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公开(公告)号:US20150080400A1
公开(公告)日:2015-03-19
申请号:US14397319
申请日:2013-04-30
申请人: TAKEDA GMBH
发明人: Angelika Hoffmeyer , Rainer Boer , Manuela Hessmann , Andreas Pahl , Torsten Dunkern , Simone Hartung , Christof Zitt , Jurgen Volz , Christiane Praechter , Mahindra Makhija , Hiteshkumar Jain , Sandip Gavade , Arati Prabhu , Manojkumar Tiwari , Ashish Keche , Sarvesh Patel
IPC分类号: C07C233/81 , C07D295/155 , C07C271/42 , C07C237/52 , A61K31/27 , A61K31/495 , A61K31/4453 , A61K31/196 , A61K45/06 , C07C235/66 , A61K31/5375
CPC分类号: C07C233/81 , A61K31/196 , A61K31/27 , A61K31/4453 , A61K31/495 , A61K31/5375 , A61K45/06 , C07C233/75 , C07C235/66 , C07C237/40 , C07C237/42 , C07C237/52 , C07C271/42 , C07D295/155
摘要: The compounds of formula (1) in which R1, R4, A and X have the meanings as given in the description, are novel effective EP2 agonists.
摘要翻译: 其中R1,R4,A和X具有说明书中给出的含义的式(1)化合物是新型有效的EP2激动剂。
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公开(公告)号:US09309187B2
公开(公告)日:2016-04-12
申请号:US14397319
申请日:2013-04-30
申请人: TAKEDA GMBH
发明人: Angelika Hoffmeyer , Rainer Boer , Manuela Hessmann , Andreas Pahl , Torsten Dunkern , Simone Hartung , Christof Zitt , Jurgen Volz , Christiane Praechter , Mahindra Makhija , Hiteshkumar Jain , Sandip Gavade , Arati Prabhu , Manojkumar Tiwari , Ashish Keche , Sarvesh Patel
IPC分类号: C07D265/30 , C07C233/81 , C07C233/75 , C07C235/66 , C07C237/40 , C07C237/42 , C07D295/155 , A61K31/196 , A61K31/27 , A61K31/4453 , A61K31/495 , A61K31/5375 , A61K45/06 , C07C237/52 , C07C271/42
CPC分类号: C07C233/81 , A61K31/196 , A61K31/27 , A61K31/4453 , A61K31/495 , A61K31/5375 , A61K45/06 , C07C233/75 , C07C235/66 , C07C237/40 , C07C237/42 , C07C237/52 , C07C271/42 , C07D295/155
摘要: The compounds of formula (1) in which R1, R4, A and X have the meanings as given in the description, are novel effective EP2 agonists.
摘要翻译: 其中R1,R4,A和X具有说明书中给出的含义的式(1)化合物是新型有效的EP2激动剂。
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