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公开(公告)号:US20100204207A1
公开(公告)日:2010-08-12
申请号:US12763344
申请日:2010-04-20
申请人: Xinchao Chen , Christopher Lawrence Cioffi , Sean Richard Dinn , Ana Maria Escribano , Maria Carmen Fernandez , Todd Fields , Robert Jason Herr , Nathan Bryan Mantlo , Eva Maria Martin De La Nava , Ana Isabel Mateo Herranz , Saravanan Parthasarathy , Xiaodong Wang
发明人: Xinchao Chen , Christopher Lawrence Cioffi , Sean Richard Dinn , Ana Maria Escribano , Maria Carmen Fernandez , Todd Fields , Robert Jason Herr , Nathan Bryan Mantlo , Eva Maria Martin De La Nava , Ana Isabel Mateo Herranz , Saravanan Parthasarathy , Xiaodong Wang
IPC分类号: A61K31/55 , C07D403/12 , C07D417/12 , C07D491/048 , C07D405/14 , C07D413/12 , C07D401/14 , A61P3/00 , A61P9/10
CPC分类号: C07D401/14 , C07D401/12 , C07D403/12 , C07D403/14 , C07D405/14 , C07D413/12 , C07D417/12 , C07D491/04
摘要: Compounds of Formula (I): wherein n, m, p, q, Y, R1, R2, R3a, R3b, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed.
摘要翻译: 式(I)化合物:其中n,m,p,q,Y,R 1,R 2,R 3a,R 3b,R 4,R 5和R 6如本文所定义,并公开了其药物组合物和使用方法。
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公开(公告)号:US07786108B2
公开(公告)日:2010-08-31
申请号:US11570542
申请日:2005-06-23
申请人: Xinchao Chen , Todd Fields , Nathan Bryan Mantlo , Xiaodong Wang
发明人: Xinchao Chen , Todd Fields , Nathan Bryan Mantlo , Xiaodong Wang
IPC分类号: A61P9/10 , A61P3/06 , A61K31/55 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/12 , C07D417/12 , C07D417/14 , C07D491/04
CPC分类号: C07D401/14 , C07D401/12 , C07D403/12 , C07D403/14 , C07D405/14 , C07D413/12 , C07D417/12 , C07D491/04
摘要: Compounds of formula I wherein n, m, p, q, Y, R1 R2, R3a, R3b, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed.
摘要翻译: 其中n,m,p,q,Y,R 1,R 2,R 3a,R 3b,R 4,R 5和R 6如本文所定义的式I化合物及其药物组合物和使用方法。
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公开(公告)号:US07749992B2
公开(公告)日:2010-07-06
申请号:US10574649
申请日:2004-10-07
申请人: Guoqing Cao , Ana Maria Escribano , Maria Carmen Fernandez , Todd Fields , Douglas Linn Gernert , Christopher Lawrence Cioffi , Robert Jason Herr , Nathan Bryan Mantlo , Eva Maria Martin De La Nava , Ana Isabel Mateo Herranz , Daniel Ray Mayhugh , Xiaodong Wang
发明人: Guoqing Cao , Ana Maria Escribano , Maria Carmen Fernandez , Todd Fields , Douglas Linn Gernert , Christopher Lawrence Cioffi , Robert Jason Herr , Nathan Bryan Mantlo , Eva Maria Martin De La Nava , Ana Isabel Mateo Herranz , Daniel Ray Mayhugh , Xiaodong Wang
IPC分类号: A61P3/06 , A61P9/10 , A61K31/55 , C07D223/14 , C07D223/16 , C07D223/32 , C07D225/06 , C07D403/04 , C07D403/12 , C07D405/06 , C07D405/12 , C07D413/04 , C07D491/04
CPC分类号: C07D223/16 , C07D223/14 , C07D223/32 , C07D225/06 , C07D403/04 , C07D403/12 , C07D405/06 , C07D405/12 , C07D413/04 , C07D491/04
摘要: Compounds of formula I wherein n, m, p, q, y, R1 R2, R3, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed as useful for treating artherosclerosis and its sequelae.
摘要翻译: 其中n,m,p,q,y,R 1,R 2,R 3,R 4,R 5和R 6如本文所定义的式I化合物,其药物组合物和使用方法被公开用于治疗动脉粥样硬化及其后遗症。
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公开(公告)号:US20070244095A1
公开(公告)日:2007-10-18
申请号:US11570542
申请日:2005-06-23
申请人: Xinchao Chen , Christopher Cioffi , Sean Dinn , Ana Escribano , Maria Fernandez , Todd Fields , Robert Herr , Nathan Mantlo , Eva Martin De La Nava , Ana Mateo-Herranz , Saravanan Parthasarathy , Xiaodong Wang
发明人: Xinchao Chen , Christopher Cioffi , Sean Dinn , Ana Escribano , Maria Fernandez , Todd Fields , Robert Herr , Nathan Mantlo , Eva Martin De La Nava , Ana Mateo-Herranz , Saravanan Parthasarathy , Xiaodong Wang
IPC分类号: A61K31/55 , C07D223/16
CPC分类号: C07D401/14 , C07D401/12 , C07D403/12 , C07D403/14 , C07D405/14 , C07D413/12 , C07D417/12 , C07D491/04
摘要: Compounds of formula I wherein n, m, p, q, Y, R1 R2, R3a, R3b, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed.
摘要翻译: 其中n,m,p,q,Y,R 1,R 2,R 3a,R 3b, R 4,R 5,R 5和R 6如本文所定义,并且公开了它们的药物组合物和使用方法。
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公开(公告)号:US20070254869A1
公开(公告)日:2007-11-01
申请号:US10574649
申请日:2004-10-07
申请人: Guoqing Cao , Ana Escribano , Maria Fernandez , Todd Fields , Douglas Gernert , Christopher Cioffi , Robert Herr , Nathan Mantlo , Eva Martin De La Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiaodong Wang
发明人: Guoqing Cao , Ana Escribano , Maria Fernandez , Todd Fields , Douglas Gernert , Christopher Cioffi , Robert Herr , Nathan Mantlo , Eva Martin De La Nava , Ana Mateo Herranz , Daniel Mayhugh , Xiaodong Wang
IPC分类号: A61K31/55 , A61P9/10 , C07D223/14 , C07D223/16
CPC分类号: C07D223/16 , C07D223/14 , C07D223/32 , C07D225/06 , C07D403/04 , C07D403/12 , C07D405/06 , C07D405/12 , C07D413/04 , C07D491/04
摘要: Compounds of formula I wherein n, m, p, q, y, R1 R2, R3, R4, R5, and R6 are as defined herein and their pharmaceutical compositions and methods of use are disclosed as useful for treating artherosclerosis and its sequelae.
摘要翻译: 其中n,m,p,q,y,R 1,R 2,R 3,R 4, R 5,R 5和R 6如本文所定义,并且它们的药物组合物和使用方法被公开用于治疗动脉粥样硬化及其后遗症。
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