发明公开
EP2386546A1 NOVEL PYRAZOLE-3-CARBOXAMIDE DERIVATE HAVING 5-HT2B RECEPTOR ANTAGONIST ACTIVITY
有权
具有5-HT2B受体拮抗剂活性的新型吡唑-3-甲酰胺衍生物
- 专利标题： NOVEL PYRAZOLE-3-CARBOXAMIDE DERIVATE HAVING 5-HT2B RECEPTOR ANTAGONIST ACTIVITY
- 专利标题（中）： 具有5-HT2B受体拮抗剂活性的新型吡唑-3-甲酰胺衍生物
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申请号： EP09827639.7申请日： 2009-11-24
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公开(公告)号： EP2386546A1公开(公告)日： 2011-11-16
- 发明人: YAMAGISHI, Tatsuya , KAWAMURA, Kiyoshi , INOUE, Tadashi , SHISHIDO, Yuji , ITO, Hiroaki
- 申请人： RaQualia Pharma Inc
- 申请人地址： 2, Aza 5-gochi Taketoyo-cho Chita-gun Aichi-ken 470 2341 JP
- 专利权人： RaQualia Pharma Inc
- 当前专利权人： RaQualia Pharma Inc
- 当前专利权人地址： 2, Aza 5-gochi Taketoyo-cho Chita-gun Aichi-ken 470 2341 JP
- 代理机构： Kalhammer, Georg
- 优先权： JP2008298821 20081121; JP2009112344 20090501
- 国际公布： WO2010058858 20100527
- 主分类号： C07D231/14
- IPC分类号： C07D231/14 ; A61K31/415 ; A61K31/4155 ; A61K31/437 ; A61K31/454 ; A61K31/5377 ; A61K31/553 ; A61P1/00 ; A61P1/04 ; A61P1/10 ; A61P1/12 ; A61P1/16 ; A61P3/04 ; A61P9/00 ; A61P9/10 ; A61P11/00 ; A61P11/06 ; A61P13/12 ; A61P17/00 ; A61P19/02 ; A61P25/02
摘要：
Disclosed is a compound represented by general formula (I) or a pharmaceutically acceptable salt thereof, which is useful as a selective antagonist of a 5-HT2 B receptor. The compound and salt are useful for treatment or prevention of various diseases and conditions associated with a 5-HT2 B receptor.
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