Lipid-A analogs: monosaccharide and dissaccharide compounds for
inhibiting binding of lipid A receptors to lipid A receptors
    3.
    发明授权
    Lipid-A analogs: monosaccharide and dissaccharide compounds for inhibiting binding of lipid A receptors to lipid A receptors 失效
    脂质-A类似物:用于抑制脂质A受体与脂质A受体结合的单糖和非糖化合物

    公开(公告)号:US5593969A

    公开(公告)日:1997-01-14

    申请号:US123590

    申请日:1993-09-17

    摘要: A compound of the formula: ##STR1## wherein: each of R.sub.1, R.sub.1 ', R.sub.2 and R.sub.2 ' independent of each other is a substituted or unsubstituted, branched or linear C.sub.1-12 alkyl, alkene or alkyne group, R.sub.3 is OH, OCH.sub.3, CH.sub.2 COOH or ##STR2## wherein each of R.sub.2" and R.sub.2 '41 independent of each other is a substituted or unsubstituted, branched or linear C.sub.1-12 alkyl, alkene or alkyne group and:A=NH.sub.2, X=P(OH), Y=Z=C, B=OCH.sub.3, orA=OH, X=P(OH), X=Z=C, B (if present)=OCH.sub.3, orA=OCO(CH.sub.2).sub.n NH.sub.2, X=P(OH), Y=Z=C, B=OCH.sub.3,wherein n=1-10, orA=OH, X=P(OH), Y=Z=C, B=O(CH.sub.2).sub.n CO.sub.2 H, wherein n=1-10, orA=OH, X=P(OH), Y=Z=C, B=(CH.sub.2).sub.n CO.sub.2 H, wherein n=1-10, orA=NH.sub.2, X=Z=C, Y=P(OH), B=OCH.sub.3, orA=OH, X=Z=C, Y=P(OH), B (if present)=OCH.sub.3, orA=OCO(CH.sub.2).sub.n NH.sub.2, X=Z=C, Y=P(OH), B=OCH.sub.3, wherein n=1-10, orA=OH, X=Z=C, Y=P(OH), B=O(CH.sub.2).sub.n CO.sub.2 H, wherein n=1-10, orA=OH, X=Z=C, Y=P(OH), B=(CH.sub.2).sub.n CO.sub.2 H, wherein n=1-11, orA=NH.sub.2, X=Y=C, Z=P(OH), B=OCH.sub.3, orA=OH, X=Y=C, Z=P(OH), B (if present)=OCH.sub.3, orA=OCO(CH.sub.2).sub.n NH.sub.2, X=Y=C, Z=P(OH), B=OCH.sub.3, wherein n=1-10, orA=OH, X=Y=C, Z=P(OH), B=O(CH.sub.2).sub.n CO.sub.2 H, wherein n=1-10, orA=OH, X=Y=C, Z=P (OH), B=(CH.sub.2).sub.n CO.sub.2 H and n=1-11 is disclosed. The compounds may be use to inhibit binding of Lipid A to Lipid A receptors.

    摘要翻译: 下式的化合物:其中:R 1,R 1',R 2和R 2'彼此独立地为取代或未取代的支链或直链C 1-12烷基,烯烃或炔基,R 3为 OH,OCH 3,CH 2 COOH或者其中每个R 2“和R 21'彼此独立地是取代或未取代的支链或直链C 1-12烷基,烯烃或炔基,并且:A = NH 2,X = P (OH),Y = Z = C,B = OCH 3或A = OH,X = P(OH),X = Z = C,B(如果存在)= OCH 3或A = OCO(CH 2)n NH 2,X = P(OH),Y = Z = C,B = OCH 3,其中n = 1-10,或A = OH,X = P(OH),Y = Z = C,B = O(CH 2)n CO 2 H,其中 n = 1-10,或A = OH,X = P(OH),Y = Z = C,B =(CH2)nCO2H,其中n = 1-10,或A = NH2,X = Z = C,Y = P(OH),B = OCH3或A = OH,X = Z = C,Y = P(OH),B(如果存在)= OCH 3或A = OCO(CH 2)n NH 2,X = Z = C ,Y = P(OH),B = OCH 3,其中n = 1-10,或A = OH,X = Z = C,Y = P(OH),B = O(CH 2)n CO 2 H,其中n = 10或A = OH,X = Z = C,Y = P(OH),B =(CH2)nCO2H,其中n = 1-11或A = NH2,X = Y = C,Z = P ),B = OCH 3或A = OH,X = Y = C,Z = P(OH),B(如果存在)= OCH 3或A = OCO(CH 2)n NH 2,X = Y = C,Z = P (OH),B = OCH 3, 其中n = 1-10,或A = OH,X = Y = C,Z = P(OH),B = O(CH 2)n CO 2 H,其中n = 1-10,或A = OH,X = Y = C ,Z = P(OH),B =(CH2)nCO2H和n = 1-11。 该化合物可用于抑制脂质A与脂质A受体的结合。

    Cyclic sulfonamide herbicides
    8.
    发明授权
    Cyclic sulfonamide herbicides 失效
    环磺酰胺除草剂

    公开(公告)号:US5874382A

    公开(公告)日:1999-02-23

    申请号:US12862

    申请日:1998-01-23

    摘要: Compounds of Formula I and II, and their agriculturally-suitable salts, are disclosed which are useful for controlling undesired vegetation ##STR1## wherein X is a direct bond; O; S; NH; N(C.sub.1 -C.sub.3 alkyl); N(C.sub.1 -C.sub.3 haloalkyl); or N(allyl);R.sup.1 is H; F; Cl; or Br;R.sup.2 is H; F; Cl; Br; CF.sub.3 ; nitro; or cyano;R.sup.4 is H; C.sub.1 -C.sub.3 alkyl; or halogen;R.sup.5 is H; C.sub.1 -C.sub.6 alkyl; C.sub.1 -C.sub.6 haloalkyl; halogen; S(O).sub.2 (C.sub.1 -C.sub.6 alkyl); or C(.dbd.O)R.sup.8 ; orR.sup.4 and R.sup.5 are taken together along with the carbon to which they are attached to form a spiro-cyclopropane ring;and R.sup.3, R.sup.8, and J are as defined in the disclosure.Also disclosed are compositions containing the compounds of Formulae I and II and a method for controlling undesired vegetation which involves contacting the vegetation or its environment with an effective amount of a compound of Formula I or II.

    摘要翻译: 公开了式I和II的化合物及其农业上合适的盐,其可用于控制不期望的植物; NH; N(C 1 -C 3烷基); N(C 1 -C 3卤代烷基); 或N(烯丙基); R1是H; F; Cl; 或Br; R2为H; F; Cl; Br; CF3; 硝基 或氰基; R4是H; C1-C3烷基; 或卤素; R5是H; C1-C6烷基; C1-C6卤代烷基; 卤素; S(O)2(C 1 -C 6烷基); 或C(= O)R 8; 或R 4和R 5与它们所连接的碳一起形成螺环丙烷环; 并且R3,R8和J如本公开所定义。 还公开了含有式I和II化合物的组合物和控制不期望植物的方法,其涉及将植物或其环境与有效量的式I或II化合物接触。

    Fungicidal hetercyclic compounds
    9.
    发明授权
    Fungicidal hetercyclic compounds 失效
    杀真菌异环化合物

    公开(公告)号:US08349870B2

    公开(公告)日:2013-01-08

    申请号:US12863875

    申请日:2009-01-22

    IPC分类号: A61K31/445 C07D405/00

    CPC分类号: C07D417/04 C07D417/14

    摘要: Disclosed are compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof, wherein E, R2, G, Z1, J and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.

    摘要翻译: 公开了式1的化合物,包括所有几何和立体异构体,N-氧化物及其盐,其中E,R 2,G,Z 1,J和n如本公开所定义。 还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法,包括施用有效量的本发明化合物或组合物。

    FUNGICIDAL HETEROCYCLIC COMPOUNDS
    10.
    发明申请
    FUNGICIDAL HETEROCYCLIC COMPOUNDS 失效
    真菌杂环化合物

    公开(公告)号:US20100292275A1

    公开(公告)日:2010-11-18

    申请号:US12863875

    申请日:2009-01-22

    IPC分类号: A01N43/80 C07D417/14 A01P3/00

    CPC分类号: C07D417/04 C07D417/14

    摘要: Disclosed are compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof, wherein E, R2, G, Z1, J and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.

    摘要翻译: 公开了式1的化合物,包括所有几何和立体异构体,N-氧化物及其盐,其中E,R 2,G,Z 1,J和n如本公开所定义。 还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法,包括施用有效量的本发明化合物或组合物。