-
公开(公告)号:US20100144730A1
公开(公告)日:2010-06-10
申请号:US12307104
申请日:2007-07-02
申请人: Kenneth Egnard Lind , Kathy Cao , Edward Yin-shiang Lin , Thinh Ba Nguyen , Bradley T. Tangonan , Daniel A. Erlanson , Kevin Guckian , Robert Lowell Simmons , Wen-cherng Lee , Lihong Sun , Stig Hansen , Nuzhat Pathan , Lei Zhang
发明人: Kenneth Egnard Lind , Kathy Cao , Edward Yin-shiang Lin , Thinh Ba Nguyen , Bradley T. Tangonan , Daniel A. Erlanson , Kevin Guckian , Robert Lowell Simmons , Wen-cherng Lee , Lihong Sun , Stig Hansen , Nuzhat Pathan , Lei Zhang
IPC分类号: A61K31/437 , C07D471/04 , C07D487/04 , C07D413/14 , A61K31/519 , A61K31/5377 , A61P35/00
CPC分类号: C07D471/04 , A61K31/4412 , A61K31/443 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4985 , A61K31/506 , A61K31/519 , A61K31/5377 , C07D211/86 , C07D213/64 , C07D401/12 , C07D401/14 , C07D405/12 , C07D405/14 , C07D407/14 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07D487/04
摘要: The present invention provides pyridinonyl PDK1 inhibitors and methods of treating cancer using the same.
摘要翻译: 本发明提供吡啶基PDK1抑制剂和使用其制备癌症的方法。
-
公开(公告)号:US08778977B2
公开(公告)日:2014-07-15
申请号:US12307104
申请日:2007-07-02
申请人: Kenneth Egnard Lind , Kathy Cao , Edward Yin-shiang Lin , Thinh Ba Nguyen , Bradley T. Tangonan , Daniel A. Erlanson , Kevin Guckian , Robert Lowell Simmons , Wen-cherng Lee , Lihong Sun , Stig Hansen , Nuzhat Pathan , Lei Zhang
发明人: Kenneth Egnard Lind , Kathy Cao , Edward Yin-shiang Lin , Thinh Ba Nguyen , Bradley T. Tangonan , Daniel A. Erlanson , Kevin Guckian , Robert Lowell Simmons , Wen-cherng Lee , Lihong Sun , Stig Hansen , Nuzhat Pathan , Lei Zhang
IPC分类号: A61K31/5377 , A61K31/506 , A61K31/519 , A61K31/4985 , A61K31/444 , A61K31/4439 , A61K31/4436 , A61K31/443 , A61K31/4412 , C07D487/04 , C07D471/04 , C07D417/14 , C07D417/12 , C07D413/14 , C07D413/12 , C07D409/14 , C07D409/12 , C07D405/14 , C07D405/12 , C07D401/14 , C07D401/12 , C07D211/86
CPC分类号: C07D471/04 , A61K31/4412 , A61K31/443 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4985 , A61K31/506 , A61K31/519 , A61K31/5377 , C07D211/86 , C07D213/64 , C07D401/12 , C07D401/14 , C07D405/12 , C07D405/14 , C07D407/14 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07D487/04
摘要: The present invention provides pyridinonyl PDK1 inhibitors and methods of treating cancer using the same.
摘要翻译: 本发明提供吡啶基PDK1抑制剂和使用其制备癌症的方法。
-
公开(公告)号:US20100256092A1
公开(公告)日:2010-10-07
申请号:US12464829
申请日:2009-05-12
申请人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Vincent S. Hernandez , Jacob J. Plattner , Charles Z. Ding , Kathy Cao , Yong-Kang Zhang , Andrew Benowitz , Tsutomu Akama , Jessica Sligar , Guofeng Jia , Ligong Ou , Neerja Saraswat , Sreekanth Ramachandran , Chris Diaper , Yanchen Zhang , Goverdhan Reddy Banda , James A. Nieman , Mehdi Keramane , Rahim Mohammed , Rajendra Subedi , Hong Liang , Rajeshwar Singh
发明人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Vincent S. Hernandez , Jacob J. Plattner , Charles Z. Ding , Kathy Cao , Yong-Kang Zhang , Andrew Benowitz , Tsutomu Akama , Jessica Sligar , Guofeng Jia , Ligong Ou , Neerja Saraswat , Sreekanth Ramachandran , Chris Diaper , Yanchen Zhang , Goverdhan Reddy Banda , James A. Nieman , Mehdi Keramane , Rahim Mohammed , Rajendra Subedi , Hong Liang , Rajeshwar Singh
CPC分类号: A61K31/33 , A61K31/43 , A61K45/06 , C07F5/025 , Y02A50/401 , Y02A50/411 , A61K2300/00
摘要: This invention relates to, among other items, 6-substituted benzoxaborole compounds and their use for treating bacterial infections.
摘要翻译: 本发明涉及6-取代的苯并恶唑化合物及其用于治疗细菌感染的用途。
-
公开(公告)号:US08343944B2
公开(公告)日:2013-01-01
申请号:US12844748
申请日:2010-07-27
申请人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
发明人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
CPC分类号: C07F5/025 , A61K31/69 , A61K45/06 , A61K2300/00
摘要: This invention largely relates to 3,4,6-trisubstituted benzoxaborole compounds, and their use for treating bacterial infections.
摘要翻译: 本发明主要涉及3,4,6-三取代苯并恶唑化合物及其用于治疗细菌感染的用途。
-
公开(公告)号:US20110136763A1
公开(公告)日:2011-06-09
申请号:US12844748
申请日:2010-07-27
申请人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
发明人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
CPC分类号: C07F5/025 , A61K31/69 , A61K45/06 , A61K2300/00
摘要: This invention largely relates to 3,4,6-trisubstituted benzoxaborole compounds, and their use for treating bacterial infections.
摘要翻译: 本发明主要涉及3,4,6-三取代苯并恶唑化合物及其用于治疗细菌感染的用途。
-
-
-
-