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    PROCESS FOR PREPARING 3-[(4S)-8-BROMO-1-METHYL-6-(2-PYRIDINYL)-4H-IMIDAZO[1,2-A][1,4]BENZODIAZEPINE-4-YL]PROPIONIC ACID METHYL ESTER OR THE BENZENE SULFONATE SALT THEREOF, AND COMPOUNDS USEFUL IN THAT PROCESS
    9.
    发明申请
    PROCESS FOR PREPARING 3-[(4S)-8-BROMO-1-METHYL-6-(2-PYRIDINYL)-4H-IMIDAZO[1,2-A][1,4]BENZODIAZEPINE-4-YL]PROPIONIC ACID METHYL ESTER OR THE BENZENE SULFONATE SALT THEREOF, AND COMPOUNDS USEFUL IN THAT PROCESS 有权
    制备3 - [（4S）-8-溴-1-甲基-6-（2-吡啶基）-4H-咪唑并[1,2-A] [1,4]苯并噻吩并[4-y]]丙酸甲酯的方法 ESTER或其中的苯甲磺酸盐及其用途的化合物

    公开(公告)号：US20150368199A1

    公开(公告)日：2015-12-24

    申请号：US14841899

    申请日：2015-09-01

    申请人： Gary Stuart Tilbrook ,  Andreas Schumacher ,  Rene Emmenegger

    发明人： Gary Stuart Tilbrook ,  Andreas Schumacher ,  Rene Emmenegger

    IPC分类号： C07D213/50

    CPC分类号： C07D401/04 ,  C07D213/40 ,  C07D213/50 ,  C07D487/04 ,  C07F9/65586

    摘要： The invention concerns a new process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4H-imidazo[1,2-a][1,4]benzodiazepine-4-yl]-propionic acid methyl ester or 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4H-imidazo[1,2-a][1,4]benzodiazepine-4-yl]propionic acid methyl ester benzene sulfonate (P) which comprises reacting 3-[(S)-7-bromo-2-((R and/or S)-2-hydroxy-propylamino)-5-pyridin-2-yl-3H-benzo[e][1,4]diazepin-3-yl]-propionic acid methyl ester of formula (EM) with an oxidizing agent and optionally treating the reaction product under acidic conditions, such as to produce the compound of formula (F) or the compound (P), and new compounds useful as starting material or as intermediate for performing that process.

    摘要翻译： 本发明涉及一种制备3 - [（4S）-8-溴-1-甲基-6-（2-吡啶基）-4H-咪唑并[1,2-a] [1,4]苯并二氮杂- 吡啶-3-基] - 丙酸甲酯或3 - [（4S）-8-溴-1-甲基-6-（2-吡啶基）-4H-咪唑并〔1,2-a〕〔1,4〕苯并二氮杂-4- 吡啶-2-基]丙酸甲酯苯磺酸盐（P），其包括使3 - [（S）-7-溴-2 - （（R和/或S）-2-羟基 - 丙基氨基） -3H-苯并[e] [1,4]二氮杂-3-基] - 丙酸甲酯与氧化剂反应，并在酸性条件下任选地处理反应产物，例如制备式 （F）或化合物（P），以及可用作原料的新化合物或用于进行该方法的中间体。

    POWER SWITCH FOR PREVENTING ACCIDENTAL ARCS
    10.
    发明申请
    POWER SWITCH FOR PREVENTING ACCIDENTAL ARCS 有权
    用于防止意外ARCS的电源开关

    公开(公告)号：US20100214724A1

    公开(公告)日：2010-08-26

    申请号：US12599224

    申请日：2008-05-09

    申请人： Samuel Dahl ,  Andreas Schumacher ,  Wolfgang Wagner

    发明人： Samuel Dahl ,  Andreas Schumacher ,  Wolfgang Wagner

    IPC分类号： H02B1/00

    CPC分类号： H02H1/0023 ,  H02H3/023 ,  H02H3/08

    摘要： A power switch disposed in a housing includes a contact breaker configured to connect and disconnect a low-voltage switchgear from a power source supplying the low-voltage switchgear, a triggering device configured to disconnect the low-voltage switchgear in an overload event, a current detection device, a control device, a first evaluation device configured to evaluate an accidental arc overcurrent, and a second evaluation device configured to evaluate the accidental arc overcurrent. The power switch is configured to be activated via an overcurrent signal generated by an arc monitoring system in response to the accidental arc overcurrent. The overcurrent signal is linked to the at least one triggering signal. The second evaluation has a threshold above a threshold of the first evaluation device. The triggering device is configured to be activated via a turn-off pulse when a signal from the current detection device is above the threshold of the second evaluation device.

    摘要翻译： 设置在壳体中的电源开关包括接触断路器，其被配置为将低压开关设备与供应低压开关设备的电源连接和断开;触发装置，其被配置为在过载事件中断开低压开关设备，电流 检测装置，控制装置，被配置为评估意外的过电流的第一评估装置，以及被配置为评估意外的电弧过电流的第二评估装置。 电源开关被配置为通过由电弧监视系统响应于意外的电弧过电流而产生的过电流信号而被激活。 过电流信号与至少一个触发信号相连。 第二评估具有高于第一评估装置的阈值的阈值。 触发装置被配置为当来自当前检测装置的信号高于第二评估装置的阈值时通过关断脉冲被激活。