2-substituted pyrimidines
    5.
    发明授权
    2-substituted pyrimidines 失效
    2-取代的嘧啶

    公开(公告)号:US07488732B2

    公开(公告)日:2009-02-10

    申请号:US10549936

    申请日:2004-03-30

    摘要: 2-Substituted pyrimidines of the formula I in which the index n and the substituents L, Ra, Rb, Rc, Rz, Ru, Rv, A′, A″ and A′″ are as defined in the description and: R1 is C3-C10-alkyl, C3-C10-alkenyl, C3-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S, R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl, and R3 is cyano, CO2Ra, C(═O)NRzRb, C(═O)—N—ORb, C(═S)—NRaRb, C(═NORa)NRzRb, C(═NRa)NRzRb, C(═O)NRa—NRzRb, C(═N—NRzRc)NRaRb, C(═O)Ra, C(═NORb)Ra, C(═N—NRzRb)Ra, CRaRb—ORz, CRaRb—NRzRc, ON(═CRaRb), O—C(═O)Ra, NRaRb′, NRa(C(═O)Rb), NRa(C(═O)ORb), NRa(C(═O)—NRzRb), NRa(C(═NRc)Rb), NRa(N═CRcRb), NRa—NRzRb, NRz—ORa, NRa(C(═NRc)—NRzRb), NRa(C(═NORc)Rb), processes for preparing these compounds, compositions comprising these compounds and their pesticidal use are described.

    摘要翻译: 其中指数n和取代基L,Ra,Rb,Rc,Rz,Ru,Rv,A',A“和A”'如说明书中所定义的式I的2-取代的嘧啶:R1 C 3 -C 10 - 烷基,C 3 -C 10 - 烯基,C 3 -C 10 - 炔基,C 3 -C 12 - 环烷基,C 3 -C 10 - 环烯基或五至十元饱和的部分不饱和或芳族杂环,其通过碳 并且含有一至四个由O,N和S组成的组的杂原子,R2是卤素,氰基,C1-C4-烷基,C2-C4-烯基,C2-C4-炔基,C1-C4-烷氧基,C3-C4 - 烯氧基或C 3 -C 4 - 炔氧基,其中R 2的烷基,烯基和炔基可以被卤素,氰基,硝基,C 1 -C 2 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代,并且R 3是氰基,CO 2 R a,C( -O)NR z R b,C(-O)-N-OR b,C(-S)-NR a R b,C(-NOR a)NR z R b,C(-NR a)NR z R b,C(O)NR a -NR b R b,C -NRaRb,C(-O)Ra,C(-NORb)Ra,C(-N-NRzRb)Ra,CRaRb-ORz,CRaRb-NRzRc,ON(-CRaRb),OC(-O)Ra,NRaRb ,NR a(C(-O)R b),NR a(C(-O)R b),NR a(C(-O)OR b) NRa-N RzRb,NRz-ORa,NRa(C(-NRc)-NRzRb),NRa(C(-NORc)Rb),制备这些化合物的方法,包含这些化合物的组合物及其杀虫剂用途。

    2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi
    8.
    发明授权
    2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi 失效
    2-(2-吡啶基)-5-苯基-6-氨基嘧啶,用于生产和用于对抗有害真菌的方法和中间产物

    公开(公告)号:US07320975B2

    公开(公告)日:2008-01-22

    申请号:US10505146

    申请日:2003-02-06

    IPC分类号: C07D401/04 A01N43/54

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(2-pyridyl)-5-phenyl-6-aminopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants

    摘要翻译: 本发明涉及式I的2-(2-吡啶基)-5-苯基-6-氨基嘧啶,其中取代基和指数具有以下含义:R 1表示卤素,羟基,杂环基, 烷氧基,烷氧基羰基,氨基甲酰基,烷基氨基羰基,二烷基氨基羰基,吗啉代羰基,吡咯烷基羰基,烷基羰基氨基,烷基氨基。 二烷基氨基,烷硫基,烷基亚磺酰基,烷基磺酰基,羟基磺酰基,氨基磺酰基,烷基氨基磺酰基,二烷基氨基磺酰基; m = 0或1-4; R 2表示氢,卤素,氰基,烷基,卤代烷基或烷氧基; R 3,R 4表示氢,烷基,卤代烷基,环烷基,卤代烷基,烯基,卤代烯基,环烯基,炔基,卤代炔基或环炔基,R 3 O 和R 4与它们连接的氮原子一起形成5或6元环,其被来自基团O,N或S的原子和/或可被取代 根据说明; R 5表示卤素,烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7,R 8表示氢,卤素,烷基或卤代烷基; R 9表示氢,卤素,羟基,氰基,烷基,烷氧基,环烷氧基,卤代烷氧基,烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物,除了其用于对抗不期望的植物之外