发明公开
EP0592677A1 Beta-LACTAM COMPOUND AND CEPHEM COMPOUND, AND PRODUCTION THEREOF
失效
Beta-Laktam和Cepham Verbindungen und Ihre Herstellung。
- 专利标题： Beta-LACTAM COMPOUND AND CEPHEM COMPOUND, AND PRODUCTION THEREOF
- 专利标题（中）： Beta-Laktam和Cepham Verbindungen und Ihre Herstellung。
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申请号： EP93903302.3申请日： 1993-02-03
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公开(公告)号： EP0592677A1公开(公告)日： 1994-04-20
- 发明人: TORII, Shigeru 4-18, Sanyodanchi 4-chome , TANAKA, Hideo 5115-34, Haga , SASAOKA, Mitio 1-16, Nakanokoshi , SHIROI, Takashi 51-41, Aza Nishinosu Tainohama , KAMEYAMA, Yutaka 24-19-406, Okudahonmachi
- 申请人： OTSUKA KAGAKU KABUSHIKI KAISHA
- 申请人地址： 2-27, Ote-dori 3-chome Chuo-ku Osaka-shi Osaka-fu 540 JP
- 专利权人： OTSUKA KAGAKU KABUSHIKI KAISHA
- 当前专利权人： OTSUKA KAGAKU KABUSHIKI KAISHA
- 当前专利权人地址： 2-27, Ote-dori 3-chome Chuo-ku Osaka-shi Osaka-fu 540 JP
- 代理机构： Barz, Peter, Dr.
- 优先权： JP30310/92 19920218; JP30311/92 19920218
- 国际公布： WO9316043 19930819
- 主分类号： C07D205/08
- IPC分类号： C07D205/08 ; C07D501/00 ; C07D501/18 ; C07D501/22 ; C07D501/57 ; C07D501/60 ; C07D205/09 ; C07D205/095
摘要：
A β-lactam compound and a 2-(substituted methyl)-3-cephem compound, both being useful as an intermediate for the synthesis of cephem antibiotics and so forth. The lactam compound is represented by general formula (I), wherein R¹ represents protected amino, etc.; R² represents hydrogen, etc.; R³ represents hydrogen or a protective group for a carboxyl group; R⁴ represents optionally substituted aryl; and R⁵ represents optionally substituted alkenyl, etc. The cephem compound is represented by general formula (II), wherein R¹, R² and R³ are each as defined above; and R⁶ represents optionally substituted aryl.
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