发明申请
US20050004043A1 Succinoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
失效
用作逆转录病毒蛋白酶抑制剂的琥珀酰氨基羟乙基氨基磺酰胺
- 专利标题: Succinoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
- 专利标题(中): 用作逆转录病毒蛋白酶抑制剂的琥珀酰氨基羟乙基氨基磺酰胺
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申请号: US10784916申请日: 2004-02-24
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公开(公告)号: US20050004043A1公开(公告)日: 2005-01-06
- 发明人: Michael Vazquez , Richard Mueller , John Talley , Daniel Getman , Gary DeCrescenzo , John Freskos
- 申请人: Michael Vazquez , Richard Mueller , John Talley , Daniel Getman , Gary DeCrescenzo , John Freskos
- 申请人地址: US IL Chicago
- 专利权人: G.D. Searle & Co.
- 当前专利权人: G.D. Searle & Co.
- 当前专利权人地址: US IL Chicago
- 主分类号: A61K31/145
- IPC分类号: A61K31/145 ; A61K38/04 ; C07C307/02 ; C07C311/06 ; C07C311/19 ; C07C327/02 ; C07D233/54 ; C07D233/64 ; C07K5/04
摘要:
Succinoylamino hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.