发明申请
US20040214812A1 4-Substituted or unsubstituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid derivatives as beta-lactamase inhibitors
失效
4-取代或未取代的7-氢-1,4-硫杂氮杂-7- [双环或三环杂芳基]取代-3,6-二羧酸衍生物作为β-内酰胺酶抑制剂
![4-Substituted or unsubstituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid derivatives as beta-lactamase inhibitors](/docs/US/2004-10-28/US20040214812A1/abs.jpg.600x600.jpg)
- 专利标题： 4-Substituted or unsubstituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid derivatives as beta-lactamase inhibitors
- 专利标题（中）： 4-取代或未取代的7-氢-1,4-硫杂氮杂-7- [双环或三环杂芳基]取代-3,6-二羧酸衍生物作为β-内酰胺酶抑制剂
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申请号： US10834301申请日： 2004-04-28
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公开(公告)号： US20040214812A1公开(公告)日： 2004-10-28
- 发明人: Tarek Suhayl Mansour , Aranapakam Mudumbai Venkatesan
- 申请人： Wyeth Holdings Corporation
- 申请人地址： US NJ Madison
- 专利权人： Wyeth Holdings Corporation
- 当前专利权人： Wyeth Holdings Corporation
- 当前专利权人地址： US NJ Madison
- 主分类号： A61K031/554
- IPC分类号： A61K031/554 ; C07D417/02
![4-Substituted or unsubstituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid derivatives as beta-lactamase inhibitors](/abs-image/US/2004/10/28/US20040214812A1/abs.jpg.150x150.jpg)
摘要：
The present invention relates to novel, low molecular weight broad spectrum compounds in particular to a class of 4-substituted or unsubstituted-7-hydro-1,4-thiazepine-7-nullbicyclic or tricyclic heteroarylnull substituted-3,6-dicarboxylic acid or their derivatives which have null-lactamase inhibitory and antibacterial properties. The compounds are therefore useful in the treatment of antibacterial infections in humans or animals, either alone or in combination with other antibiotics.
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