Polymorph form II of tanaproget
    1.
    发明授权
    Polymorph form II of tanaproget 失效
    tanaproget的多晶型II

    公开(公告)号:US08114869B2

    公开(公告)日:2012-02-14

    申请号:US13106494

    申请日:2011-05-12

    摘要: Tanaproget polymorph Form II, processes for preparing tanaproget polymorph Form II, pharmaceutical compositions including tanaproget polymorph Form II, micronized tanaproget polymorph Form II, and processes for converting Form II to tanaproget Form I are provided. Also provided are methods of contraception, hormone replacement therapy, stimulation of food intake and treating or preventing uterine myometrial fibroids, benign prostatic hypertrophy, benign and malignant neoplastic disease, dysfunctional bleeding, uterine leiomyomata, endometriosis, polycystic ovary syndrome, or carcinomas and adenocarcinomas comprising administering polymorph Form II to a mammalian subject.

    摘要翻译: Tanaproget多晶型物II,制备tanaproget多晶型II的方法,包括tanaproget多晶型II,微粉化tanaproget多晶型II的药物组合物,以及将II型转化成tanaproget形式I的方法。 还提供了避孕,激素替代疗法,刺激食物摄取和治疗或预防子宫肌层肌瘤,良性前列腺肥大,良性和恶性肿瘤性疾病,功能障碍性出血,子宫平滑肌瘤,子宫内膜异位症,多囊卵巢综合征或癌和腺癌的方法,包括 向哺乳动物受试者施用多晶型II。

    Polymorph Form II of Tanaproget
    2.
    发明申请
    Polymorph Form II of Tanaproget 失效
    Tanaproget的多晶型II型

    公开(公告)号:US20110212953A1

    公开(公告)日:2011-09-01

    申请号:US13106494

    申请日:2011-05-12

    摘要: Tanaproget polymorph Form II, processes for preparing tanaproget polymorph Form II, pharmaceutical compositions including tanaproget polymorph Form II, micronized tanaproget polymorph Form II, and processes for converting Form II to tanaproget Form I are provided. Also provided are methods of contraception, hormone replacement therapy, stimulation of food intake and treating or preventing uterine myometrial fibroids, benign prostatic hypertrophy, benign and malignant neoplastic disease, dysfunctional bleeding, uterine leiomyomata, endometriosis, polycystic ovary syndrome, or carcinomas and adenocarcinomas comprising administering polymorph Form II to a mammalian subject.

    摘要翻译: Tanaproget多晶型物II,制备tanaproget多晶型II的方法,包括tanaproget多晶型II,微粉化tanaproget多晶型II的药物组合物,以及将II型转化成tanaproget形式I的方法。 还提供了避孕,激素替代疗法,刺激食物摄取和治疗或预防子宫肌层肌瘤,良性前列腺肥大,良性和恶性肿瘤性疾病,功能障碍性出血,子宫平滑肌瘤,子宫内膜异位症,多囊卵巢综合征或癌和腺癌的方法,包括 向哺乳动物受试者施用多晶型II。

    Process for preparing polymorph form II of tanaproget
    3.
    发明授权
    Process for preparing polymorph form II of tanaproget 有权
    制备tanaproget多晶型II的方法

    公开(公告)号:US07968709B2

    公开(公告)日:2011-06-28

    申请号:US12792978

    申请日:2010-06-03

    IPC分类号: C07D265/18

    摘要: Tanaproget polymorph Form II, processes for preparing tanaproget polymorph Form II, pharmaceutical compositions including tanaproget polymorph Form II, micronized tanaproget polymorph Form II, and processes for converting Form II to tanaproget Form I are provided. Also provided are methods of contraception, hormone replacement therapy, stimulation of food intake and treating or preventing uterine myometrial fibroids, benign prostatic hypertrophy, benign and malignant neoplastic disease, dysfunctional bleeding, uterine leiomyomata, endometriosis, polycystic ovary syndrome, or carcinomas and adenocarcinomas comprising administering polymorph Form II to a mammalian subject.

    摘要翻译: Tanaproget多晶型物II,制备tanaproget多晶型II的方法,包括tanaproget多晶型II,微粉化tanaproget多晶型II的药物组合物,以及将II型转化成tanaproget形式I的方法。 还提供了避孕,激素替代疗法,刺激食物摄取和治疗或预防子宫肌层肌瘤,良性前列腺肥大,良性和恶性肿瘤性疾病,功能障碍性出血,子宫平滑肌瘤,子宫内膜异位症,多囊卵巢综合征或癌和腺癌的方法,包括 向哺乳动物受试者施用多晶型II。

    Polymorph form II of tanaproget
    4.
    发明授权
    Polymorph form II of tanaproget 失效
    tanaproget的多晶型II

    公开(公告)号:US07759341B2

    公开(公告)日:2010-07-20

    申请号:US11412015

    申请日:2006-04-26

    IPC分类号: A61K31/536

    摘要: Tanaproget polymorph Form II, processes for preparing tanaproget polymorph Form II, pharmaceutical compositions including tanaproget polymorph Form II, micronized tanaproget polymorph Form II, and processes for converting Form II to tanaproget Form I are provided. Also provided are methods of contraception, hormone replacement therapy, stimulation of food intake and treating or preventing uterine myometrial fibroids, benign prostatic hypertrophy, benign and malignant neoplastic disease, dysfunctional bleeding, uterine leiomyomata, endometriosis, polycystic ovary syndrome, or carcinomas and adenocarcinomas comprising administering polymorph Form II to a mammalian subject.

    摘要翻译: Tanaproget多晶型物II,制备tanaproget多晶型II的方法,包括tanaproget多晶型II,微粉化tanaproget多晶型II的药物组合物,以及将II型转化成tanaproget形式I的方法。 还提供了避孕,激素替代疗法,刺激食物摄取和治疗或预防子宫肌层肌瘤,良性前列腺肥大,良性和恶性肿瘤性疾病,功能障碍性出血,子宫平滑肌瘤,子宫内膜异位症,多囊卵巢综合征或癌和腺癌的方法,包括 向哺乳动物受试者施用多晶型II。

    Polymorph Form II of Tanaproget
    5.
    发明申请
    Polymorph Form II of Tanaproget 审中-公开
    Tanaproget的多晶型II型

    公开(公告)号:US20120115858A1

    公开(公告)日:2012-05-10

    申请号:US13347080

    申请日:2012-01-10

    摘要: Tanaproget polymorph Form II, processes for preparing tanaproget polymorph Form II, pharmaceutical compositions including tanaproget polymorph Form II, micronized tanaproget polymorph Form II, and processes for converting Form II to tanaproget Form I are provided. Also provided are methods of contraception, hormone replacement therapy, stimulation of food intake and treating or preventing uterine myometrial fibroids, benign prostatic hypertrophy, benign and malignant neoplastic disease, dysfunctional bleeding, uterine leiomyomata, endometriosis, polycystic ovary syndrome, or carcinomas and adenocarcinomas comprising administering polymorph Form II to a mammalian subject.

    摘要翻译: Tanaproget多晶型物II,制备tanaproget多晶型II的方法,包括tanaproget多晶型II,微粉化tanaproget多晶型II的药物组合物,以及将II型转化成tanaproget形式I的方法。 还提供了避孕,激素替代疗法,刺激食物摄取和治疗或预防子宫肌层肌瘤,良性前列腺肥大,良性和恶性肿瘤性疾病,功能障碍性出血,子宫平滑肌瘤,子宫内膜异位症,多囊卵巢综合征或癌和腺癌的方法,包括 向哺乳动物受试者施用多晶型II。

    Polymorph Form II of Tanaproget
    6.
    发明申请
    Polymorph Form II of Tanaproget 有权
    Tanaproget的多晶型II型

    公开(公告)号:US20100267715A1

    公开(公告)日:2010-10-21

    申请号:US12792978

    申请日:2010-06-03

    摘要: Tanaproget polymorph Form II, processes for preparing tanaproget polymorph Form II, pharmaceutical compositions including tanaproget polymorph Form II, micronized tanaproget polymorph Form II, and processes for converting Form II to tanaproget Form I are provided. Also provided are methods of contraception, hormone replacement therapy, stimulation of food intake and treating or preventing uterine myometrial fibroids, benign prostatic hypertrophy, benign and malignant neoplastic disease, dysfunctional bleeding, uterine leiomyomata, endometriosis, polycystic ovary syndrome, or carcinomas and adenocarcinomas comprising administering polymorph Form II to a mammalian subject.

    摘要翻译: Tanaproget多晶型物II,制备tanaproget多晶型II的方法,包括tanaproget多晶型II,微粉化tanaproget多晶型II的药物组合物,以及将II型转化成tanaproget形式I的方法。 还提供了避孕,激素替代疗法,刺激食物摄取和治疗或预防子宫肌层肌瘤,良性前列腺肥大,良性和恶性肿瘤性疾病,功能障碍性出血,子宫平滑肌瘤,子宫内膜异位症,多囊卵巢综合征或癌和腺癌的方法,包括 向哺乳动物受试者施用多晶型II。

    Mirror
    8.
    外观设计
    Mirror 有权

    公开(公告)号:USD950965S1

    公开(公告)日:2022-05-10

    申请号:US29720973

    申请日:2020-01-16

    申请人: Yan Xu

    设计人: Yan Xu