发明公开
EP3319940A1 NEW INDOLE COMPOUNDS HAVING ANTIPROTOZOAL ACTIVITY AND ITS USE AS WELL AS METHODS FOR PRODUCING THE SAME
审中-公开
具有抗原活性的新吲哚化合物及其用途以及生产相同物质的方法
- 专利标题： NEW INDOLE COMPOUNDS HAVING ANTIPROTOZOAL ACTIVITY AND ITS USE AS WELL AS METHODS FOR PRODUCING THE SAME
- 专利标题（中）： 具有抗原活性的新吲哚化合物及其用途以及生产相同物质的方法
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申请号： EP15736269.0申请日： 2015-07-10
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公开(公告)号： EP3319940A1公开(公告)日： 2018-05-16
- 发明人: KUNICK, Conrad , LANDE, Hoang , GRUENEFELD, Johann , DZIKOWSKI, Ron , NASEREDDIN, Abed
- 申请人： Technische Universität Braunschweig , Yissum Research Development Company of the Hebrew University of Jerusalem Ltd.
- 申请人地址： Universitätsplatz 2 38106 Braunschweig DE
- 专利权人： Technische Universität Braunschweig,Yissum Research Development Company of the Hebrew University of Jerusalem Ltd.
- 当前专利权人： Technische Universität Braunschweig,Yissum Research Development Company of the Hebrew University of Jerusalem Ltd.
- 当前专利权人地址： Universitätsplatz 2 38106 Braunschweig DE
- 代理机构： Gramm, Lins & Partner Patent- und Rechtsanwälte PartGmbB
- 国际公布： WO2017008826 20170119
- 主分类号： C07D209/12
- IPC分类号： C07D209/12
摘要：
In a first aspect, the present invention relates to new compounds as depicted in formula (I). In particular, compounds according to the present invention are bisindolylcyclobuten-dione-based structures having antiprotozoal activity. In a further aspect, pharmaceutical compositions containing the same are provided as well as the use of the compounds and pharmaceutical compositions for the prophylaxis and treatment of parasite based diseases including malaria. Finally, methods for the treatment of parasite diseases including malaria are provided.
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