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公开(公告)号:US09868705B2
公开(公告)日:2018-01-16
申请号:US15023159
申请日:2014-09-25
发明人: John Katzenellenbogen , Donald McDonnell , John D. Norris , Alexander Parent , Julie Pollock , Jillian Gunther , Kathryn E. Carlson , Teresa Martin
IPC分类号: C07D239/48 , F23K3/00 , F23K1/04 , F23G5/04 , F01K5/02 , C07D213/24 , C07D213/74 , C07D239/26 , C07D239/30 , C07D239/34 , C07D239/47 , C07D239/52 , C07D239/54 , C07D239/58 , C07D241/12 , C07D241/16 , C07D241/18 , C07D401/14 , C07D403/08 , C07D403/14 , C07D407/08 , C07D409/14
CPC分类号: C07D239/48 , A61K45/06 , C07D213/24 , C07D213/74 , C07D239/26 , C07D239/30 , C07D239/34 , C07D239/47 , C07D239/52 , C07D239/54 , C07D239/58 , C07D241/12 , C07D241/16 , C07D241/18 , C07D401/14 , C07D403/08 , C07D403/14 , C07D407/08 , C07D409/08 , C07D409/14 , F01K5/02 , F23G5/04 , F23K1/04 , F23K3/00 , F23K2201/20 , F23K2203/103
摘要: The present disclosure provides tetra-substituted cyclobutane inhibitors of Androgen Receptor Action, and methods of using such inhibitors, for the treatment of hormone-refractory cancers.