Invention Grant
- Patent Title: Methods for preparing fused bicyclic 2, 4-diaminopyrimidine derivatives
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Application No.: US15537954Application Date: 2015-12-23
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Publication No.: US10259794B2Publication Date: 2019-04-16
- Inventor: Shawn P. Allwein , Roger P. Bakale , Dale R. Mowrey , Daniel E. Petrillo , Sander Kluwer
- Applicant: CEPHALON, INC.
- Applicant Address: US PA Frazer
- Assignee: CEPHALON, INC.
- Current Assignee: CEPHALON, INC.
- Current Assignee Address: US PA Frazer
- Agency: Sterne, Kessler, Goldstein & Fox P.L.L.C.
- International Application: PCT/US2015/000301 WO 20151223
- International Announcement: WO2016/105529 WO 20160630
- Main IPC: C07D241/04
- IPC: C07D241/04 ; C07D295/135 ; C07D403/12 ; A61K31/495

Abstract:
The present disclosure is directed to improved methods useful for the preparation of, for example, 2-[[5-chloro-2-[[(6S)-6-[4-(2-hydroxyethyl)piperazin-1-yl]-1-methoxy-6,7,8,9-tetrahydro-5Hbenzo[7]annulen-2-yl]amino]pyrimidin-4-yl]amino]-N-methyl-benzamide (CEP-37440).
Public/Granted literature
- US20170369451A1 METHODS FOR PREPARING FUSED BICYCLIC 2, 4-DIAMINOPYRIMIDINE DERIVATIVES Public/Granted day:2017-12-28
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