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公开(公告)号:US20090298829A1
公开(公告)日:2009-12-03
申请号:US12305935
申请日:2007-07-13
申请人: Sung Pil Choi , In Ae Ahn , Sang Hyup Lee , Sang Dae Lee , Mi Sook Shin , Koo Lee , Deog Young Choi , Dong Sup Shim , Hyeon Joo Yim , Min Kyung Yoon , Soo Yong Chung , Jung Ae Lee , Yong Hwa Ha , Young Kwan Kim , Oeuk Park , Hyun Min Lee , Youn Hoa Kim
发明人: Sung Pil Choi , In Ae Ahn , Sang Hyup Lee , Sang Dae Lee , Mi Sook Shin , Koo Lee , Deog Young Choi , Dong Sup Shim , Hyeon Joo Yim , Min Kyung Yoon , Soo Yong Chung , Jung Ae Lee , Yong Hwa Ha , Young Kwan Kim , Oeuk Park , Hyun Min Lee , Youn Hoa Kim
IPC分类号: A61K31/4025 , C07D401/06 , C07D413/14 , A61K31/5377 , A61P3/04 , A61P3/10 , A61P29/00 , A61P15/00
CPC分类号: C07D207/16 , C07D207/48 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要: The present invention relates to a compound of the following formula 1, pharmaceutically acceptable salt and isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.
摘要翻译: 本发明涉及有效作为黑皮质素受体激动剂的下式1化合物,其药学上可接受的盐和异构体,以及包含与活性成分相同的黑皮质素受体激动剂组合物。
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公开(公告)号:US07879852B2
公开(公告)日:2011-02-01
申请号:US12305935
申请日:2007-07-13
申请人: Sung Pil Choi , In Ae Ahn , Sang Hyup Lee , Sang Dae Lee , Mi Sook Shin , Koo Lee , Deog Young Choi , Dong Sup Shim , Hyeon Joo Yim , Min Kyung Yoon , Soo Yong Chung , Jung Ae Lee , Yong Hwa Ha , Young Kwan Kim , Oeuk Park , Hyun Min Lee , Youn Hoa Kim
发明人: Sung Pil Choi , In Ae Ahn , Sang Hyup Lee , Sang Dae Lee , Mi Sook Shin , Koo Lee , Deog Young Choi , Dong Sup Shim , Hyeon Joo Yim , Min Kyung Yoon , Soo Yong Chung , Jung Ae Lee , Yong Hwa Ha , Young Kwan Kim , Oeuk Park , Hyun Min Lee , Youn Hoa Kim
IPC分类号: A61K31/401 , A61K31/4025 , A61K31/422 , A61K31/427 , A61K31/4439 , A61K31/5377 , C07D207/14 , C07D213/72 , C07D263/48 , C07D277/54 , C07D295/28
CPC分类号: C07D207/16 , C07D207/48 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要: The present invention relates to a compound of the following formula 1, pharmaceutically acceptable salt and isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.
摘要翻译: 本发明涉及有效作为黑皮质素受体激动剂的下式1化合物,其药学上可接受的盐和异构体,以及包含与活性成分相同的黑皮质素受体激动剂组合物。
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公开(公告)号:US20110224219A1
公开(公告)日:2011-09-15
申请号:US13128725
申请日:2009-11-10
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
IPC分类号: A61K31/501 , C07D403/14 , A61K31/497 , A61P15/10 , A61P3/04
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
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公开(公告)号:US08183243B2
公开(公告)日:2012-05-22
申请号:US13158920
申请日:2011-06-13
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
IPC分类号: C07D405/14
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
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公开(公告)号:US20110237795A1
公开(公告)日:2011-09-29
申请号:US13158734
申请日:2011-06-13
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
IPC分类号: C07D403/14
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
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公开(公告)号:US08288386B2
公开(公告)日:2012-10-16
申请号:US13128725
申请日:2009-11-10
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
IPC分类号: A61K31/496 , A61K31/501 , A61K31/506 , C07D401/14 , C07D403/06 , C07D403/14 , C07D405/14 , C07D417/14
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
摘要翻译: 本发明涉及对黑皮质素受体或其药学上可接受的盐或异构体具有良好的激动作用的化合物和包含其作为活性成分的黑皮质素受体激动剂组合物。
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公开(公告)号:US08236955B2
公开(公告)日:2012-08-07
申请号:US13158734
申请日:2011-06-13
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
IPC分类号: C07D403/06
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
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公开(公告)号:US20110245500A1
公开(公告)日:2011-10-06
申请号:US13158920
申请日:2011-06-13
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
IPC分类号: C07D405/14
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
摘要翻译: 本发明涉及对黑皮质素受体或其药学上可接受的盐或异构体具有良好的激动作用的化合物和包含其作为活性成分的黑皮质素受体激动剂组合物。
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公开(公告)号:US20100120783A1
公开(公告)日:2010-05-13
申请号:US12615407
申请日:2009-11-10
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , In Ae Ahn , Sung Pil Choi , Hyun Ho Lee , Dong Sup Shim , Soo Yong Chung , Hyun Min Lee
IPC分类号: A61K31/496 , C07D403/14 , C07D405/14 , C07D409/14 , C07D401/14 , A61K31/501 , A61P3/04 , A61P3/10 , A61P29/00 , A61P15/00
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
摘要翻译: 本发明涉及对黑皮质素受体或其药学上可接受的盐或异构体具有良好的激动作用的化合物和包含其作为活性成分的黑皮质素受体激动剂组合物。
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公开(公告)号:US08039622B2
公开(公告)日:2011-10-18
申请号:US12615407
申请日:2009-11-10
申请人: Koo Lee , Sang Dae Lee , Sang Pil Moon , Dong Sup Shim , Soo Yong Chung
发明人: Koo Lee , Sang Dae Lee , Sang Pil Moon , Dong Sup Shim , Soo Yong Chung
IPC分类号: C07D405/14 , C07D401/14 , C07D403/06 , C07D403/14 , C07D409/14
CPC分类号: C07D417/14 , A61K31/4025 , A61K31/496 , C07D207/16 , C07D401/14 , C07D403/06 , C07D405/14 , C07D409/14
摘要: The present invention relates to a compound having a good agonistic activity to melanocortin receptor, or pharmaceutically acceptable salt or isomer thereof, and an agonistic composition for melanocortin receptor comprising the same as an active ingredient.
摘要翻译: 本发明涉及对黑皮质素受体或其药学上可接受的盐或异构体具有良好的激动作用的化合物和包含其作为活性成分的黑皮质素受体激动剂组合物。
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