-
公开(公告)号:US07314879B2
公开(公告)日:2008-01-01
申请号:US10500476
申请日:2003-01-21
申请人: Ryan Thomas Backer , Caño Ivan Collado , Oscar De Frutos-Garcia , Christopher William Doecke , Matthew Joseph Fisher , Steven Lee Kuklish , Vincent Mancuso , Michael John Martinelli , Jeffrey Thomas Mullaney , Paul Leslie Ornstein , Chaoyu Xie
发明人: Ryan Thomas Backer , Caño Ivan Collado , Oscar De Frutos-Garcia , Christopher William Doecke , Matthew Joseph Fisher , Steven Lee Kuklish , Vincent Mancuso , Michael John Martinelli , Jeffrey Thomas Mullaney , Paul Leslie Ornstein , Chaoyu Xie
IPC分类号: A61K31/496 , C07D401/12 , C07D405/12 , C07D407/12
CPC分类号: C07D217/26 , C07D209/44 , C07D211/26 , C07D211/96 , C07D295/033 , C07D309/04 , C07D335/02 , C07D401/12 , C07D405/12 , C07D409/12
摘要: The present invention relates to melanocortin receptor agonist of the formula (I): which is useful in the treatment for obesity, diabetes, and male and/or female sexual dysfunction
摘要翻译: 本发明涉及式(I)的黑皮质素受体激动剂:其可用于治疗肥胖症,糖尿病和男性和/或女性性功能障碍
-
公开(公告)号:US07169777B2
公开(公告)日:2007-01-30
申请号:US10466250
申请日:2002-01-23
申请人: Ryan Thomas Backer , Karin Briner , Ivan Collado Caño , Oscar De Frutos Garcia , Christopher William Doecke , Matthew Joseph Fisher , Cristina Garcia-Paredes , Steven Lee Kuklish , Vincent Mancuso , Michael John Martinelli , Ana Isabel Mateo Herranz , Jeffrey Thomas Mullaney , Paul Leslie Ornstein , Zhipei Wu , Chaoyu Xie
发明人: Ryan Thomas Backer , Karin Briner , Ivan Collado Caño , Oscar De Frutos Garcia , Christopher William Doecke , Matthew Joseph Fisher , Cristina Garcia-Paredes , Steven Lee Kuklish , Vincent Mancuso , Michael John Martinelli , Ana Isabel Mateo Herranz , Jeffrey Thomas Mullaney , Paul Leslie Ornstein , Zhipei Wu , Chaoyu Xie
IPC分类号: A61K31/496 , A61K31/5377 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D413/14 , A61K31/551
CPC分类号: C07D209/48 , A61K38/00 , C07D209/44 , C07D217/12 , C07D217/16 , C07D217/26 , C07K5/06191
摘要: The present invention relates to melanocortin receptor agonist of the formula I useful in the treatment of obesity, diabetes, and male and/or female sexual dysfunction
摘要翻译: 本发明涉及式I的黑皮质素受体激动剂,其用于治疗肥胖症,糖尿病以及男性和/或女性性功能障碍
-
3.
公开(公告)号:US07157463B2
公开(公告)日:2007-01-02
申请号:US10466249
申请日:2002-01-23
申请人: Ryan Thomas Backer , Karin Briner , Christopher William Doecke , Matthew Joseph Fisher , Steven Lee Kuklish , Vincent Mancuso , Michael John Martinelli , Jeffrey Thomas Mullaney , Chaoyu Xie
发明人: Ryan Thomas Backer , Karin Briner , Christopher William Doecke , Matthew Joseph Fisher , Steven Lee Kuklish , Vincent Mancuso , Michael John Martinelli , Jeffrey Thomas Mullaney , Chaoyu Xie
IPC分类号: A61K31/496 , C07D401/12 , C07D403/12 , C07D403/14
CPC分类号: C07D401/12 , C07D209/44 , C07D217/26 , C07D401/14
摘要: The present invention relates to melanocortin receptor agonists of formula I, which is useful in the treatment of obesity, diabetes and male and/or female sexual dysfunction
摘要翻译: 本发明涉及式I的黑皮质素受体激动剂,其可用于治疗肥胖症,糖尿病和男性和/或女性性功能障碍
-
公开(公告)号:US07291619B2
公开(公告)日:2007-11-06
申请号:US10466121
申请日:2002-01-23
申请人: Christopher Kelly Biggers , Karin Briner , Christopher William Doecke , Matthew Joseph Fisher , Larry Wayne Hertel , Vincent Mancuso , Michael John Martinelli , John Philip Mayer , Paul Leslie Ornstein , Timothy Ivo Richardson , Jikesh Arvind Shah , Qing Shi , Zhipei Wu , Chaoyu Xie
发明人: Christopher Kelly Biggers , Karin Briner , Christopher William Doecke , Matthew Joseph Fisher , Larry Wayne Hertel , Vincent Mancuso , Michael John Martinelli , John Philip Mayer , Paul Leslie Ornstein , Timothy Ivo Richardson , Jikesh Arvind Shah , Qing Shi , Zhipei Wu , Chaoyu Xie
IPC分类号: A61K31/496 , C07D217/26 , C07D209/44
CPC分类号: A61K45/06 , C07D209/44 , C07D217/14 , C07D217/26 , C07D401/12 , C07D401/14 , C07D405/12 , C07D409/12 , C07D417/12
摘要: The present invention relates to melanocortin receptor agonists of formula (I), which is useful in the treatment of obesity, diabetes and male and/or female sexual dysfunction
摘要翻译: 本发明涉及式(I)的黑皮质素受体激动剂,其可用于治疗肥胖症,糖尿病和男性和/或女性性功能障碍
-
5.Piperazine- and piperidine-derivatives as melanocortin receptor agonists 失效
标题翻译: 哌嗪和哌啶衍生物作为黑皮质素受体激动剂公开(公告)号:US07186715B2
公开(公告)日:2007-03-06
申请号:US10466248
申请日:2002-01-23
申请人: Karin Briner , Christopher William Doecke , Vincent Mancuso , Michael John Martinelli , Timothy Ivo Richardson , Roger Ryan Rothhaar , Qing Shi , Chaoyu Xie
发明人: Karin Briner , Christopher William Doecke , Vincent Mancuso , Michael John Martinelli , Timothy Ivo Richardson , Roger Ryan Rothhaar , Qing Shi , Chaoyu Xie
IPC分类号: A61K31/496 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14
CPC分类号: A61K45/06 , C07D209/44 , C07D217/14 , C07D217/26 , C07D401/12 , C07D401/14 , C07D405/12 , C07D409/12 , C07D417/12
摘要: The present invention relates to melanocortin receptor agonists of formula I, which is useful in the treatment of obesity, diabetes and male and/or female sexual dysfunction
摘要翻译: 本发明涉及式I的黑皮质素受体激动剂,其可用于治疗肥胖症,糖尿病和男性和/或女性性功能障碍
-
公开(公告)号:US20050075344A1
公开(公告)日:2005-04-07
申请号:US10500476
申请日:2003-01-21
申请人: Ryan Backer , Ivan Collado Caño , Oscar De Furtos-Garcia , Christopher Doecke , Matthew Fisher , Steven Kuklish , Vincent Mancuso , Michael Martinelli , Jeffrey Mullaney , Paul Ornstein , Chaoyu Xie
发明人: Ryan Backer , Ivan Collado Caño , Oscar De Furtos-Garcia , Christopher Doecke , Matthew Fisher , Steven Kuklish , Vincent Mancuso , Michael Martinelli , Jeffrey Mullaney , Paul Ornstein , Chaoyu Xie
IPC分类号: A61K31/496 , A61K45/00 , A61P3/04 , A61P3/10 , A61P15/08 , A61P15/10 , A61P43/00 , C07B53/00 , C07B61/00 , C07C67/343 , C07C69/73 , C07C69/734 , C07D209/44 , C07D211/26 , C07D211/96 , C07D217/26 , C07D295/02 , C07D295/033 , C07D309/04 , C07D335/02 , C07D401/12 , C07D405/12 , C07D409/12 , A61K31/495 , C07D43/02 , C07D49/02
CPC分类号: C07D217/26 , C07D209/44 , C07D211/26 , C07D211/96 , C07D295/033 , C07D309/04 , C07D335/02 , C07D401/12 , C07D405/12 , C07D409/12
摘要: The present invention relates to melanocortin receptor agonist of the formula (I): which is useful in the treatment for obesity, diabetes, and male and/or female sexual dysfunction.
摘要翻译: 本发明涉及式(I)的黑皮质素受体激动剂:其可用于治疗肥胖症,糖尿病和男性和/或女性性功能障碍。
-
-
-
-
-