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1.Androgen receptor modulators and method of treating disease using the same 有权
标题翻译: 雄激素受体调节剂及其治疗方法相同公开(公告)号:US07268232B2
公开(公告)日:2007-09-11
申请号:US11130669
申请日:2005-05-16
申请人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Winther Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Boas Thygesen
发明人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Winther Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Boas Thygesen
IPC分类号: C07D451/02 , C07D401/00 , C07D405/00 , C07D409/00 , C07D413/00
CPC分类号: C07D207/08 , C07C255/58 , C07D207/09 , C07D207/10 , C07D207/12 , C07D207/14 , C07D207/16 , C07D207/20 , C07D211/22 , C07D211/32 , C07D211/34 , C07D211/38 , C07D211/42 , C07D211/46 , C07D211/48 , C07D211/58 , C07D211/60 , C07D211/62 , C07D211/64 , C07D211/70 , C07D215/20 , C07D215/40 , C07D215/48 , C07D217/02 , C07D217/04 , C07D217/22 , C07D217/24 , C07D221/20 , C07D221/22 , C07D237/34 , C07D241/42 , C07D285/14 , C07D295/06 , C07D295/073 , C07D295/096 , C07D295/155 , C07D451/00 , C07D451/02 , C07D451/04 , C07D451/06 , C07D471/04 , C07D471/08 , C07D471/10 , C07D487/08 , C07D491/10 , C07F9/572 , C07F9/6561
摘要: Disclosed herein are bicycloaryl compounds of Formula (I) that selectively modulate nuclear receptors, preferably the androgen receptor, or a pharmaceutically acceptable salt, ester, amide, or prodrug thereof, and methods of treating disease comprising administering a compound of Formula (I) to a patient in need thereof.
摘要翻译: 本文公开了式(I)的双环芳基化合物,其选择性调节核受体,优选雄激素受体或其药学上可接受的盐,酯,酰胺或前药,以及治疗疾病的方法,包括给予式(I)化合物至 有需要的患者。
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2.
公开(公告)号:US20090270449A1
公开(公告)日:2009-10-29
申请号:US12495514
申请日:2009-06-30
申请人: NATHALIE SCHLIENGER , Mikkel Boas Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Winther Lund , Roger Olsson
发明人: NATHALIE SCHLIENGER , Mikkel Boas Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Winther Lund , Roger Olsson
IPC分类号: A61K31/46 , C07D451/02
CPC分类号: C07D451/02 , C07D451/06
摘要: Disclosed herein is a novel class of aminophenyl compounds having the structure: wherein R1 is cyano or nitro and ring A is a bi- or tricyclic bridged heterocycle and to their use as modulators of androgen receptor for the treatment or prevention of conditions relating thereto.
摘要翻译: 本文公开了一类新的具有以下结构的氨基苯基化合物:其中R1是氰基或硝基,环A是双环或三环桥连杂环,并且其作为雄激素受体的调节剂用于治疗或预防与之有关的病症。
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3.
公开(公告)号:US07585877B2
公开(公告)日:2009-09-08
申请号:US11329267
申请日:2006-01-09
申请人: Nathalie Schlienger , Mikkel Boas Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Winther Lund , Roger Olsson
发明人: Nathalie Schlienger , Mikkel Boas Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Winther Lund , Roger Olsson
IPC分类号: A01N43/42 , A61K31/44 , C07D451/02
CPC分类号: C07D451/02 , C07D451/06
摘要: Disclosed herein is a novel class of aminophenyl compounds having the structure: wherein R1 is cyano or nitro and ring A is a bi- or tricyclic bridged heterocycle and to their use as modulators of androgen receptor for the treatment or prevention of conditions relating thereto.
摘要翻译: 本文公开了一类新的具有以下结构的氨基苯基化合物:其中R1是氰基或硝基,环A是双环或三环桥连杂环,并且其作为雄激素受体的调节剂用于治疗或预防与之有关的病症。
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4.ANDROGEN RECEPTOR MODULATORS AND METHOD OF TREATING DISEASE USING THE SAME 审中-公开
标题翻译: 雄激素受体调节剂及其治疗疾病的方法公开(公告)号:US20080009489A1
公开(公告)日:2008-01-10
申请号:US11770586
申请日:2007-06-28
申请人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Thygesen
发明人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Thygesen
IPC分类号: A61K31/439 , A61K31/40 , A61K31/445 , A61K31/5375 , A61P15/00 , A61P21/00 , A61P35/00 , A61P5/00 , C12N5/00
CPC分类号: C07D207/08 , C07C255/58 , C07D207/09 , C07D207/10 , C07D207/12 , C07D207/14 , C07D207/16 , C07D207/20 , C07D211/22 , C07D211/32 , C07D211/34 , C07D211/38 , C07D211/42 , C07D211/46 , C07D211/48 , C07D211/58 , C07D211/60 , C07D211/62 , C07D211/64 , C07D211/70 , C07D215/20 , C07D215/40 , C07D215/48 , C07D217/02 , C07D217/04 , C07D217/22 , C07D217/24 , C07D221/20 , C07D221/22 , C07D237/34 , C07D241/42 , C07D285/14 , C07D295/06 , C07D295/073 , C07D295/096 , C07D295/155 , C07D451/00 , C07D451/02 , C07D451/04 , C07D451/06 , C07D471/04 , C07D471/08 , C07D471/10 , C07D487/08 , C07D491/10 , C07F9/572 , C07F9/6561
摘要: Disclosed herein are bicycloaryl compounds of Formula (I) that selectively modulate nuclear receptors, preferably the androgen receptor, or a pharmaceutically acceptable salt, ester, amide, or prodrug thereof, and methods of treating disease comprising administering a compound of Formula (I) to a patient in need thereof.
摘要翻译: 本文公开了式(I)的双环芳基化合物,其选择性调节核受体,优选雄激素受体或其药学上可接受的盐,酯,酰胺或前药,以及治疗疾病的方法,包括给予式(I)化合物至 有需要的患者。
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5.Androgen receptor modulators and methods of treating disease using the same 审中-公开
标题翻译: 雄激素受体调节剂和使用其治疗疾病的方法公开(公告)号:US20070004679A1
公开(公告)日:2007-01-04
申请号:US11348949
申请日:2006-02-06
申请人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Thygesen , Douglas Bonhaus
发明人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Thygesen , Douglas Bonhaus
IPC分类号: A61K31/675 , A61K31/54 , A61K31/5375 , A61K31/445 , A61K31/40 , A61K31/495
CPC分类号: A61K31/40 , A61K31/439 , A61K31/445 , A61K31/504 , A61K31/5375 , C07D207/08 , C07D207/09 , C07D207/12 , C07D207/14 , C07D207/16 , C07D211/32 , C07D211/34 , C07D211/38 , C07D211/46 , C07D211/48 , C07D211/58 , C07D211/60 , C07D211/62 , C07D215/20 , C07D215/40 , C07D215/48 , C07D217/02 , C07D217/22 , C07D221/20 , C07D221/22 , C07D237/34 , C07D241/42 , C07D285/14 , C07D295/06 , C07D295/155 , C07D451/02 , C07D451/04 , C07D451/06 , C07D471/08 , C07D471/10 , C07D487/08 , C07D491/10
摘要: Disclosed herein are bicycloaryl compounds of Formula (I) that selectively modulate nuclear receptors, preferably the androgen receptor, or a pharmaceutically acceptable salt, ester, amide, or prodrug thereof, and methods of treating disease comprising administering a compound of Formula (I) to a patient in need thereof.
摘要翻译: 本文公开了式(I)的双环芳基化合物,其选择性调节核受体,优选雄激素受体或其药学上可接受的盐,酯,酰胺或前药,以及治疗疾病的方法,包括给予式(I)化合物至 有需要的患者。
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6.Androgen receptor modulators and method of treating disease using the same 有权
标题翻译: 雄激素受体调节剂及其治疗方法相同公开(公告)号:US20060014739A1
公开(公告)日:2006-01-19
申请号:US11130669
申请日:2005-05-16
申请人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Thygesen
发明人: Nathalie Schlienger , Jan Pawlas , Alma Fejzic , Roger Olsson , Birgitte Lund , Fabrizio Badalassi , Rasmus Lewinsky , Mikkel Thygesen
IPC分类号: A61K31/537 , C07D211/06 , C07D265/30 , A61K31/445
CPC分类号: C07D207/08 , C07C255/58 , C07D207/09 , C07D207/10 , C07D207/12 , C07D207/14 , C07D207/16 , C07D207/20 , C07D211/22 , C07D211/32 , C07D211/34 , C07D211/38 , C07D211/42 , C07D211/46 , C07D211/48 , C07D211/58 , C07D211/60 , C07D211/62 , C07D211/64 , C07D211/70 , C07D215/20 , C07D215/40 , C07D215/48 , C07D217/02 , C07D217/04 , C07D217/22 , C07D217/24 , C07D221/20 , C07D221/22 , C07D237/34 , C07D241/42 , C07D285/14 , C07D295/06 , C07D295/073 , C07D295/096 , C07D295/155 , C07D451/00 , C07D451/02 , C07D451/04 , C07D451/06 , C07D471/04 , C07D471/08 , C07D471/10 , C07D487/08 , C07D491/10 , C07F9/572 , C07F9/6561
摘要: Disclosed herein are bicycloaryl compounds of Formula (I) that selectively modulate nuclear receptors, preferably the androgen receptor, or a pharmaceutically acceptable salt, ester, amide, or prodrug thereof, and methods of treating disease comprising administering a compound of Formula (I) to a patient in need thereof.
摘要翻译: 本文公开了式(I)的双环芳基化合物,其选择性调节核受体,优选雄激素受体或其药学上可接受的盐,酯,酰胺或前药,以及治疗疾病的方法,包括给予式(I)化合物至 有需要的患者。
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公开(公告)号:US20060160845A1
公开(公告)日:2006-07-20
申请号:US11329267
申请日:2006-01-09
申请人: Nathalie Schlienger , Mikkel Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Lund , Roger Olsson
发明人: Nathalie Schlienger , Mikkel Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Lund , Roger Olsson
IPC分类号: C07D451/02 , A61K31/46
CPC分类号: C07D451/02 , C07D451/06
摘要: Disclosed herein is a novel class of aminophenyl compounds having the structure: wherein R1 is cyano or nitro and ring A is a bi- or tricyclic bridged heterocycle and to their use as modulators of androgen receptor for the treatment or prevention of conditions relating thereto.
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8.
公开(公告)号:US20060173037A1
公开(公告)日:2006-08-03
申请号:US11348929
申请日:2006-02-06
申请人: Nathalie Schlienger , Mikkel Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Lund , Roger Olsson
发明人: Nathalie Schlienger , Mikkel Thygesen , Jan Pawlas , Fabrizio Badalassi , Rasmus Lewinsky , Birgitte Lund , Roger Olsson
IPC分类号: C07D451/02 , A61K31/46
CPC分类号: C07D451/06 , C07D451/02
摘要: Disclosed herein is a novel class of aminophenyl compounds having the structure: wherein R1 is cyano or nitro and ring A is a bi- or tricyclic bridged heterocycle and to their use as modulators of androgen receptor for the treatment or prevention of conditions relating thereto.
摘要翻译: 本文公开了一类新型的具有以下结构的氨基苯基化合物:其中R 1是氰基或硝基,环A是双环或三环桥连杂环,并且它们用作治疗雄激素受体的调节剂 或预防与此相关的条件。
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公开(公告)号:US08822548B2
公开(公告)日:2014-09-02
申请号:US12915354
申请日:2010-10-29
申请人: Roger Olsson , Lene Hyldtoft , Fabrice Piu , Magnus Gustafsson , Vladimir Sherbukhin , Birgitte Winther Lund
发明人: Roger Olsson , Lene Hyldtoft , Fabrice Piu , Magnus Gustafsson , Vladimir Sherbukhin , Birgitte Winther Lund
IPC分类号: A61K31/055 , A61K31/05 , C07C37/055 , C07C37/62 , C07D263/32 , C07C39/42
CPC分类号: C07C37/055 , C07C17/263 , C07C17/2632 , C07C37/14 , C07C37/62 , C07C39/17 , C07C39/42 , C07C43/21 , C07C43/225 , C07C43/23 , C07C43/30 , C07C43/303 , C07C45/71 , C07C49/517 , C07C49/753 , C07C49/84 , C07C59/72 , C07C65/17 , C07C65/26 , C07C69/017 , C07C69/24 , C07C69/76 , C07C307/02 , C07C2601/14 , C07C2601/18 , C07C2602/20 , C07C2602/24 , C07D213/30 , C07D263/32 , C07D265/06 , C07D265/10 , C07D295/096 , C07D309/06 , C07D313/04 , C07D319/06 , C07D333/06 , C07D333/16 , C07F9/12 , C07C25/24 , C07C22/08 , C07C25/18
摘要: Disclosed herein are methods of treatment and prevention of diseases and disorders related to estrogen receptors comprising administering novel di-aromatic compounds to patients in need thereof.
摘要翻译: 本文公开了治疗和预防与雌激素受体相关的疾病和病症的方法,包括向有需要的患者施用新的二芳族化合物。
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公开(公告)号:US07825265B2
公开(公告)日:2010-11-02
申请号:US11269913
申请日:2005-11-08
申请人: Roger Olsson , Lene Hyldtoft , Fabrice Piu , Magnus Gustafsson , Vladimir Sherbukhin , Birgitte Winther Lund
发明人: Roger Olsson , Lene Hyldtoft , Fabrice Piu , Magnus Gustafsson , Vladimir Sherbukhin , Birgitte Winther Lund
IPC分类号: C07D309/00 , C07D321/00 , C07D405/00
CPC分类号: C07C37/055 , C07C17/263 , C07C17/2632 , C07C37/14 , C07C37/62 , C07C39/17 , C07C39/42 , C07C43/21 , C07C43/225 , C07C43/23 , C07C43/30 , C07C43/303 , C07C45/71 , C07C49/517 , C07C49/753 , C07C49/84 , C07C59/72 , C07C65/17 , C07C65/26 , C07C69/017 , C07C69/24 , C07C69/76 , C07C307/02 , C07C2601/14 , C07C2601/18 , C07C2602/20 , C07C2602/24 , C07D213/30 , C07D263/32 , C07D265/06 , C07D265/10 , C07D295/096 , C07D309/06 , C07D313/04 , C07D319/06 , C07D333/06 , C07D333/16 , C07F9/12 , C07C25/24 , C07C22/08 , C07C25/18
摘要: Disclosed herein are novel di-aromatic compounds and methods for using various di-aromatic compounds for treatment and prevention of diseases and disorders related to estrogen receptors.
摘要翻译: 本文公开了新型二芳族化合物和使用各种二芳族化合物治疗和预防与雌激素受体相关的疾病和病症的方法。
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