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发明公开
CN102186839A 氮杂环丁烷多取代的化合物、其制备及其治疗用途 无效 - 撤回

氮杂环丁烷多取代的化合物、其制备及其治疗用途
摘要：
本发明涉及式(I)化合物，其中：R为(C1-C6)烷基、卤代(C1-C6)烷基；R1为氢原子；R2为杂芳族基团或杂芳族(C1-C4)烷基，所述基团任选被取代；R3和R4彼此独立地表示任选被取代的苯基；Y为氢原子、卤素、氰基、(C1-C6)烷基、卤代(C1-C6)烷基、(C1-C6)烷氧基、卤代(C1-C6)烷氧基或(C1-C6)烷基S(O)p基团；且p为0-2。所述化合物可为碱形式或与酸的加成盐的形式。本发明还涉及制备该化合物的方法及其治疗用途。
摘要（英）：

The invention relates to compounds of the formula (I) where: R is a (C1-C6)alkyl group, a halo(C1-C6)alkyl group; R1 is a hydrogen atom; R2 is a heteroaromatic group or a heteroaromatic(C1-C4)alkyl group, said groups being optionally substituted; R3 and R4 represent independently from each other an optionally substituted phenyl group; Y is a hydrogen atom, a halogen, a cyano, a (C1-C6)alkyl group, a halo(C1-C6)alkyl group, a (C1-C6)alkoxy group, a halo(C1-C6)alkoxy group or a (C1-C6)alkylS(0)p group; and p is 0 to 2. Said compounds can be in the form of a base or a salt for addition to an acid. The invention also relates to a method for preparing same and to the therapeutic application thereof.

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