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公开(公告)号:US06274737B1
公开(公告)日:2001-08-14
申请号:US09574413
申请日:2000-05-19
申请人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
发明人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
IPC分类号: C07D40510
CPC分类号: C07D307/79 , C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/65517
摘要: Novel indane and indene derivatives are described which are endothelin receptor antagonists.
摘要翻译: 描述了作为内皮素受体拮抗剂的新型茚满和茚衍生物
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公开(公告)号:US06448260B2
公开(公告)日:2002-09-10
申请号:US09901951
申请日:2001-07-10
申请人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
发明人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
IPC分类号: A61K3144
CPC分类号: C07D307/79 , C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/65517
摘要: Novel indane and indene derivatives are described which are endothelin receptor antagonists.
摘要翻译: 描述了作为内皮素受体拮抗剂的新型茚满和茚衍生物。
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公开(公告)号:US5719182A
公开(公告)日:1998-02-17
申请号:US442443
申请日:1995-05-16
申请人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
发明人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
IPC分类号: C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D307/79 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/655 , A61K31/36 , A61K31/19 , A61K31/335 , A61K31/44 , C07D317/64 , C07D317/70
CPC分类号: C07D307/79 , C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/65517
摘要: Novel indane and indene derivatives are described which are endothelin receptor antagonists.
摘要翻译: 描述了作为内皮素受体拮抗剂的新型茚满和茚衍生物。
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公开(公告)号:US06271399B1
公开(公告)日:2001-08-07
申请号:US08459985
申请日:1995-06-02
申请人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
发明人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
IPC分类号: C07D31754
CPC分类号: C07D307/79 , C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/65517
摘要: Indane and indene compounds are described which are endothelin receptor antagonists.
摘要翻译: 描述了吲哚和茚化合物,其是内皮素受体拮抗剂
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公开(公告)号:US5817693A
公开(公告)日:1998-10-06
申请号:US336444
申请日:1994-11-09
申请人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
发明人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
IPC分类号: C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D307/79 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/655 , A61K31/36 , C07D317/54
CPC分类号: C07D307/79 , C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/65517
摘要: Novel indane and indene derivatives are described which are endothelin receptor antagonists.
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公开(公告)号:US6087389A
公开(公告)日:2000-07-11
申请号:US99373
申请日:1998-06-18
申请人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
发明人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
IPC分类号: C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D307/79 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/655 , A61K31/335 , C07C255/03 , C07C317/04 , C07D319/14
CPC分类号: C07D307/79 , C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/65517
摘要: Novel indane and indene derivatives are described which are endothelin receptor antagonists.
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公开(公告)号:US5719183A
公开(公告)日:1998-02-17
申请号:US459686
申请日:1995-06-02
申请人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
发明人: Russell Donovan Cousins , John Duncan Elliott , Maria Amparo Lago , Jack Dale Leber , Catherine Elizabeth Peishoff
IPC分类号: C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D307/79 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/655 , A61K31/36 , A61K31/19 , A61K31/335 , A61K31/44
CPC分类号: C07D307/79 , C07C45/71 , C07C49/84 , C07C62/30 , C07C62/32 , C07C62/34 , C07C69/734 , C07C69/738 , C07C69/757 , C07D317/60 , C07D405/08 , C07D405/12 , C07F9/65517
摘要: Novel indane and indene derivatives are described which are endothelin receptor antagonists.
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