发明公开
- 专利标题： DIPEPTOID-PRODRUGS UND IHRE VERWENDUNG
- 专利标题（英）： Dipeptoid prodrugs and the use thereof
- 专利标题（中）： Dipeptoid前药和它们的用途
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申请号： EP09764200.3申请日： 2009-12-03
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公开(公告)号： EP2379540A1公开(公告)日： 2011-10-26
- 发明人: LERCHEN, Hans-Georg , MEIBOM, Daniel , VAKALOPOULOS, Alexandros , ALBRECHT-KÜPPER, Barbara , KELDENICH, Jörg , ZIMMERMANN, Katja , NELL, Peter , KRENZ, Ursula
- 申请人： Bayer Pharma Aktiengesellschaft
- 申请人地址： Müllerstrasse 178 13353 Berlin DE
- 专利权人： Bayer Pharma Aktiengesellschaft
- 当前专利权人： Bayer Pharma Aktiengesellschaft
- 当前专利权人地址： Müllerstrasse 178 13353 Berlin DE
- 优先权： DE102008062567 20081216
- 国际公布： WO2010072314 20100701
- 主分类号： C07D413/12
- IPC分类号： C07D413/12 ; A61K31/4439 ; C07K5/062 ; C07K5/065 ; C07K5/068 ; C07K5/072 ; C07K5/078
摘要：
The invention relates to dipeptide-like prodrug derivates of the formula (I), where R
PD is a group of the formula (Ia), (Ib), (Ic) or (Id), wherein # means the linking site to each O atom, to a method for the production thereof, to the use thereof for treating and/or preventing illnesses, and to the use thereof for producing pharmaceuticals for treating and/or preventing illnesses, particularly cardiovascular diseases.
PD is a group of the formula (Ia), (Ib), (Ic) or (Id), wherein # means the linking site to each O atom, to a method for the production thereof, to the use thereof for treating and/or preventing illnesses, and to the use thereof for producing pharmaceuticals for treating and/or preventing illnesses, particularly cardiovascular diseases.
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