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公开(公告)号:US4847289A
公开(公告)日:1989-07-11
申请号:US59084
申请日:1987-06-08
申请人: John J. Baldwin , Charles M. Habecker , Samuel L. Graham , Wasyl Halczenko , George D. Hartman , Harvey Schwam , Gerald S. Ponticello , Kenneth L. Shepard
发明人: John J. Baldwin , Charles M. Habecker , Samuel L. Graham , Wasyl Halczenko , George D. Hartman , Harvey Schwam , Gerald S. Ponticello , Kenneth L. Shepard
IPC分类号: A61K31/38 , A61K31/381 , A61P9/12 , A61P27/02 , A61P27/06 , C07D333/34 , C07D409/12
CPC分类号: C07D409/12 , C07D333/34
摘要: Aryl (or aralkyl)-sulfonylthiophene-2-sulfonamides containing a basic functional group as a substituent are efficacious in the treatment of elevated intraocular pressure and glaucoma following topical ocular administration.