发明公开
- 专利标题： CONDENSED HETEROARYL DERIVATIVES
- 专利标题（中）： KONDENSIERTE HETEROARYLDERIVATE
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申请号： EP01925981.1申请日： 2001-04-26
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公开(公告)号： EP1277738A1公开(公告)日： 2003-01-22
- 发明人: HAYAKAWA, Masahiko , KAIZAWA, Hiroyuki , MORITOMO, Hiroyuki , KAWAGUCHI, Ken-ichi , KOIZUMI, Tomonobu , YAMANO, Mayumi , MATSUDA, Koyo , OKADA, Minoru , OHTA, Mitsuaki
- 申请人： YAMANOUCHI PHARMACEUTICAL CO. LTD. , LUDWIG INSTITUTE FOR CANCER RESEARCH , IMPERIAL CANCER RESEARCH TECHNOLOGY LIMITED
- 申请人地址： No. 3-11 Nihonbashi-Honcho, 2-chome Chuo-ku Tokyo 103-8411 JP
- 专利权人： YAMANOUCHI PHARMACEUTICAL CO. LTD.,LUDWIG INSTITUTE FOR CANCER RESEARCH,IMPERIAL CANCER RESEARCH TECHNOLOGY LIMITED
- 当前专利权人： YAMANOUCHI PHARMACEUTICAL CO. LTD.,LUDWIG INSTITUTE FOR CANCER RESEARCH,IMPERIAL CANCER RESEARCH TECHNOLOGY LIMITED
- 当前专利权人地址： No. 3-11 Nihonbashi-Honcho, 2-chome Chuo-ku Tokyo 103-8411 JP
- 代理机构： Bates, Philip Ian
- 优先权： JP2000128472 20000427
- 国际公布： WO01083456 20011108
- 主分类号： C07D215/42
- IPC分类号： C07D215/42 ; C07D239/94 ; C07D471/04 ; C07D491/147 ; C07D471/14 ; C07D495/14 ; C07D413/04 ; C07D401/04 ; C07D401/12 ; C07D409/04 ; C07D409/12 ; C07D405/04 ; C07D405/12 ; C07D403/04 ; C07D417/12 ; C07D487/04 ; C07D495/04 ; C07D491/048 ; A61K31/5377 ; A61K31/519 ; A61K31/517
摘要：
The present invention provides a pharmaceutical composition which is useful as a phosphatidylinositol 3 kinase (PI3K) inhibitor and an antitumor agent, and it provides a novel bicyclic or tricyclic fused heteroaryl derivative or a salt thereof which possesses an excellent PI3K inhibiting activity and cancer cell growth inhibiting activity.
公开/授权文献
- EP1277738B1 CONDENSED HETEROARYL DERIVATIVES 公开/授权日：2011-03-30
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