摘要:
Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2′ and R3′, R2′, R3′ are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要:
The invention relates to fungicidal mixtures, containing the following in a synergistically effective quantity as active components: 1) the triazolopyrimidine derivative of formula (I); and 2) a phenylamidine derivative of formula (II), in which the variables are defined as follows: R1, R4, R5 represent alkyl, alkenyl or alkynyl; R2, R3 represent cyano, alkyl, alkenyl, alkynyl, alkoxy, alkoxyalkyl, benzyloxy or alkylcarbonyl; m represents 0 or 1; A represents a direct bond, —O—, —S—, NRd, CHRe or —O—CHRe; R6 represents phenyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing between one and four heteroatoms from the group comprising O, N or S, whereby the groups can be substituted according to the description. The invention also relates to a method for controlling pathogenic fungi using mixtures of compounds (I) and (II), to the use of compounds (I) and (II) for producing mixtures of this type and to agents that contain said mixtures.
摘要翻译:本发明涉及杀真菌混合物,其具有协同有效量作为活性成分:1)式(I)的三唑并嘧啶衍生物; 和2)式(II)的苯基脒衍生物,其中变量定义如下:R 1,R 4,R 5, 代表烷基,烯基或炔基; R 2,R 3代表氰基,烷基,烯基,炔基,烷氧基,烷氧基烷基,苄氧基或烷基羰基; m表示0或1; A表示直接键,-O-,-S-,NR d,CHR e或-O-CHR e; R 6表示苯基或五元或六元饱和,部分不饱和或芳族杂环,其含有一个至四个来自O,N或S的基团的杂原子,其中基团可以根据 的描述。 本发明还涉及使用化合物(I)和(II)的混合物来控制致病真菌的方法,用于制备这种类型的混合物和含有所述混合物的试剂的化合物(I)和(II)。
摘要:
The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; L1, L2, L3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译:本发明涉及式I的6-(2,4,6-三卤代苯基)三唑并嘧啶,其中取代基如下:R 1是烷基,卤代烷基,环烷基,卤代环烷基,烯基, 卤代烯基,环烯基,卤代环烯基,炔基,卤代炔基或苯基,萘基或五或六元饱和的部分不饱和或芳族杂环,其含有一至四个由O,N和S组成的组的杂原子,R 2 R 1是氢或R 1,R 2和R 2中所提及的基团之一,与它们的氮原子一起 还可以形成通过N连接的五元或六元杂环基或杂芳基,并且可以含有一个至三个其它由O,N和S组成的组的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; L 1,L 2,L 3 3是氯或氟,其中至少一个基团是氯; X是氰基,烷基,烷氧基,烯氧基,卤代烷氧基或卤代烯氧基; 制备这些化合物的方法,包含它们的组合物及其用于控制植物病原性有害真菌的用途。
摘要:
6-(2-Halo-4-alkoxyphenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, phenylalkyl, mono- or dialkoxyalkyl; R1, R2 and/or R3 may be substituted as mentioned in the description; L is hydrogen, fluorine or chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译:其中取代基如下定义的式I的6-(2-卤代-4-烷氧基苯基)三唑并嘧啶:R 1是烷基,卤代烷基,环烷基,卤代环烷基,烯基,卤代烯基,环烯基,卤代环烯基 ,炔基,卤代炔基或苯基,萘基或五元或六元饱和的部分不饱和或芳族杂环,其含有一至四个由O,N和S组成的组的杂原子,R 2, 是氢或R 1,R 1和R 2所提及的基团之一与它们所连接的氮原子一起也可以 形成通过N连接的五元或六元杂环基或杂芳基,并且可以含有一个至三个由O,N和S组成的组的另外的杂原子作为环成员; R 3是烷基,卤代烷基,烯基,卤代烯基,炔基,卤代炔基,苯基烷基,单或二烷氧基烷基; R 1,R 2和/或R 3可以如说明书中所述被取代; L是氢,氟或氯; X是氰基,烷基,烷氧基,烯氧基,卤代烷氧基或卤代烯氧基; 制备这些化合物的方法,包含它们的组合物及其用于控制植物病原性有害真菌的用途。
摘要:
The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R2 represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R1 and/or R2 being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.
摘要翻译:本发明涉及式(I)的5,6-二烷基-7-氨基 - 三唑并嘧啶,其中取代基定义如下:R 1表示烷基,烷氧基烷基,烯基或炔基; R 2表示根据描述被取代的烷基,烷氧基烷基,烯基或炔基,R 1和/或R 2 2。 本发明还涉及一种生产所述化合物的方法,含有后者的药剂及其用于控制植物致病真菌的用途。
摘要:
Fungicidal mixtures, comprising, as active components, 1) a sulfamoyl compound of the formula I, in which the substituents are as defined below: R1 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, alkylthio, alkoxycarbonyl, phenyl, benzyl, formyl or CH═NOA; A is hydrogen, alkyl, alkylcarbonyl; R2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxycarbonyl; R3 is halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, alkylthio, alkoxycarbonyl, formyl or CH═NOA; n is 0, 1, 2, 3 or 4; R4 is hydrogen, halogen, cyano, alkyl or haloalkyl; and 2) at least one active compound selected from the following groups: A) azoles; B) strobilurins; C) acylalanines; D) amine derivatives; E) anilinopyrimidines; F) dicarboximides; G) cinnamides and analogs; H) dithiocarbamates; I) heterocylic compounds; K) sulfur and copper fungicides; L) nitrophenyl derivatives; M) phenylpyrroles; N) sulfenic acid derivatives; O) other fungicides; according to the description; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of a compound I with active compounds of groups A) to O) and the use of the compounds I with active compounds of groups A) to O) for preparing such mixtures, and also compositions comprising these mixtures.
摘要翻译:作为活性组分的杀真菌混合物,1)式I的氨磺酰基化合物,其中取代基如下:R 1是氢,卤素,氰基,烷基,卤代烷基,烷氧基, 烷硫基,烷氧基羰基,苯基,苄基,甲酰基或CH-NOA; A是氢,烷基,烷基羰基; R 2是氢,卤素,氰基,烷基,卤代烷基,烷氧基羰基; R 3是卤素,氰基,硝基,烷基,卤代烷基,烷氧基,烷硫基,烷氧基羰基,甲酰基或CH-NOA; n为0,1,2,3或4; R 4是氢,卤素,氰基,烷基或卤代烷基; 和2)至少一种选自以下组的活性化合物:A)唑类; B)嗜球果伞素 C)酰基丙氨酸; D)胺衍生物; E)苯胺嘧啶嘧啶; F)二羧酰亚胺; G)肉桂酸酯类似物; H)二硫代氨基甲酸盐; I)杂环化合物; K)硫和铜杀菌剂; L)硝基苯基衍生物; M)苯基吡咯; N)亚磺酸衍生物; O)其他杀菌剂; 根据说明; 协同有效量的方法,使用化合物I与基团A)至O)的活性化合物的混合物控制有害真菌的方法,以及将化合物I与基团A)至O)的活性化合物用于制备此类混合物的用途,以及 也包含这些混合物的组合物
摘要:
Fungicidal mixtures comprising, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) the benzamide of the formula II in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with the compound II and the use of the compound I with the compound II for preparing such mixtures, and also compositions comprising these mixtures.
摘要:
The invention relates to 6-(2,3,6-trifluorophenyl)-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R2 represents hydrogen or one of the groups cited for R1; R1 and R2, together with the nitrogen atom, to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded via N and can contain one to three additional heteroatoms from the groups O, N and S as a ring member; R1 and/or R2 can be substituted in accordance with the description; X represents cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy. The invention also relates to methods for producing said compounds, to agents containing the latter and to their use for combating plant-pathogenic fungi.
摘要翻译:本发明涉及式(I)的6-(2,3,6-三氟苯基) - 三唑并嘧啶,其中取代基定义如下:R 1表示烷基,卤代烷基,环烷基,卤代环烷基, 烯基,卤代烯基,环烯基,卤代环烯基,炔基,卤代炔基或苯基,萘基或含有一至四个O,N或S基的杂原子的五元或六元饱和的部分不饱和或芳族杂环; R 2表示氢或R 1所引用的基团之一; R 1和R 2与它们所键合的氮原子一起也可以形成五或六元杂环基或杂芳基,其通过 并且可以含有一个至三个作为环成员的来自基团O,N和S的另外的杂原子; R 1和/或R 2可以根据描述代替; X表示氰基,烷基,烷氧基,烯氧基,卤代烷氧基或卤代烯氧基。 本发明还涉及生产所述化合物的方法,含有后者的试剂和用于对抗植物致病性真菌的用途。
摘要:
6-(2,4,6-Trifluorophenyl)triazolopyrimidines of the formula I in which the substituents have the following meanings: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl, cycloalkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned in R1, R1 and R2 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered ring which is interrupted by an atom from the group consisting of O, N and S, and/or R1 and/or R2 can be substituted according to the description; X is cyano, C1-C4-alkoxy, C3-C4-alkenyloxy, C1-C2-haloalkoxy or C3-C4-halo-alkenyloxy; process for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.
摘要:
The invention relates to 7-aminomethyl-1,2,4-triazolo[1,5-a]pyrimidine compounds of general formula (I) and the agriculturally compatible salts of said compounds. In said formula: R1 and R2 represent hydrogen, alkyl, haloalkyl, alkoxy, cycloalkyl, bicycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1 to 4 heteroatoms from the group containing O, N or S, or R1 and R2, together with the nitrogen atom to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded by means of N and can contain 1 to 3 additional heteroatoms from the group containing O, N and S as the ring member and can be substituted according to the description; R3 and R4 represent hydrogen, alkyl, haloalkyl, haloalkoxy, alkoxy, or alkoxyalkyl; X represents halogen, cyano, a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1, 2 or 3 heteroatoms from the group containing O, N or S as the ring member, alkyl, alkoxy, alkenyl or alkynyl, whereby the latter 4 groups can be substituted according to the description; L is defined as cited in the claims and the description; and m represents 0, 1, 2, 3, 4 or 5. The invention also relates to the use of the triazolopyrimidine compounds of general formula (I) and their agriculturally compatible salts for controlling plant-pathogenic fungi, to a method for controlling plant-pathogenic fungi, containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound and at least one liquid or solid carrier.