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公开(公告)号:US20140243370A1
公开(公告)日:2014-08-28
申请号:US14131471
申请日:2012-08-22
IPC分类号: A61K31/4439 , A61K31/429 , A61K31/454 , C07D513/04
CPC分类号: C07D513/04 , A61K31/429 , A61K31/4439 , A61K31/454
摘要: Novel compounds of formula (I) wherein R1 to R4 and X have the meaning according to the claims, are glucosidase inhibitors, and can be employed, inter alia, for the treatment of Alzheimer's disease.
摘要翻译: 式(I)的新化合物,其中R 1至R 4和X具有权利要求所述的含义,其为葡糖苷酶抑制剂,并且可用于治疗阿尔茨海默氏病。
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公开(公告)号:US10138233B2
公开(公告)日:2018-11-27
申请号:US14900215
申请日:2014-06-24
申请人: Merck Patent GmbH , Henry Yu , Thomas E. Richardson , Marianne Donnelly , Ngan Nguyen , Xuliang Jiang
IPC分类号: C07D471/04 , C07D498/04 , C07D493/14 , C07D471/02 , C07D498/14
摘要: The present invention relates to imidazole compounds, and pharmaceutically acceptable compositions thereof, useful as positive allosteric modulators of follicle stimulating hormone receptor (FSHR).
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公开(公告)号:US10081637B2
公开(公告)日:2018-09-25
申请号:US14900209
申请日:2014-06-24
申请人: MERCK PATENT GMBH , Henry Yu , Marianne Donnelly , Ngan Nguyen , Xuliang Jiang
发明人: Henry Yu , Marianne Donnelly , Ngan Nguyen , Xuliang Jiang
IPC分类号: C07D491/052
CPC分类号: C07D491/052
摘要: The present invention relates to pyrazole compounds, and pharmaceutically acceptable compositions thereof, useful as positive allosteric modulators of follicle stimulating hormone receptor (FSHR).
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