发明公开
EP2161260A1 Semisynthesis process for the preparation of 10 deacetyl-n-debenzoyl-paclitaxel
有权
Semisyntheseverfahren zur Herstellung von 10-Deacetyl-n-Debenzoyl-Paclitaxel
- 专利标题： Semisynthesis process for the preparation of 10 deacetyl-n-debenzoyl-paclitaxel
- 专利标题（中）： Semisyntheseverfahren zur Herstellung von 10-Deacetyl-n-Debenzoyl-Paclitaxel
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申请号： EP09175976.1申请日： 2005-10-07
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公开(公告)号： EP2161260A1公开(公告)日： 2010-03-10
- 发明人: Bombardelli, Ezio , Gabetta, Bruno , Gambini, Andrea , Fontana, Gabriele
- 申请人： INDENA S.p.A.
- 申请人地址： Viale Ortles, 12 20139 Milano IT
- 专利权人： INDENA S.p.A.
- 当前专利权人： INDENA S.p.A.
- 当前专利权人地址： Viale Ortles, 12 20139 Milano IT
- 代理机构： Minoja, Fabrizio
- 优先权： US616840P 20041008; EP04425752 20041008; EP05007888 20050411
- 主分类号： C07D305/14
- IPC分类号： C07D305/14
摘要：
The invention relates to a process for the preparation of 10-deacetyl-N-debenzoyl-paclitaxel ( I )
a synthon useful for the preparation of taxanes with antitumour activity, and intermediates for the preparation thereof.
The invention also discloses a process for the preparation of Docetaxel starting from said compound of formula (I).
a synthon useful for the preparation of taxanes with antitumour activity, and intermediates for the preparation thereof.
The invention also discloses a process for the preparation of Docetaxel starting from said compound of formula (I).
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