公开(公告)号：US4026940A

公开(公告)日：1977-05-31

申请号：US624285

申请日：1975-10-20

申请人： Keiichi Sugimoto ,  Koji Nishijima ,  Hiroshi Akimoto ,  Tadashi Hanaoka ,  Nobuharu Kakeya

发明人： Keiichi Sugimoto ,  Koji Nishijima ,  Hiroshi Akimoto ,  Tadashi Hanaoka ,  Nobuharu Kakeya

IPC分类号： C07C309/70 ,  C07D307/12 ,  C07C143/68

CPC分类号： C07C309/70 ,  C07D307/12

摘要： .alpha.-Sulfophenylacetic acid derivatives of the general formula: ##STR1## (wherein R is a substituted or unsubstituted primary alcohol, cyclic alcohol or phenol compound residue), which are of value as intermediates of antibacterial agents, are selectively produced in a high yield by bringing a diester compound of the general formula: ##STR2## (wherein R has the same meaning as defined above) into contact with a strong acid.

摘要翻译： 通过以下方式选择性地制备具有下列通式的α-磺基苯乙酸衍生物：其中R为取代或未取代的伯醇，环醇或酚化合物残基）作为抗菌剂的中间体，以高产率由 得到通式如下的二酯化合物：其中R与上述定义相同）与强酸接触。

公开(公告)号：US4057544A

公开(公告)日：1977-11-08

申请号：US417527

申请日：1973-11-20

申请人： Keiichi Sugimoto ,  Koji Nishijima ,  Hiroshi Akimoto ,  Tadashi Hanaoka ,  Nobuharu Kakeya

发明人： Keiichi Sugimoto ,  Koji Nishijima ,  Hiroshi Akimoto ,  Tadashi Hanaoka ,  Nobuharu Kakeya

IPC分类号： C07D499/12 ,  A61K31/43 ,  A61P31/04 ,  C07D207/08 ,  C07D307/12 ,  C07D499/62 ,  C07D499/68 ,  C07D499/46

CPC分类号： C07D307/12 ,  C07D207/08

摘要： Novel penicillins of the formula ##STR1## wherein R is a branched chain alkyl group of from 3 to 14 carbon atoms, and their pharmaceutically acceptable salts, are easily absorbed in the blood and tissues through oral administration and show excellent antimicrobial activity against Gram-positive and Gram-negative bacteria, particularly against microorganisms of the genus Pseudomonas, such as Pseudomonas aeruginosa.

摘要翻译： 其中R为3〜14个碳原子的支链烷基及其药学上可接受的盐的新型青霉素通过口服给药容易地吸收在血液和组织中，并显示出优异的抗革兰氏阳性的抗微生物活性 和革兰氏阴性细菌，特别是针对假单胞菌属（Pseudomonas）的微生物，如铜绿假单胞菌（Pseudomonas aeruginosa）。

公开(公告)号：US4048158A

公开(公告)日：1977-09-13

申请号：US645913

申请日：1975-12-31

申请人： Keiichi Sugimoto ,  Koji Nishijima ,  Tadashi Hanaoka ,  Hiroshi Akimoto ,  Nobuharu Kakeya

发明人： Keiichi Sugimoto ,  Koji Nishijima ,  Tadashi Hanaoka ,  Hiroshi Akimoto ,  Nobuharu Kakeya

IPC分类号： C07D499/04 ,  C07D499/00 ,  C07D499/62

CPC分类号： C07D499/00

摘要： Novel d-.alpha.-isobutylsulfobenzylpenicillin hemi-solvate crystals of the formula: ##STR1## (wherein A is a solvent selected from the class consisting of alcohols, ketones, ethers and esters) have excellent antibacterial activities and improved stability in terms of shelf-life.

摘要翻译： 下式的新型d-α-异丁基磺苄青霉素半溶剂化物晶体：其中A是选自醇，酮，醚和酯的溶剂，具有优异的抗菌活性和改善保质期的稳定性 。

公开(公告)号：US3954826A

公开(公告)日：1976-05-04

申请号：US486835

申请日：1974-07-09

申请人： Keiichi Sugimoto ,  Koji Nishijima ,  Hiroshi Akimoto ,  Tadashi Hanaoka ,  Nobuharu Kakeya

发明人： Keiichi Sugimoto ,  Koji Nishijima ,  Hiroshi Akimoto ,  Tadashi Hanaoka ,  Nobuharu Kakeya

IPC分类号： C07C309/03 ,  C07C309/73 ,  C07D207/08 ,  C07D307/12 ,  C07D499/62 ,  C07C143/68

CPC分类号： C07D207/08 ,  C07C309/00 ,  C07D307/12

摘要： .alpha.-Sulfophenylacetic acid derivatives of the general formula: ##EQU1## (wherein R is a substituted or unsubsituted primary alcohol, cyclic alcohol or phenol compound residue), which are of value as intermediates of antibacterial agents, are selectively produced in a high yield by bringing a diester compound of the general formula: ##EQU2## (wherein R has the same meaning as defined above) into contact with a strong acid.

摘要翻译： 选择性地以高产率制备具有通式为-CHCOOH | SO 3 R（其中R为取代或未取代的伯醇，环醇或酚化合物残基）的α-磺基苯乙酸衍生物，其为抗菌剂的中间体 通过将具有通式：CH 3 | -CHCOO-C-CH 3 || SO 3 R CH 3（其中R具有与上述相同的含义）的二酯化合物与强酸接触。

公开(公告)号：US07766661B2

公开(公告)日：2010-08-03

申请号：US12211300

申请日：2008-09-16

申请人： Akira Kuwahara ,  Takuya Takahashi ,  Seiya Takahashi ,  Hiroshi Akimoto ,  Hiroshi Endo ,  Yoshiaki Ishiyama

发明人： Akira Kuwahara ,  Takuya Takahashi ,  Seiya Takahashi ,  Hiroshi Akimoto ,  Hiroshi Endo ,  Yoshiaki Ishiyama

IPC分类号： H01R9/09

CPC分类号： H05K1/0204 ,  F21K9/00 ,  F21V29/70 ,  F21V29/74 ,  H01L23/3735 ,  H01L23/3737 ,  H01L23/433 ,  H01L2924/0002 ,  H05K3/0061 ,  H05K2201/0133 ,  H05K2201/10106 ,  H01L2924/00

摘要： A heat transfer member which is capable of enhancing efficiency of heat dissipation, and a connector including the heat transfer member. On the surface of an elastic body arranged between an LED and a heat sink, a heat conduction metal thin film that transfers heat generated in the LED to the heat sink is formed. The member may also include an electrical conduction metal film, whereby the member may serve as both a heat transfer member and as an electrical connector.

摘要翻译： 能够提高散热效率的传热构件和包括传热构件的连接器。 在布置在LED和散热器之间的弹性体的表面上，形成将LED中产生的热量传递到散热器的导热金属薄膜。 该构件还可以包括导电金属膜，由此该构件可以用作传热构件和电连接器两者。

公开(公告)号：US07209591B2

公开(公告)日：2007-04-24

申请号：US10620879

申请日：2003-07-15

申请人： Hiroshi Akimoto ,  Oleksandr V. Monastyrskyi

发明人： Hiroshi Akimoto ,  Oleksandr V. Monastyrskyi

IPC分类号： G06K9/36 ,  H04N5/228 ,  H04B1/66

CPC分类号： H04N19/184 ,  H04N19/51 ,  H04N19/93

摘要： A method for motion accounting and compensation while encoding allows improvement of the restored image quality. Image is a predicted frame in video sequence. Motion compensation is understood as an error residual signal compressing scheme, executed during video sequence encoding. According to the teachings of the current invention, errors are accounted for during encoding. Error accounting is subtracting the original image from the predicted frame. The error values are written to the output stream compactly with the minimum code length. The stored error values are added to the predicted frame during the decoding process. The method taught herein is applied for all the predicted frames from the video sequence, thereby allowing one to improve the quality of decompressed video film that was compressed with a significant compression ratio.

摘要翻译： 一种用于编码时运动记帐和补偿的方法可以提高恢复的图像质量。 图像是视频序列中的预测帧。 运动补偿被理解为在视频序列编码期间执行的误差残差信号压缩方案。 根据本发明的教导，在编码期间考虑到错误。 错误计费是从预测帧中减去原始图像。 错误值以最小代码长度紧凑地写入输出流。 存储的误差值在解码过程中被添加到预测帧。 本文教导的方法适用于来自视频序列的所有预测帧，从而允许以提高压缩比压缩的解压缩视频胶片的质量。

公开(公告)号：US07080451B2

公开(公告)日：2006-07-25

申请号：US10723102

申请日：2003-11-26

申请人： Kazuhisa Saito ,  Asuka Hosoda ,  Hiroshi Akimoto

发明人： Kazuhisa Saito ,  Asuka Hosoda ,  Hiroshi Akimoto

IPC分类号： H01R43/16

CPC分类号： H01R4/028 ,  H05K3/3426 ,  H05K3/3447 ,  Y02P70/613 ,  Y10T29/49204 ,  Y10T29/49211 ,  Y10T29/49224 ,  Y10T29/5193

摘要： A method of manufacturing an electronic component with a contact having a terminal section for brazing and a contact section includes steps that construct a contact base member of a material that is poorly wettable, forms a primer plating layer of a material that is poorly wettable to the weld brazing material on the base member, forms a finish plating layer of a material that is highly wettable to the weld brazing material on the primer plating layer, and selectively removes a portion of the finish plating layer to obtain an exposed region of the primer plating layer that serves as an arresting region for arresting the weld brazing material from creeping up and migrating along the highly wettable finish plating layer in brazing the terminal section to the brazing pad of a wiring board.

摘要翻译： 一种制造具有用于钎焊的端子部分的接触件的电子部件的方法和接触部分包括构建不良润湿性材料的接触基底部件的步骤，形成不良润湿性的材料的底漆镀层 焊接钎焊材料形成在底涂层上的焊接钎焊材料高度可润湿的材料的精加工镀层，并且选择性地除去精整镀层的一部分以获得底镀层的暴露区域 作为用于阻止焊接钎料的爬行区域的阻挡区域，在钎焊终端部分到布线板的钎焊焊盘的同时沿着高度可润湿的精加工镀层迁移。

公开(公告)号：US06702624B2

公开(公告)日：2004-03-09

申请号：US09274859

申请日：1999-03-23

申请人： Hiroshi Akimoto ,  Katsumi Arai ,  Katsuma Ushijima ,  Takahiro Abe

发明人： Hiroshi Akimoto ,  Katsumi Arai ,  Katsuma Ushijima ,  Takahiro Abe

IPC分类号： H01R1700

CPC分类号： H01R12/57 ,  H01L23/057 ,  H01L23/49861 ,  H01L2924/0002 ,  H01R12/716 ,  H01R43/24 ,  H01L2924/00

摘要： An electronic component has an insert member embedded in a resin portion by an insert molding method, with a part of the insert member exposed at an outer surface of the resin portion. At least a part of the exposed portion of the insert member is depressed relative to the outer surface of the resin portion.

摘要翻译： 电子部件具有通过插入成型方法嵌入在树脂部中的插入部件，插入部件的一部分露出在树脂部的外表面。 插入构件的暴露部分的至少一部分相对于树脂部分的外表面被压下。

公开(公告)号：US5223620A

公开(公告)日：1993-06-29

申请号：US830884

申请日：1992-02-04

申请人： Hiroaki Nomura ,  Hiroshi Akimoto ,  Tetsuo Miwa

发明人： Hiroaki Nomura ,  Hiroshi Akimoto ,  Tetsuo Miwa

IPC分类号： C07D239/95 ,  C07D471/04

CPC分类号： C07D471/04 ,  C07D239/95

摘要： New fused pyrimidines of the general formula (I): ##STR1## wherein the ring A is a pyridine ring which may be hydrogenated or a benzene ring which may be hydrogenated, X is an amino group or a hydroxyl group, R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are independently hydrogen, fluorine or a lower alkyl group, and --COOR.sup.5 and --COOR.sup.6 are independently a carboxyl group which may be esterified, and salts thereof have excellent anti-tumor effects, and they can be produced by the following reaction scheme: ##STR2## in which A is, X, R.sup.1 to R.sup.4, --COOR.sup.5 have the above meanings.

摘要翻译： 通式（I）的新的稠合嘧啶：其中环+ E，crc / A /是可被氢化的吡啶环或可被氢化的苯环，X是氨基或 羟基，R1，R2，R3和R4独立地是氢，氟或低级烷基，-COOR5和-COOR6独立地是可被酯化的羧基，其盐具有优异的抗肿瘤效果，并且它们 可以通过以下反应方案制备：其中+ E，crc / A / is，X，R 1至R 4，-COOR 5具有上述含义的 + TR 。

公开(公告)号：US4946846A

公开(公告)日：1990-08-07

申请号：US329374

申请日：1989-03-27

申请人： Hiroaki Nomura ,  Hiroshi Akimoto ,  Tetsuo Miwa

发明人： Hiroaki Nomura ,  Hiroshi Akimoto ,  Tetsuo Miwa

IPC分类号： A61K31/505 ,  A61K31/517 ,  A61P35/00 ,  C07D239/95 ,  C07D471/04

CPC分类号： C07D471/04 ,  C07D239/95

摘要： New fused pyrimidines of the general formula (I): ##STR1## wherein the ring .circle. A is a pyridine ring which may be hydrogenated or a benzene ring which may be hydrogenated, X is an amino group or a hydroxyl group, R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are independently hydrogen, fluorine or a lower alkyl group, and --COOR.sup.5 and --COOR.sup.6 are independently a carboxyl group which may be esterified, and salts thereof have excellent anti-tumor effects, and they can be produced by the following reaction scheme: ##STR2## in which .circle. A is, X, R.sup.1 to R.sup.4, --COOR.sup.5 have the above meanings.