发明公开
EP2058310A1 PYRAZOLOPYRIDINE CARBOXAMIDE DERIVATIVE AND PHOSPHODIESTERASE (PDE) INHIBITOR COMPRISING THE DERIVATIVE
审中-公开
磷酸二氢吡啶类衍生物（PDE）-HEMMER
- 专利标题： PYRAZOLOPYRIDINE CARBOXAMIDE DERIVATIVE AND PHOSPHODIESTERASE (PDE) INHIBITOR COMPRISING THE DERIVATIVE
- 专利标题（中）： 磷酸二氢吡啶类衍生物（PDE）-HEMMER
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申请号： EP07806367.4申请日： 2007-08-30
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公开(公告)号： EP2058310A1公开(公告)日： 2009-05-13
- 发明人: KOHNO, Yasushi , OCHIAI, Koji , KOJIMA, Akihiko
- 申请人： Kyorin Pharmaceutical Co., Ltd.
- 申请人地址： 5, Kandasurugadai 2-chome, Chiyoda-ku Tokyo 101-8311 JP
- 专利权人： Kyorin Pharmaceutical Co., Ltd.
- 当前专利权人： Kyorin Pharmaceutical Co., Ltd.
- 当前专利权人地址： 5, Kandasurugadai 2-chome, Chiyoda-ku Tokyo 101-8311 JP
- 代理机构： Vossius & Partner
- 优先权： JP2006237168 20060901
- 国际公布： WO2008026687 20080306
- 主分类号： C07D471/04
- IPC分类号： C07D471/04 ; A61K31/437 ; A61K31/444 ; A61P7/02 ; A61P9/04 ; A61P9/12 ; A61P11/00 ; A61P11/06 ; A61P15/10 ; A61P25/00 ; A61P25/14 ; A61P25/16 ; A61P25/28 ; A61P27/16 ; A61P29/00 ; A61P37/08 ; A61P43/00
摘要：
A novel pyrazolopyridine carboxamide derivative is provided that is useful as a pharmaceutical drug having phosphodiesterase inhibitory activity.
The pyrazolopyridine carboxamide derivative is represented by the following general formula (1):
(Example: 2-ethyl-7-methoxypyrazolo[1,5-a]pyridine-4-carboxylic acid (3,5-dichloropyridin-4-yl)amide).
The pyrazolopyridine carboxamide derivative is represented by the following general formula (1):
(Example: 2-ethyl-7-methoxypyrazolo[1,5-a]pyridine-4-carboxylic acid (3,5-dichloropyridin-4-yl)amide).
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