发明公开
- 专利标题： PROSTAGLANDIN DERIVATIVES
- 专利标题（中）： 前列腺素衍生物
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申请号： EP00951967.9申请日： 2000-08-11
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公开(公告)号： EP1219600A1公开(公告)日： 2002-07-03
- 发明人: SATO, Fumie , TANAMI, Tohru, c/o Taisho Pharmaceutical Co Ltd , TANAKA, Hideo, c/o Taisho Pharmaceutical Co Ltd , ONO, Naoya, c/o Taisho Pharmaceutical Co Ltd , YAGI, Makoto, c/o Taisho Pharmaceutical Co Ltd
- 申请人： TAISHO PHARMACEUTICAL CO., LTD , Sato, Fumie
- 申请人地址： 24-1 Takata 3-chome, Toshima-ku Tokyo 170-8633 JP
- 专利权人： TAISHO PHARMACEUTICAL CO., LTD,Sato, Fumie
- 当前专利权人： TAISHO PHARMACEUTICAL CO., LTD,Sato, Fumie
- 当前专利权人地址： 24-1 Takata 3-chome, Toshima-ku Tokyo 170-8633 JP
- 代理机构： VOSSIUS & PARTNER
- 优先权： JP22916899 19990813
- 国际公布： WO0112596 20010222
- 主分类号： C07C405/00
- IPC分类号： C07C405/00 ; A61K31/5575 ; A61P13/12 ; A61P9/10 ; A61P9/04 ; A61P9/12 ; A61P25/20
摘要：
A prostaglandin derivative represented by the formula:
wherein X is a halogen atom, R 1 is a hydrogen atom, a C 1-10 alkyl group or a C 3-10 cycloalkyl group, m is an integer of 0 to 5, and Y is a group represented by the formula:
wherein R 2 is a C 3-10 cycloalkyl group, a C 3-10 cycloalkyl group substituted with C 1-4 alkyl group(s), a C 1-4 alkyl group substituted with C 3-10 cycloalkyl group(s), a C 1-10 alkyl group, a C 2-10 alkenyl group, a C 2-10 alkynyl group or a bridged cyclic hydrocarbon group, or a group represented by the formula:
wherein n is an integer of 1 to 8; a pharmaceutically acceptable salt thereof or a hydrate thereof.
wherein X is a halogen atom, R 1 is a hydrogen atom, a C 1-10 alkyl group or a C 3-10 cycloalkyl group, m is an integer of 0 to 5, and Y is a group represented by the formula:
wherein R 2 is a C 3-10 cycloalkyl group, a C 3-10 cycloalkyl group substituted with C 1-4 alkyl group(s), a C 1-4 alkyl group substituted with C 3-10 cycloalkyl group(s), a C 1-10 alkyl group, a C 2-10 alkenyl group, a C 2-10 alkynyl group or a bridged cyclic hydrocarbon group, or a group represented by the formula:
wherein n is an integer of 1 to 8; a pharmaceutically acceptable salt thereof or a hydrate thereof.
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