发明公开
- 专利标题: ANTIBACTERIAL OXADIAZOLONE DERIVATIVES
- 专利标题(中): 抗菌剂奥沙西唑衍生物
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申请号: EP14701232.2申请日: 2014-01-08
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公开(公告)号: EP2943492A1公开(公告)日: 2015-11-18
- 发明人: HUBSCHWERLEN, Christian , RUEEDI, Georg , ZUMBRUNN, Cornelia
- 申请人: Actelion Pharmaceuticals Ltd.
- 申请人地址: Gewerbestrasse 16 4123 Allschwil CH
- 专利权人: Actelion Pharmaceuticals Ltd.
- 当前专利权人: Actelion Pharmaceuticals Ltd.
- 当前专利权人地址: Gewerbestrasse 16 4123 Allschwil CH
- 代理机构: Ruhlmann, Eric
- 优先权: EP13150707 20130109; EP13159274 20130314
- 国际公布: WO2014108836 20140717
- 主分类号: C07D471/06
- IPC分类号: C07D471/06 ; C07D471/16 ; C07D487/06 ; C07D519/00 ; A61K31/437 ; A61K31/4375 ; A61K31/4985 ; A61K31/536 ; A61P31/04
摘要:
The invention relates to antibacterial compounds of formula I wherein U represents CH or N; V represents CH or N, provided that at least one of U and V does not represent N; R represents H, halogen, methyl, methoxy, cyano or ethynyl; either W represents a phenyl group substituted in para position with (C1-C3)alkyl, (C1-C3)alkoxy or (C1-C3)thioalkoxy and optionally in meta position with halogen, or W is a group having one of the formulae W1 and W2 below wherein Q is O or S and X is CH or N; and salts of such compounds.
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