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公开(公告)号:US06777426B2
公开(公告)日:2004-08-17
申请号:US09933106
申请日:2001-08-20
IPC分类号: C07D23324
CPC分类号: C07D401/06 , C07D233/50 , C07D401/12 , C07D403/12 , C07D471/04 , C07D491/04 , C07D495/04
摘要: This invention is directed to novel imidazole and imidazoline derivatives which are selective agonists for cloned human &agr;2 adrenergic receptors. This invention is also related to the use of these compounds for the treatment of any disease where modulation of the &agr;2 receptors may be useful. The invention further provides for a pharmaceutical composition comprising a therapeutically effective amount of the above-defined compounds and a pharmaceutically acceptable carrier.
摘要翻译: 本发明涉及新的咪唑和咪唑啉衍生物,其是用于克隆的人α2肾上腺素能受体的选择性激动剂。 本发明还涉及这些化合物用于治疗其中α2受体调节可能有用的任何疾病的用途。 本发明还提供了包含治疗有效量的上述化合物和药学上可接受的载体的药物组合物。
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公开(公告)号:US06696572B2
公开(公告)日:2004-02-24
申请号:US10167628
申请日:2002-06-12
申请人: George Richard Meyer
发明人: George Richard Meyer
IPC分类号: C07D23324
CPC分类号: C23F11/149 , C09K8/54 , C23F11/161
摘要: The present invention relates to a process for making and a method for using a corrosion inhibitor composition to reduce the corrosion rate of a metal by a fluid containing a corrosion agent. The corrosion inhibitor composition comprises at least a quaternized compound. Examples of the quaternized compound are quaternized imino imidazolines and quaternized amido imidazolines.
摘要翻译: 本发明涉及一种制备方法和一种使用缓蚀剂组合物以通过含有腐蚀剂的流体降低金属的腐蚀速率的方法。 腐蚀抑制剂组合物至少包含季铵化合物。 季铵化合物的实例是季铵化亚氨基咪唑啉和季铵化酰胺咪唑啉。
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