Invention Grant
- Patent Title: Aminotriazolopyridines as kinase inhibitors
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Application No.: US16484604Application Date: 2018-02-12
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Publication No.: US10913738B2Publication Date: 2021-02-09
- Inventor: Junqing Guo , Amy C. Hart , John E. Macor , Michael E. Mertzman , William J. Pitts , Steven H. Spergel , Scott Hunter Watterson , Murugaiah Andappan Murugaiah Subbaiah , Jie Chen , Carolyn Diane Dzierba , Guanglin Luo , Jianliang Shi , Sing-Yuen Sit
- Applicant: BRISTOL-MYERS SQUIBB COMPANY
- Applicant Address: US NJ Princeton
- Assignee: BRISTOL-MYERS SQUIBB COMPANY
- Current Assignee: BRISTOL-MYERS SQUIBB COMPANY
- Current Assignee Address: US NJ Princeton
- Agent Mary K. VanAtten
- International Application: PCT/US2018/017755 WO 20180212
- International Announcement: WO2018/148626 WO 20180816
- Main IPC: C07D471/04
- IPC: C07D471/04 ; A61P29/00 ; A61P19/02 ; A61P17/06 ; A61P1/00

Abstract:
Compounds having formula (I) (IX), and enantiomers, and diastereomers, stereoisomers, pharmaceutically acceptable salts and prodrugs thereof, are useful as kinase modulators, including RIPK1 modulation. All the variables are as defined herein: (I), (II), (III), (IV), (V), (VI), (VII), (VIII), (IX).
Public/Granted literature
- US20190389859A1 AMINOTRIAZOLOPYRIDINES AS KINASE INHIBITORS Public/Granted day:2019-12-26
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