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公开(公告)号:US07470705B2
公开(公告)日:2008-12-30
申请号:US10598473
申请日:2005-03-17
申请人: Michael Gregory Bell , Guoqing Cao , Ana Maria Escribano , Maria Carmen Fernandez , Peter Ambrose Lander , Nathan Bryan Mantlo , Eva Maria Martin de la Nava , Ana Isabel Mateo Herranz , Daniel Ray Mayhugh , Xiaodong Wang
发明人: Michael Gregory Bell , Guoqing Cao , Ana Maria Escribano , Maria Carmen Fernandez , Peter Ambrose Lander , Nathan Bryan Mantlo , Eva Maria Martin de la Nava , Ana Isabel Mateo Herranz , Daniel Ray Mayhugh , Xiaodong Wang
IPC分类号: A01N43/42 , A61K31/44 , C07D471/02
CPC分类号: C07D495/04 , C07D471/04 , C07D487/04
摘要: The present invention discloses compounds of formula (I) wherein A, n, q, K, W, X, Y; Z, R1, R2, R3, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed as useful for treating dyslipidemia and its sequelae.
摘要翻译: 本发明公开了式(I)的化合物,其中A,n,q,K,W,X,Y; Z,R 1,R 2,R 3,R 4,R 5和R 6如本文所定义,其药物组合物和使用方法被公开用于治疗血脂障碍及其后遗症。
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公开(公告)号:US07749992B2
公开(公告)日:2010-07-06
申请号:US10574649
申请日:2004-10-07
申请人: Guoqing Cao , Ana Maria Escribano , Maria Carmen Fernandez , Todd Fields , Douglas Linn Gernert , Christopher Lawrence Cioffi , Robert Jason Herr , Nathan Bryan Mantlo , Eva Maria Martin De La Nava , Ana Isabel Mateo Herranz , Daniel Ray Mayhugh , Xiaodong Wang
发明人: Guoqing Cao , Ana Maria Escribano , Maria Carmen Fernandez , Todd Fields , Douglas Linn Gernert , Christopher Lawrence Cioffi , Robert Jason Herr , Nathan Bryan Mantlo , Eva Maria Martin De La Nava , Ana Isabel Mateo Herranz , Daniel Ray Mayhugh , Xiaodong Wang
IPC分类号: A61P3/06 , A61P9/10 , A61K31/55 , C07D223/14 , C07D223/16 , C07D223/32 , C07D225/06 , C07D403/04 , C07D403/12 , C07D405/06 , C07D405/12 , C07D413/04 , C07D491/04
CPC分类号: C07D223/16 , C07D223/14 , C07D223/32 , C07D225/06 , C07D403/04 , C07D403/12 , C07D405/06 , C07D405/12 , C07D413/04 , C07D491/04
摘要: Compounds of formula I wherein n, m, p, q, y, R1 R2, R3, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed as useful for treating artherosclerosis and its sequelae.
摘要翻译: 其中n,m,p,q,y,R 1,R 2,R 3,R 4,R 5和R 6如本文所定义的式I化合物,其药物组合物和使用方法被公开用于治疗动脉粥样硬化及其后遗症。
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公开(公告)号:US20070173526A1
公开(公告)日:2007-07-26
申请号:US10598473
申请日:2005-03-17
申请人: Michael Bell , Guoqing Cao , Ana Escribano , Maria Fernandez , Peter Lander , Nathan Mantlo , Eva Martin de la Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiaodong Wang
发明人: Michael Bell , Guoqing Cao , Ana Escribano , Maria Fernandez , Peter Lander , Nathan Mantlo , Eva Martin de la Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiaodong Wang
IPC分类号: A61K31/4745 , A61K31/4743 , C07D498/02 , C07D471/02
CPC分类号: C07D495/04 , C07D471/04 , C07D487/04
摘要: The present invention discloses compounds of formula (I) wherein A, n, q, K, W, X, Y; Z, R1, R2, R3, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed as useful for treating dyslipidemia and its sequelae.
摘要翻译: 本发明公开了式(I)的化合物,其中A,n,q,K,W,X,Y; Z,R 1,R 2,R 3,R 4,R 5,..., >和R 6'如本文所定义,并且其药物组合物和使用方法被公开用于治疗血脂异常及其后遗症。
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公开(公告)号:US20070254869A1
公开(公告)日:2007-11-01
申请号:US10574649
申请日:2004-10-07
申请人: Guoqing Cao , Ana Escribano , Maria Fernandez , Todd Fields , Douglas Gernert , Christopher Cioffi , Robert Herr , Nathan Mantlo , Eva Martin De La Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiaodong Wang
发明人: Guoqing Cao , Ana Escribano , Maria Fernandez , Todd Fields , Douglas Gernert , Christopher Cioffi , Robert Herr , Nathan Mantlo , Eva Martin De La Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiaodong Wang
IPC分类号: A61K31/55 , A61P9/10 , C07D223/14 , C07D223/16
CPC分类号: C07D223/16 , C07D223/14 , C07D223/32 , C07D225/06 , C07D403/04 , C07D403/12 , C07D405/06 , C07D405/12 , C07D413/04 , C07D491/04
摘要: Compounds of formula I wherein n, m, p, q, y, R1 R2, R3, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed as useful for treating artherosclerosis and its sequelae.
摘要翻译: 其中n,m,p,q,y,R 1,R 2,R 3,R 4, R 5,R 5和R 6如本文所定义,并且它们的药物组合物和使用方法被公开用于治疗动脉粥样硬化及其后遗症。
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公开(公告)号:US20070208003A1
公开(公告)日:2007-09-06
申请号:US10598686
申请日:2005-03-17
申请人: Michael Bell , Guoqing Cao , Ana Escribano , Maria Fernandez , Nathan Mantlo , Eva Martin de la Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiadong Wang
发明人: Michael Bell , Guoqing Cao , Ana Escribano , Maria Fernandez , Nathan Mantlo , Eva Martin de la Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiadong Wang
IPC分类号: A61K31/55 , C07D498/02 , C07D487/02
CPC分类号: C07D495/04 , C07D471/04 , C07D487/04
摘要: The present invention discloses compounds of formula I wherein A, n, m, j, q, y, W, X, Y, Z, R1, R2, R3, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed as useful for treating dyslipidemia and its sequelae.
摘要翻译: 本发明公开了式I的化合物,其中A,n,m,j,q,y,w,X,Y,Z,R 1,R 2,R R 4,R 5,R 5和R 6如本文所定义,并且它们的药物组合物和方法 公开了用于治疗血脂异常及其后遗症的用途。
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