧基，C1-C6-烷基磺酰基，C1-C6-卤代烷基磺酰基， 甲酰基，氰基，C 1 -C 6 - 烷硫基或可以被卤素原子，C 1 -C 6烷基或C 1 -C 6 - 卤代烷基取代的苯基，以及它们的农业上可用的盐。 本发明还涉及使用这些杀真菌剂防治植物中真菌的方法。

公开(公告)号：US06680283B1

公开(公告)日：2004-01-20

申请号：US10410788

申请日：2003-04-11

申请人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： A01N4336

CPC分类号： A01N43/36 ,  A01N37/32 ,  A01N37/36 ,  A01N37/38 ,  A01N41/02 ,  A01N41/10 ,  C07D207/50

摘要： Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I where R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl; R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl, R13 is hydrogen, C1-C6-alkyl, R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen, and their agriculturally useful salts are described.

摘要翻译： 具有杀真菌作用的农药组合物包含作为活性化合物的式I其中R 1为氢，C 1 -C 6烷基，C 1 -C 6烷基羰基，甲酰基或C 1 -C 6卤代烷基羰基; R 2为卤素， C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基， C 6 - 烷基亚磺酰基，卤代-C 1 -C 6 - 烷基磺酰基，氰基或基团NR 13 R 14; R 3 -R 12是氢，卤素，C 1 -C 8 - 环烷基，C 1 -C 6 - 烷基 卤代-C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，卤代-C 1 -C 6 - 烷氧基，C 1 -C 6烷基磺酰基，卤代-C 1 -C 6烷基磺酰基，甲酰基，C 1 -C 6烷基羰基，氰基，C 1 -C 6 - 烷硫基或苯基，其可以是未取代的或被卤素，C 1 -C 6 - 烷基或卤代-C 1 -C 6烷基取代，R 13是氢，C 1 -C 6烷基，R 14是C 1 -C 6 - 烷基，C 1 -C 8 - 环烷基或与R 13和它们所连接的氮原子一起是饱和或不饱和的杂环五元或六元环，其含有一个或两个选自以下的杂原子： 描述了由氮和氧组成的组及其农业上有用的盐。

公开(公告)号：US07101900B2

公开(公告)日：2006-09-05

申请号：US11061470

申请日：2005-02-22

申请人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： A61K31/15 ,  A61K31/381 ,  C07D213/44 ,  C07D333/20 ,  C07D251/158

CPC分类号： C07C259/14 ,  A01N37/52 ,  C07C2601/02

摘要： Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described.In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1–C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1–C6-alkyl, thienyl-C1–C4-alkyl, or pyrazolyl-C1–C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy, C1–C6-alkylcarbonyl; n is 0–5; p is, depending on the number of free valencies, 0–4.

摘要翻译： 描述了新的苯甲酰胺肟衍生物，其制备方法和中间体及其作为杀真菌剂的用途。 在本发明的上下文中，苯甲酰胺肟衍生物是式I的化合物，其中：A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基，其中一个碳可被氧，氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基 ，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基，噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基，R 3 - （CH 3）3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 - 烷基，C 1 - C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 3 > 4个 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - - 烷氧基烷氧基，C 1 -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量，0-4。

公开(公告)号：US06881742B1

公开(公告)日：2005-04-19

申请号：US10089148

申请日：2000-10-05

申请人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： A61P31/10 ,  A01N37/52 ,  A61K31/165 ,  C07C259/14 ,  A01N43/10 ,  A01N33/08 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  C07D213/44 ,  C07D213/78 ,  C07D231/14 ,  C07D239/28 ,  C07D277/30

CPC分类号： C07C259/14 ,  A01N37/52 ,  C07C2601/02

摘要： Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described.In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1-C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1-C6-alkyl, thienyl-C1-C4-alkyl, or pyrazolyl-C1-C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy, C1-C6-alkylcarbonyl; n is 0-5; p is, depending on the number of free valencies, 0-4.

摘要翻译： 描述了新的苯甲酰胺肟衍生物，其制备方法和中间体及其作为杀真菌剂的用途。 在本发明的上下文中，苯甲酰胺肟衍生物是式I的化合物，其中：A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基，其中一个碳可被氧，氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基 ，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基，噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基，R 3 - （CH 3）3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 - 烷基，C 1 - C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 3 > 4个 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - - 烷氧基烷氧基，C 1 -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量，0-4。

公开(公告)号：US06586369B1

公开(公告)日：2003-07-01

申请号：US10204349

申请日：2002-08-20

申请人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Joachim Rheinheimer ,  Karl Eicken ,  Ingo Rose ,  Thomas Grote ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： C07D20718

CPC分类号： C07D207/50 ,  A01N37/32 ,  A01N37/36 ,  A01N37/38 ,  A01N41/02 ,  A01N41/10 ,  A01N43/36

摘要： Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I where R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl; R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl, R13 is hydrogen, C1-C6-alkyl, R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen, and their agriculturally useful salts are described.

摘要翻译： 具有杀真菌作用的农药组合物，包含作为活性化合物的式I化合物，其中R 1是氢，C 1 -C 6烷基，C 1 -C 6烷基羰基，甲酰基或C 1 -C 6卤代烷基羰基; R 2是卤素，C 1 -C 6烷硫基， C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6 - 烷基亚磺酰基， C 1 -C 6 - 烷基磺酰基，氰基或NR 13 R 14基; R 3 -R 12是氢，卤素，C 1 -C 8 - 环烷基，C 1 -C 6烷基，卤代-C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基， C 1 -C 6 - 烷基磺酰基，卤代-C 1 -C 6 - 烷基磺酰基，甲酰基，C 1 -C 6 - 烷基羰基，氰基，C 1 -C 6 - 烷硫基或苯基，其可以是未取代的或被卤素取代， 或卤代-C 1 -C 6烷基，R 13是氢，C 1 -C 6烷基，R 14是C 1 -C 6 - 烷基，C 1 -C 8 - 环烷基，或者与R 13和它们所连接的氮原子一起是饱和或 不饱和杂环五元或六元环，其含有一个或两个选自组的杂原子 描述了氮和氧及其农业上有用的盐。

公开(公告)号：US06680402B2

公开(公告)日：2004-01-20

申请号：US10261122

申请日：2002-10-01

申请人： Karl Eicken ,  Joachim Rheinheimer ,  Frank Wetterich ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Karl Eicken ,  Joachim Rheinheimer ,  Frank Wetterich ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： C07C25549

CPC分类号： C07D333/24 ,  A01N37/52 ,  A01N43/10 ,  A01N43/56 ,  C07C255/53 ,  C07C255/54 ,  C07C259/18

摘要： Benzamidoxime derivatives of the formula I: where R1 is difluoromethyl or trifluoromethyl R2 is hydrogen or fluorine R3 is C1-C4-alkyl which may be substituted by cyano, C1-C4-haloalkyl, C1-C4-alkoxy-C1-C4-alkyl, C3-C6-alkenyl, C3-C6-haloalkenyl, C3-C6-alkynyl, C3-C8-cycloalkyl-C1-C4-alkyl R4 is phenyl-C1-C6-alkyl which may carry one or more substitutents selected from the group consisting of halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy and C1-C4-haloalkoxy on the phenyl ring, or is thienyl-C1-C4-alkyl which may carry one or more substituents selected from the group consisting of halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy and C1-C4-haloalkoxy on the thienyl ring, or is pyrazolyl-C1-C4-alkyl which may carry one or more substituents selected from the group consisting of halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy and C1-C4-haloalkoxy on the pyrazole ring, are prepared, and intermediates for their preparation and their use as fungicides are described.

摘要翻译： 式I的苯甲酰胺肟衍生物：其中R 1是二氟甲基或三氟甲基R 2是氢或氟，R 3是可以被氰基，C 1 -C 4卤代烷基，C 1 -C 4 - 烷氧基 - C 1 -C 4 - 烷基，C 3 -C 6 - 烯基，C 3 -C 6 - 卤代烯基，C 3 -C 6 - 炔基，C 3 -C 8 - 环烷基-C 1 -C 4 - 烷基R 4是苯基-C 1 -C 6 - 或更多的选自苯基环上的卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 烷氧基和C 1 -C 4 - 卤代烷氧基的取代基，可以携带的噻吩基-C 1 -C 4烷基 一个或多个选自噻吩基环上的卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 烷氧基和C 1 -C 4 - 卤代烷氧基的取代基，其可以是吡唑基-C 1 -C 4烷基， 在吡唑环上携带一个或多个选自卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 烷氧基和C 1 -C 4 - 卤代烷氧基的取代基，制备中间体和 描述了它们作为杀真菌剂的用途。

公开(公告)号：US06509501B2

公开(公告)日：2003-01-21

申请号：US10093634

申请日：2002-03-11

申请人： Karl Eicken ,  Joachim Rheinheimer ,  Frank Wetterich ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Karl Eicken ,  Joachim Rheinheimer ,  Frank Wetterich ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： C07C25148

CPC分类号： C07D333/24 ,  A01N37/52 ,  A01N43/10 ,  A01N43/56 ,  C07C255/53 ,  C07C255/54 ,  C07C259/18

摘要： Benzamidoxime derivatives of the formula I where R1 is difluoromethyl or trifluoromethyl R2 is hydrogen or fluorine R3 is C1-C4-alkyl which may be substituted by cyano, C1-C4-haloalkyl, C1-C4-alkoxy-C1-C4-alkyl, C3-C6-alkenyl, C3-C6-haloalkenyl, C3-C6-alkynyl, C3-C8-cycloalkyl-C1-C4-alkyl R4 is phenyl-C1-C6-alkyl which may carry one or more substitutents selected from the group consisting of halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy and C1-C4-haloalkoxy on the phenyl ring, or is thienyl-C1-C4-alkyl which may carry one or more substituents selected from the group consisting of halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy and C1-C4-haloalkoxy on the thienyl ring, or is pyrazolyl-C1-C4-alkyl which may carry one or more substituents selected from the group consisting of halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy and C1-C4-haloalkoxy on the pyrazole ring, are prepared, and intermediates for their preparation and their use as fungicides are described.

摘要翻译： 式I的苯甲酰胺肟衍生物，其中R 1是二氟甲基或三氟甲基，R 2是氢或氟，R 3是可被氰基，C 1 -C 4卤代烷基，C 1 -C 4 - 烷氧基-C 1 -C 4 - 烷基，C 3 -C 6 - 烯基 ，C 3 -C 6 - 卤代链烯基，C 3 -C 6 - 炔基，C 3 -C 8 - 环烷基-C 1 -C 4 - 烷基基团R 4是苯基-C 1 -C 6 - 烷基，其可以带有一个或多个选自卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 烷氧基和C 1 -C 4 - 卤代烷氧基，可以带有一个或多个选自卤素，C 1 -C 4 - 在噻吩环上的C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 烷氧基和C 1 -C 4 - 卤代烷氧基，可以带有一个或多个选自卤素，C 1 -C 4 - C 1-4 - 烷基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 烷氧基和C 1 -C 4 - 卤代烷氧基，并且描述了制备中间体及其作为杀真菌剂的用途。