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公开(公告)号:US20100256092A1
公开(公告)日:2010-10-07
申请号:US12464829
申请日:2009-05-12
申请人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Vincent S. Hernandez , Jacob J. Plattner , Charles Z. Ding , Kathy Cao , Yong-Kang Zhang , Andrew Benowitz , Tsutomu Akama , Jessica Sligar , Guofeng Jia , Ligong Ou , Neerja Saraswat , Sreekanth Ramachandran , Chris Diaper , Yanchen Zhang , Goverdhan Reddy Banda , James A. Nieman , Mehdi Keramane , Rahim Mohammed , Rajendra Subedi , Hong Liang , Rajeshwar Singh
发明人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Vincent S. Hernandez , Jacob J. Plattner , Charles Z. Ding , Kathy Cao , Yong-Kang Zhang , Andrew Benowitz , Tsutomu Akama , Jessica Sligar , Guofeng Jia , Ligong Ou , Neerja Saraswat , Sreekanth Ramachandran , Chris Diaper , Yanchen Zhang , Goverdhan Reddy Banda , James A. Nieman , Mehdi Keramane , Rahim Mohammed , Rajendra Subedi , Hong Liang , Rajeshwar Singh
CPC分类号: A61K31/33 , A61K31/43 , A61K45/06 , C07F5/025 , Y02A50/401 , Y02A50/411 , A61K2300/00
摘要: This invention relates to, among other items, 6-substituted benzoxaborole compounds and their use for treating bacterial infections.
摘要翻译: 本发明涉及6-取代的苯并恶唑化合物及其用于治疗细菌感染的用途。
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公开(公告)号:US20110136763A1
公开(公告)日:2011-06-09
申请号:US12844748
申请日:2010-07-27
申请人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
发明人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
CPC分类号: C07F5/025 , A61K31/69 , A61K45/06 , A61K2300/00
摘要: This invention largely relates to 3,4,6-trisubstituted benzoxaborole compounds, and their use for treating bacterial infections.
摘要翻译: 本发明主要涉及3,4,6-三取代苯并恶唑化合物及其用于治疗细菌感染的用途。
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公开(公告)号:US08343944B2
公开(公告)日:2013-01-01
申请号:US12844748
申请日:2010-07-27
申请人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
发明人: Yi Xia , Michael Richard Kevin Alley , Yasheen Zhou , Rajeshwar Singh , Charles Ding , Kathy Cao , Jacob J. Plattner , Ligong Ou , Guofeng Jia , Neerja Saraswat , Sreekanth Ramachandran , Ding Zhou
CPC分类号: C07F5/025 , A61K31/69 , A61K45/06 , A61K2300/00
摘要: This invention largely relates to 3,4,6-trisubstituted benzoxaborole compounds, and their use for treating bacterial infections.
摘要翻译: 本发明主要涉及3,4,6-三取代苯并恶唑化合物及其用于治疗细菌感染的用途。
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公开(公告)号:US20060287309A1
公开(公告)日:2006-12-21
申请号:US11466822
申请日:2006-08-24
申请人: Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
发明人: Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
IPC分类号: A61K31/5383 , A61K31/519 , A61K31/525 , A61K31/496 , A61K31/4745 , C07D491/02 , C07D487/02
CPC分类号: C07D471/04
摘要: This invention relates to compounds of the formula 1 wherein G, D, A, Z, Q, X, Y, R1, and R4 through R7 are defined as in the specification, processes for preparing the same and intermediates used in making the same, and pharmaceutical compositions containing such compounds and their use in the treatment of central nervous system disorders and other disorders.
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5.[1,8]NAPHTHYRIDIN-2-ONES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA 审中-公开
标题翻译: [1,8]萘啶-2-酮及相关化合物治疗苦参碱公开(公告)号:US20060287310A1
公开(公告)日:2006-12-21
申请号:US11466828
申请日:2006-08-24
申请人: Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
发明人: Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
IPC分类号: A61K31/5383 , A61K31/519 , A61K31/496 , A61K31/4745 , C07D471/02 , C07D491/02 , C07D487/02
CPC分类号: C07D471/04
摘要: This invention relates to compounds of the formula 1 wherein G, D, A, Z, Q, X, Y, R1, and R4 through R7 are defined as in the specification, processes for preparing the same and intermediates used in making the same, and pharmaceutical compositions containing such compounds and their use in the treatment of central nervous system disorders and other disorders.
摘要翻译: 本发明涉及式1的化合物,其中G,D,A,Z,Q,X,Y,R 1和R 4至R 7 在说明书中定义,其制备方法和用于制备其的中间体,以及含有这些化合物的药物组合物及其在治疗中枢神经系统疾病和其它疾病中的用途。
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6.[1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia 失效
标题翻译: [1,8]萘啶-2-酮和相关化合物用于治疗精神分裂症公开(公告)号:US20050043309A1
公开(公告)日:2005-02-24
申请号:US10900210
申请日:2004-07-28
申请人: Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
发明人: Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
IPC分类号: A61P25/18 , C07D471/04 , C07D498/04 , A61K31/525 , A61K31/519 , C07D487/02
CPC分类号: C07D471/04
摘要: This invention relates to compounds of the formula 1 wherein G, D, A, Z, Q, X, Y, R1, and R4 through R7 are defined as in the specification, processes for preparing the same and intermediates used in making the same, and pharmaceutical compositions containing such compounds and their use in the treatment of central nervous system disorders and other disorders.
摘要翻译: 本发明涉及式1的化合物,其中G,D,A,Z,Q,X,Y,R 1和R 4至R 7如本说明书中所定义, 用于制造相同物质的中间体以及含有这些化合物的药物组合物及其在治疗中枢神经系统疾病和其它疾病中的用途。
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