- 专利标题： PHARMACEUTICAL COMPOSITION CONTAINING TRIAZINE DERIVATIVE
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申请号： EP22876159.9申请日： 2022-09-27
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公开(公告)号： EP4410292A1公开(公告)日： 2024-08-07
- 发明人: TACHIBANA Yuki , UEHARA Shota , UNOH Yuto , NAKAHARA Kenji , TAODA Yoshiyuki , KASAMATSU Koji , YAMATSU Yukiko , ANDO Shigeru , FUKAO Keita , NOBORI Haruaki , KURODA Takayuki , TOBA Shinsuke , UEMURA Kentaro , MARUYAMA Yuki , SASAKI Michihito , SAWA Hirofumi
- 申请人： Shionogi & Co., Ltd , National University Corporation Hokkaido University
- 申请人地址： JP Osaka-shi, Osaka 541-0045 1-8, Doshomachi 3-chome Chuo-ku
- 专利权人： Shionogi & Co., Ltd,National University Corporation Hokkaido University
- 当前专利权人： Shionogi & Co., Ltd,National University Corporation Hokkaido University
- 当前专利权人地址： JP Osaka-shi, Osaka 541-0045 1-8, Doshomachi 3-chome Chuo-ku
- 代理机构： Vossius & Partner Patentanwälte Rechtsanwälte mbB
- 优先权： JP 21157929 2021.09.28
- 国际申请： JP2022035803 2022.09.27
- 国际公布： WO2023054292 2023.04.06
- 主分类号： A61K31/5355
- IPC分类号： A61K31/5355 ; A61K31/53 ; A61K31/5377 ; A61P31/12 ; A61P31/14 ; A61P43/00
摘要：
The present invention provides a pharmaceutical composition comprising a compound exhibiting coronavirus proliferation inhibitory activity.
A pharmaceutical composition comprising a compound represented by the formula: wherein Y is N; R1 is substituted or unsubstituted aromatic heterocyclyl; R2 is substituted or unsubstituted 6-membered aromatic carbocyclyl; R3 is substituted or unsubstituted aromatic heterocyclyl; -X- is -NH-; m is 0 or 1; R5a is a hydrogen atom; R5b is a hydrogen atom; n is 1; R4a is a hydrogen atom; and R4b is a hydrogen atom, or a pharmaceutically acceptable salt thereof.
A pharmaceutical composition comprising a compound represented by the formula: wherein Y is N; R1 is substituted or unsubstituted aromatic heterocyclyl; R2 is substituted or unsubstituted 6-membered aromatic carbocyclyl; R3 is substituted or unsubstituted aromatic heterocyclyl; -X- is -NH-; m is 0 or 1; R5a is a hydrogen atom; R5b is a hydrogen atom; n is 1; R4a is a hydrogen atom; and R4b is a hydrogen atom, or a pharmaceutically acceptable salt thereof.
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