发明申请
- 专利标题: Pharmaceutical compositions containing sulphonic acid derivatives
- 专利标题(中): 含有磺酸衍生物的药物组合物
-
申请号: US10549221申请日: 2004-03-05
-
公开(公告)号: US20060160849A1公开(公告)日: 2006-07-20
- 发明人: Beatriz Banfi Tosi , Guillermo Gimenez Gallego , Serafin Valverde Lopez , Rosa Lozano Puerto , Pedro Sanchez Cuevas
- 申请人: Beatriz Banfi Tosi , Guillermo Gimenez Gallego , Serafin Valverde Lopez , Rosa Lozano Puerto , Pedro Sanchez Cuevas
- 优先权: ESP200300563 20030307
- 国际申请: PCT/ES04/00104 WO 20040305
- 主分类号: A61K31/47
- IPC分类号: A61K31/47 ; A61K31/185
摘要:
A naphthalenesulfonic acid or quinolinesulfonic acid of formula (I), wherein A is N or a CR8 formula group, where R8 is H, OH, NR10R11, independently from one another, where R10 and R11 represent H or C1-C6 alkyl or a group of formula NH—CO—R12, where R12 is C1-C6 alkyl or C6-C10 aryl; R1 and R2 represent H or SO3R9, independently from one another, where R9 is H, ammonium or a cation of an alkali or alkaline-earth metal; R3 is H or OH; and R4, R5, R6 and R7 represent H, an NR10R11 or NH—CO—R12 group, independently from one another; on the condition that (i) at least one of R1 or R2 is SO3R9, and (ii) at least one of R4, R5, R6 or R7 is an NR10R11 or NH—CO—R12 group, or their pharmaceutically acceptable salts; and a pharmaceutically acceptable excipient.
信息查询