发明公开
- 专利标题： INDOLES WHICH ACT AS VIA RECEPTOR ANTAGONISTS
- 专利标题（中）： 威盛受体拮抗剂适合...吲哚
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申请号： EP07847501.9申请日： 2007-11-29
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公开(公告)号： EP2089381A1公开(公告)日： 2009-08-19
- 发明人: BISSANTZ, Caterina , GRUNDSCHOBER, Christophe , MASCIADRI, Raffaello , RATNI, Hasane , ROGERS-EVANS, Mark , SCHNIDER, Patrick
- 申请人： F.HOFFMANN-LA ROCHE AG
- 申请人地址： Grenzacherstrasse 124 4070 Basel CH
- 专利权人： F.HOFFMANN-LA ROCHE AG
- 当前专利权人： F.HOFFMANN-LA ROCHE AG
- 当前专利权人地址： Grenzacherstrasse 124 4070 Basel CH
- 代理机构： Wasner, Marita
- 优先权： EP06125663 20061208
- 国际公布： WO2008068184 20080612
- 主分类号： C07D401/14
- IPC分类号： C07D401/14 ; C07D491/04 ; A61K31/4427 ; A61P25/22 ; A61P25/24
摘要：
The present invention is concerned with novel indol-2-yl-carbonyl-piperidin- benzoimidazolon and indol-2-yl-carbonyl-piperidin-benzoxazolon derivatives as V1a receptor antagonists, their manufacture, pharmaceutical compositions containing them and their use as medicaments. The active compounds of the present invention are useful in the prevention and/or treatment of anxiety and depressive disorders and other diseases. Present invention comprises compounds of the general formula (I) wherein R1 to R11, X and Y are as defined in the specification.
公开/授权文献
- EP2089381B1 INDOLES WHICH ACT AS VIA RECEPTOR ANTAGONISTS 公开/授权日：2010-06-30
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