发明公开
EP1448534A1 6-MEMBERED UNSATURATED HETEROCYCLIC COMPOUNDS USEFUL FOR SELECTIVE INHIBITION OFTHE COAGULATION CASCADE
审中-公开
6-GLIEDRIGEUNGESÄTTIGTEHETEROCYCLEN VERWENDBARFÜRSELEKTIVE HEMMUNG DER COAGULATIONSKASKADE
- 专利标题： 6-MEMBERED UNSATURATED HETEROCYCLIC COMPOUNDS USEFUL FOR SELECTIVE INHIBITION OFTHE COAGULATION CASCADE
- 专利标题（中）： 6-GLIEDRIGEUNGESÄTTIGTEHETEROCYCLEN VERWENDBARFÜRSELEKTIVE HEMMUNG DER COAGULATIONSKASKADE
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申请号： EP02800488.5申请日： 2002-10-03
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公开(公告)号： EP1448534A1公开(公告)日： 2004-08-25
- 发明人: SOUTH, Michael, S. , WEBBER, Ronald, K. , HUANG, Horng-Chih , TOTH, Mihaly, V. , MOORMANN, Alan, E. , SNYDER, Jeffrey, S. , SCHOLTEN, Jeffrey, A. , GARLAND, Danny, J. , RUEPPEL, Melvin, L. , NEUMANN, William, L. , LONG, Scott , WEI, Huang , TRUJILLO, John , PARLOW, John, J. , JONES, Darin, E. , CASE, Brenda , HAYES, Michael, J. , ZENG, Qingping , ABBAS, Zaheer , FENTON, Ricky L. , KUSTURIN, Carrie L. , HAYAT, Rahman K. , SAMPLE, Kirby R. , SCHWEITZER, Barbara A. , WOOD, Rhonda S. , SZALONY, Jim , SULEYMANOV, Osman D. , SALYERS, Anita , NICHOLSON, Nancy S.
- 申请人： Pharmacia Corporation
- 申请人地址： Corporate Patent Department,P.O. Box 1027 St. Louis, MO 63006 US
- 专利权人： Pharmacia Corporation
- 当前专利权人： Pharmacia Corporation
- 当前专利权人地址： Corporate Patent Department,P.O. Box 1027 St. Louis, MO 63006 US
- 代理机构： Albrecht, Thomas, Dr.
- 优先权： US326721P 20011003; US338623P 20011024; US332857P 20011106; US333292P 20011114; US332107P 20011121; US332014P 20011121
- 国际公布： WO2003029224 20030410
- 主分类号： C07D239/47
- IPC分类号： C07D239/47 ; C07D241/20 ; C07D403/12 ; C07D409/12 ; C07D401/12 ; C07D403/10 ; C07D403/04 ; C07D471/04 ; A61K31/4965 ; A61K31/513 ; A61P7/02
摘要：
The present invention relates to compounds, and prodrugs thereof, composition and methods useful for preventing and treating thrombotic conditions in mammals. The compounds of the present invention, and prodrugs thereof, selectively inhibit certain proteases of the coagulation cascade.
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