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公开(公告)号:US20110060122A1
公开(公告)日:2011-03-10
申请号:US12759076
申请日:2010-04-13
IPC分类号: C07K1/113
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
摘要翻译: 公开了制备具有含氨基侧链的糖肽膦酸酯衍生物的方法。 几个工艺步骤在单个反应容器中进行,而不分离中间反应产物,从而产生较少的废物并提高该方法的总体效率和产率。
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公开(公告)号:US08093354B2
公开(公告)日:2012-01-10
申请号:US12759076
申请日:2010-04-13
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
摘要翻译: 公开了制备具有含氨基侧链的糖肽膦酸酯衍生物的方法。 几个工艺步骤在单个反应容器中进行,而不分离中间反应产物,从而产生较少的废物并提高该方法的总体效率和产率。
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公开(公告)号:US06979723B2
公开(公告)日:2005-12-27
申请号:US10226428
申请日:2002-08-23
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
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公开(公告)号:US07728104B2
公开(公告)日:2010-06-01
申请号:US11977436
申请日:2007-10-24
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
摘要翻译: 公开了制备具有含氨基侧链的糖肽膦酸酯衍生物的方法。 几个工艺步骤在单个反应容器中进行,而不分离中间反应产物,从而产生较少的废物并提高该方法的总体效率和产率。
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公开(公告)号:US20080227963A1
公开(公告)日:2008-09-18
申请号:US11977436
申请日:2007-10-24
IPC分类号: C07G11/00
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
摘要翻译: 公开了制备具有含氨基侧链的糖肽膦酸酯衍生物的方法。 几个工艺步骤在单个反应容器中进行,而不分离中间反应产物,从而产生较少的废物并提高该方法的总体效率和产率。
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公开(公告)号:US07301004B2
公开(公告)日:2007-11-27
申请号:US11437066
申请日:2006-05-19
IPC分类号: A61K38/14 , C07K9/0014
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
摘要翻译: 公开了制备具有含氨基侧链的糖肽膦酸酯衍生物的方法。 几个工艺步骤在单个反应容器中进行,而不分离中间反应产物,从而产生较少的废物并提高该方法的总体效率和产率。
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公开(公告)号:US07074890B2
公开(公告)日:2006-07-11
申请号:US10926148
申请日:2004-08-25
IPC分类号: A61K38/00
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
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公开(公告)号:US07160984B2
公开(公告)日:2007-01-09
申请号:US11268913
申请日:2005-11-08
申请人: Junning Lee , Jyanwei Liu
发明人: Junning Lee , Jyanwei Liu
CPC分类号: C07K9/008
摘要: Disclosed are processes for preparing glycopeptide antibiotic derivatives having an amino-containing side chain. The multi-step process is conducted in a single reaction vessel without isolation of intermediate reaction products.
摘要翻译: 公开了制备具有含氨基侧链的糖肽抗生素衍生物的方法。 多步法在不分离中间反应产物的单一反应容器中进行。
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公开(公告)号:US07015305B2
公开(公告)日:2006-03-21
申请号:US10226988
申请日:2002-08-23
申请人: Junning Lee , Jyanwei Liu
发明人: Junning Lee , Jyanwei Liu
IPC分类号: A61K38/00
CPC分类号: C07K9/008
摘要: Disclosed are processes for preparing glycopeptide antibiotic derivatives having an amino-containing side chain. The multi-step process is conducted in a single reaction vessel without isolation of intermediate reaction products.
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公开(公告)号:US20050020488A1
公开(公告)日:2005-01-27
申请号:US10926148
申请日:2004-08-25
申请人: Michael Leadbetter , Martin Linsell , Junning Lee , Jyanwei Liu
发明人: Michael Leadbetter , Martin Linsell , Junning Lee , Jyanwei Liu
摘要: Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.
摘要翻译: 公开了制备具有含氨基侧链的糖肽膦酸酯衍生物的方法。 几个工艺步骤在单个反应容器中进行,而不分离中间反应产物,从而产生较少的废物并提高该方法的总体效率和产率。
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