发明公开
EP2102170A2 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
审中-公开
糖皮质激素模拟物，其制备方法，药物组合物及其用途
- 专利标题： GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
- 专利标题（中）： 糖皮质激素模拟物，其制备方法，药物组合物及其用途
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申请号： EP07864855.7申请日： 2007-11-29
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公开(公告)号： EP2102170A2公开(公告)日： 2009-09-23
- 发明人: KUZMICH, Daniel , DISALVO, Darren , RAZAVI, Hossein , BURKE, Michael Jason
- 申请人： Boehringer Ingelheim International GmbH , Boehringer Ingelheim Pharma GmbH & Co. KG
- 申请人地址： Binger Strasse 173 55216 Ingelheim DE
- 专利权人： Boehringer Ingelheim International GmbH,Boehringer Ingelheim Pharma GmbH & Co. KG
- 当前专利权人： Boehringer Ingelheim International GmbH,Boehringer Ingelheim Pharma GmbH & Co. KG
- 当前专利权人地址： Binger Strasse 173 55216 Ingelheim DE
- 代理机构： Zwickl, Markus
- 优先权： US868844P 20061206
- 国际公布： WO2008070507 20080612
- 主分类号： C07D231/56
- IPC分类号： C07D231/56 ; C07D401/14 ; C07D403/04 ; C07D403/06 ; C07D409/06 ; C07D417/06 ; C07D471/04 ; C07D487/04 ; C07D498/04 ; C07D519/00 ; A61K31/437 ; A61K31/416 ; A61P5/44 ; A61P5/46
摘要：
Compounds of Formula (IA), and Formula (IB), wherein R1, R2, R3, A, B, C, D, E, G, X, Y, and Z are as defined herein, or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.
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